FR2416901B1 - - Google Patents

Info

Publication number
FR2416901B1
FR2416901B1 FR7903452A FR7903452A FR2416901B1 FR 2416901 B1 FR2416901 B1 FR 2416901B1 FR 7903452 A FR7903452 A FR 7903452A FR 7903452 A FR7903452 A FR 7903452A FR 2416901 B1 FR2416901 B1 FR 2416901B1
Authority
FR
France
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
FR7903452A
Other languages
French (fr)
Other versions
FR2416901A1 (fr
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
F Hoffmann La Roche AG
Original Assignee
F Hoffmann La Roche AG
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by F Hoffmann La Roche AG filed Critical F Hoffmann La Roche AG
Publication of FR2416901A1 publication Critical patent/FR2416901A1/fr
Application granted granted Critical
Publication of FR2416901B1 publication Critical patent/FR2416901B1/fr
Granted legal-status Critical Current

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07HSUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H15/00Compounds containing hydrocarbon or substituted hydrocarbon radicals directly attached to hetero atoms of saccharide radicals
    • C07H15/20Carbocyclic rings
    • C07H15/22Cyclohexane rings, substituted by nitrogen atoms
    • CCHEMISTRY; METALLURGY
    • C12BIOCHEMISTRY; BEER; SPIRITS; WINE; VINEGAR; MICROBIOLOGY; ENZYMOLOGY; MUTATION OR GENETIC ENGINEERING
    • C12NMICROORGANISMS OR ENZYMES; COMPOSITIONS THEREOF; PROPAGATING, PRESERVING, OR MAINTAINING MICROORGANISMS; MUTATION OR GENETIC ENGINEERING; CULTURE MEDIA
    • C12N9/00Enzymes; Proenzymes; Compositions thereof; Processes for preparing, activating, inhibiting, separating or purifying enzymes
    • C12N9/99Enzyme inactivation by chemical treatment
    • CCHEMISTRY; METALLURGY
    • C12BIOCHEMISTRY; BEER; SPIRITS; WINE; VINEGAR; MICROBIOLOGY; ENZYMOLOGY; MUTATION OR GENETIC ENGINEERING
    • C12PFERMENTATION OR ENZYME-USING PROCESSES TO SYNTHESISE A DESIRED CHEMICAL COMPOUND OR COMPOSITION OR TO SEPARATE OPTICAL ISOMERS FROM A RACEMIC MIXTURE
    • C12P19/00Preparation of compounds containing saccharide radicals
    • C12P19/26Preparation of nitrogen-containing carbohydrates

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Wood Science & Technology (AREA)
  • Zoology (AREA)
  • Genetics & Genomics (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • General Health & Medical Sciences (AREA)
  • Biotechnology (AREA)
  • Molecular Biology (AREA)
  • Biochemistry (AREA)
  • Microbiology (AREA)
  • General Engineering & Computer Science (AREA)
  • General Chemical & Material Sciences (AREA)
  • Biomedical Technology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Medicinal Chemistry (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Peptides Or Proteins (AREA)
  • Enzymes And Modification Thereof (AREA)
  • Saccharide Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
FR7903452A 1978-02-14 1979-02-12 Derives amines de sucre utiles notamment comme medicaments Granted FR2416901A1 (fr)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB583478 1978-02-14

Publications (2)

Publication Number Publication Date
FR2416901A1 FR2416901A1 (fr) 1979-09-07
FR2416901B1 true FR2416901B1 (enrdf_load_stackoverflow) 1980-10-24

Family

ID=9803510

Family Applications (1)

Application Number Title Priority Date Filing Date
FR7903452A Granted FR2416901A1 (fr) 1978-02-14 1979-02-12 Derives amines de sucre utiles notamment comme medicaments

Country Status (26)

Country Link
US (1) US4273765A (enrdf_load_stackoverflow)
EP (1) EP0003616B1 (enrdf_load_stackoverflow)
JP (1) JPS54163511A (enrdf_load_stackoverflow)
AR (1) AR219150A1 (enrdf_load_stackoverflow)
AT (1) AT367451B (enrdf_load_stackoverflow)
AU (1) AU527318B2 (enrdf_load_stackoverflow)
CA (1) CA1121290A (enrdf_load_stackoverflow)
DE (2) DE2905649A1 (enrdf_load_stackoverflow)
DK (1) DK149599C (enrdf_load_stackoverflow)
ES (1) ES477653A1 (enrdf_load_stackoverflow)
FI (1) FI63062C (enrdf_load_stackoverflow)
FR (1) FR2416901A1 (enrdf_load_stackoverflow)
GR (1) GR72817B (enrdf_load_stackoverflow)
HU (1) HU181442B (enrdf_load_stackoverflow)
IE (1) IE47916B1 (enrdf_load_stackoverflow)
IL (1) IL56626A0 (enrdf_load_stackoverflow)
LU (1) LU80906A1 (enrdf_load_stackoverflow)
MC (1) MC1253A1 (enrdf_load_stackoverflow)
NL (1) NL7901182A (enrdf_load_stackoverflow)
NO (1) NO153011C (enrdf_load_stackoverflow)
NZ (1) NZ189625A (enrdf_load_stackoverflow)
PH (1) PH15084A (enrdf_load_stackoverflow)
PT (1) PT69218A (enrdf_load_stackoverflow)
SE (1) SE7901276L (enrdf_load_stackoverflow)
YU (1) YU41437B (enrdf_load_stackoverflow)
ZA (1) ZA79528B (enrdf_load_stackoverflow)

Families Citing this family (37)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE3166093D1 (en) 1981-01-05 1984-10-18 Takeda Chemical Industries Ltd N-substituted pseudo-aminosugars, their production and use
JPS57146713A (en) * 1981-03-09 1982-09-10 Akira Endo Hypoglycemic
US4595678A (en) * 1982-03-19 1986-06-17 Takeda Chemical Industries, Ltd. N-substituted pseudo-aminosugars and pharmaceutical compositions containing same
US4678812A (en) * 1986-05-30 1987-07-07 E. I. Du Pont De Nemours And Company Trehalose as stabilizer and tableting excipient
US4762857A (en) * 1986-05-30 1988-08-09 E. I. Du Pont De Nemours And Company Trehalose as stabilizer and tableting excipient
US4885361A (en) * 1987-07-31 1989-12-05 Hoffmann-La Roche Inc. Sulfated oligosaccharides
DK0559795T3 (da) * 1990-11-30 1996-01-29 Monoclonetics Int Fremgangsmåder til diagnosticering af kroniske smerter i lænderegionen og halshvrivelsøjlen
TW381025B (en) * 1993-08-05 2000-02-01 Hoffmann La Roche Pharmaceutical composition containing a glucosidase inhibitor and a lipase inhibitor
ATE343391T1 (de) * 2000-05-24 2006-11-15 Pfizer Behandlung von pansenacidose mit amylasehemmern
US7022684B2 (en) * 2000-05-24 2006-04-04 Pfizer Inc. Treatment of rumen acidosis with α-amylase inhibitors
CN1882327A (zh) 2003-11-19 2006-12-20 症变治疗公司 含磷的新的拟甲状腺素药
US7262318B2 (en) * 2004-03-10 2007-08-28 Pfizer, Inc. Substituted heteroaryl- and phenylsulfamoyl compounds
US20050288340A1 (en) * 2004-06-29 2005-12-29 Pfizer Inc Substituted heteroaryl- and phenylsulfamoyl compounds
BRPI0518300A2 (pt) * 2004-11-23 2008-11-11 Warner Lambert Co derivados de Ácido 7-(2h-pirazol-3-il)-3,5-diidràxi-heptanàico como inibidores da hmg co-a reductase para o tratamento de lipidemia
US7741317B2 (en) 2005-10-21 2010-06-22 Bristol-Myers Squibb Company LXR modulators
US7888376B2 (en) 2005-11-23 2011-02-15 Bristol-Myers Squibb Company Heterocyclic CETP inhibitors
JP5498168B2 (ja) 2006-12-01 2014-05-21 ブリストル−マイヤーズ スクイブ カンパニー アテローム性動脈硬化および循環器疾患の治療のためのcetp阻害剤としてのn−((3−ベンジル)−2,2−(ビス−フェニル)−プロパン−1−アミン誘導体
US8969514B2 (en) 2007-06-04 2015-03-03 Synergy Pharmaceuticals, Inc. Agonists of guanylate cyclase useful for the treatment of hypercholesterolemia, atherosclerosis, coronary heart disease, gallstone, obesity and other cardiovascular diseases
MX354786B (es) 2007-06-04 2018-03-21 Synergy Pharmaceuticals Inc Agonistas de guanilato ciclasa utiles para el tratamiento de trastornos gastrointestinales, inflamacion, cancer y otros trastornos.
WO2009125819A1 (ja) * 2008-04-11 2009-10-15 アステラス製薬株式会社 アミノ糖化合物及びその生産方法
CA2930674A1 (en) 2008-06-04 2009-12-10 Synergy Pharmaceuticals Inc. Agonists of guanylate cyclase useful for the treatment of gastrointestinal disorders, inflammation, cancer and other disorders
CA2730603C (en) 2008-07-16 2019-09-24 Synergy Pharmaceuticals Inc. Agonists of guanylate cyclase useful for the treatment of gastrointestinal disorders, inflammation, cancer and other disorders
US20120046364A1 (en) 2009-02-10 2012-02-23 Metabasis Therapeutics, Inc. Novel Sulfonic Acid-Containing Thyromimetics, and Methods for Their Use
CA2799708A1 (en) 2010-05-21 2011-11-24 Pfizer Inc. 2-phenyl benzoylamides
WO2012027331A1 (en) 2010-08-27 2012-03-01 Ironwood Pharmaceuticals, Inc. Compositions and methods for treating or preventing metabolic syndrome and related diseases and disorders
US9616097B2 (en) 2010-09-15 2017-04-11 Synergy Pharmaceuticals, Inc. Formulations of guanylate cyclase C agonists and methods of use
CA2828343A1 (en) 2011-03-04 2012-09-13 The Scripps Research Institute Edn3-like peptides and uses thereof
US20150050371A1 (en) 2012-03-09 2015-02-19 Biotropics Malaysia Berhad Extract Formulations of Rhodamnia Cinerea And Uses Thereof
AU2014235215A1 (en) 2013-03-15 2015-10-01 Synergy Pharmaceuticals Inc. Agonists of guanylate cyclase and their uses
JP2016514670A (ja) 2013-03-15 2016-05-23 シナジー ファーマシューティカルズ インコーポレイテッド 他の薬物と組み合わせたグアニル酸シクラーゼ受容体アゴニスト
AU2014255381A1 (en) 2013-04-17 2015-10-08 Pfizer Inc. N-piperidin-3-ylbenzamide derivatives for treating cardiovascular diseases
CN113388007A (zh) 2013-06-05 2021-09-14 博士医疗爱尔兰有限公司 鸟苷酸环化酶c的超纯激动剂、制备和使用所述激动剂的方法
MX389591B (es) 2014-08-29 2025-03-20 Tes Pharma S R L INHIBIDORES DE ACIDO A-AMINO-ß-CARBOXIMUCONICO SEMIALDEHIDO DESCARBOXILASA
WO2016055901A1 (en) 2014-10-08 2016-04-14 Pfizer Inc. Substituted amide compounds
AR109950A1 (es) 2016-10-14 2019-02-06 Tes Pharma S R L INHIBIDORES DE LA ÁCIDO a-AMINO-b-CARBOXIMUCÓNICO SEMIALDEHÍDO DESCARBOXILASA
CN113302189B (zh) 2018-11-20 2025-09-05 Tes制药有限责任公司 α-氨基-β-羧基己二烯二酸半醛去羧酶的抑制剂
KR20210116548A (ko) 2019-01-18 2021-09-27 아스트라제네카 아베 Pcsk9 억제제 및 이의 이용 방법

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE2064092C2 (de) * 1970-12-28 1983-06-01 Bayer Ag, 5090 Leverkusen Inhibitoren für Glykosidhydrolasen aus Actinomyceten
DE2347782C3 (de) * 1973-09-22 1979-10-11 Bayer Ag, 5090 Leverkusen Aminozuckerderivate, Verfahren zu ihrer Herstellung sowie diese Verbindungen enthaltende Arzneimittel
US4062950A (en) * 1973-09-22 1977-12-13 Bayer Aktiengesellschaft Amino sugar derivatives
US4065557A (en) * 1974-03-21 1977-12-27 Bayer Aktiengesellschaft Amino sugars and their use in improving the meat:fat ratio in animals
USRE29903E (en) 1975-03-19 1979-02-06 American Cyanamid Company Antibacterial antibiotics AM31α, AM31β and AM31γ
DE2614393C3 (de) * 1976-04-02 1980-04-03 Bayer Ag, 5090 Leverkusen Aminozucker-Derivate und diese Verbindungen enthaltende Arzneimittel

Also Published As

Publication number Publication date
DK61179A (da) 1979-08-15
EP0003616B1 (de) 1982-02-24
YU41437B (en) 1987-06-30
IE790274L (en) 1979-08-14
PT69218A (en) 1979-03-01
FI63062C (fi) 1983-04-11
SE7901276L (sv) 1979-08-15
JPS54163511A (en) 1979-12-26
EP0003616A3 (en) 1979-09-05
HU181442B (en) 1983-07-28
AU527318B2 (en) 1983-02-24
LU80906A1 (de) 1980-09-24
AT367451B (de) 1982-07-12
DE2962165D1 (en) 1982-03-25
AU4402879A (en) 1979-08-23
EP0003616A2 (de) 1979-08-22
PH15084A (en) 1982-07-02
US4273765A (en) 1981-06-16
CA1121290A (en) 1982-04-06
NL7901182A (nl) 1979-08-16
ZA79528B (en) 1980-02-27
MC1253A1 (fr) 1980-01-14
FR2416901A1 (fr) 1979-09-07
GR72817B (enrdf_load_stackoverflow) 1983-12-06
NZ189625A (en) 1981-05-01
ATA108879A (de) 1981-11-15
IL56626A0 (en) 1979-05-31
NO153011C (no) 1986-01-02
NO153011B (no) 1985-09-23
NO790469L (no) 1979-08-15
AR219150A1 (es) 1980-07-31
DK149599C (da) 1987-06-01
DE2905649A1 (de) 1979-08-16
FI790486A7 (fi) 1979-08-15
DK149599B (da) 1986-08-04
ES477653A1 (es) 1980-03-01
FI63062B (fi) 1982-12-31
IE47916B1 (en) 1984-07-25
JPS643877B2 (enrdf_load_stackoverflow) 1989-01-23
YU34879A (en) 1983-01-21

Similar Documents

Publication Publication Date Title
FR2416901B1 (enrdf_load_stackoverflow)
FR2414553B1 (enrdf_load_stackoverflow)
FR2414756B1 (enrdf_load_stackoverflow)
FR2414924B1 (enrdf_load_stackoverflow)
DE2800351C3 (enrdf_load_stackoverflow)
DE2954155A1 (enrdf_load_stackoverflow)
FR2416213B1 (enrdf_load_stackoverflow)
FR2415912B1 (enrdf_load_stackoverflow)
FR2415698B1 (enrdf_load_stackoverflow)
FR2416676B1 (enrdf_load_stackoverflow)
FR2414133B1 (enrdf_load_stackoverflow)
FR2416801B1 (enrdf_load_stackoverflow)
BG26015A1 (enrdf_load_stackoverflow)
BG25857A1 (enrdf_load_stackoverflow)
BG26546A1 (enrdf_load_stackoverflow)
BG26450A1 (enrdf_load_stackoverflow)
BG25875A1 (enrdf_load_stackoverflow)
BG26292A1 (enrdf_load_stackoverflow)
BG25843A1 (enrdf_load_stackoverflow)
BG25974A1 (enrdf_load_stackoverflow)
BG26267A1 (enrdf_load_stackoverflow)
BG26022A1 (enrdf_load_stackoverflow)
BG26017A1 (enrdf_load_stackoverflow)
BG26013A1 (enrdf_load_stackoverflow)
BG25874A1 (enrdf_load_stackoverflow)

Legal Events

Date Code Title Description
TP Transmission of property
ST Notification of lapse