FR2375167A1 - Derives de trifluoromethyl-3 benzene - Google Patents

Derives de trifluoromethyl-3 benzene

Info

Publication number
FR2375167A1
FR2375167A1 FR7639033A FR7639033A FR2375167A1 FR 2375167 A1 FR2375167 A1 FR 2375167A1 FR 7639033 A FR7639033 A FR 7639033A FR 7639033 A FR7639033 A FR 7639033A FR 2375167 A1 FR2375167 A1 FR 2375167A1
Authority
FR
France
Prior art keywords
alkyl
benzamide
cpds
esp
pyrrolidinyl
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
FR7639033A
Other languages
English (en)
Other versions
FR2375167B1 (fr
Inventor
Jean-Pierre Kaplan
Henry Najer
Bernard Michel Raizon
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Synthelabo SA
Original Assignee
Synthelabo SA
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Synthelabo SA filed Critical Synthelabo SA
Priority to FR7639033A priority Critical patent/FR2375167A1/fr
Priority to NO774402A priority patent/NO774402L/no
Priority to FI773911A priority patent/FI773911A/fi
Priority to IL53680A priority patent/IL53680A0/xx
Priority to NZ186075A priority patent/NZ186075A/xx
Priority to DE19772757406 priority patent/DE2757406A1/de
Priority to DK575877A priority patent/DK575877A/da
Priority to GB53570/77A priority patent/GB1556566A/en
Priority to SE7714659A priority patent/SE7714659L/xx
Priority to AU31921/77A priority patent/AU3192177A/en
Priority to ZA00777613A priority patent/ZA777613B/xx
Priority to NL7714301A priority patent/NL7714301A/xx
Priority to JP15630677A priority patent/JPS5382771A/ja
Priority to BE183809A priority patent/BE862281R/fr
Priority to LU78773A priority patent/LU78773A1/fr
Priority to ES465366A priority patent/ES465366A2/es
Priority to GR55032A priority patent/GR66082B/el
Publication of FR2375167A1 publication Critical patent/FR2375167A1/fr
Application granted granted Critical
Publication of FR2375167B1 publication Critical patent/FR2375167B1/fr
Granted legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C45/00—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds
    • C07C45/41—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by hydrogenolysis or reduction of carboxylic groups or functional derivatives thereof
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C17/00—Preparation of halogenated hydrocarbons
    • C07C17/093—Preparation of halogenated hydrocarbons by replacement by halogens
    • C07C17/16—Preparation of halogenated hydrocarbons by replacement by halogens of hydroxyl groups
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C205/00—Compounds containing nitro groups bound to a carbon skeleton
    • C07C205/07—Compounds containing nitro groups bound to a carbon skeleton the carbon skeleton being further substituted by halogen atoms
    • C07C205/11—Compounds containing nitro groups bound to a carbon skeleton the carbon skeleton being further substituted by halogen atoms having nitro groups bound to carbon atoms of six-membered aromatic rings
    • C07C205/12—Compounds containing nitro groups bound to a carbon skeleton the carbon skeleton being further substituted by halogen atoms having nitro groups bound to carbon atoms of six-membered aromatic rings the six-membered aromatic ring or a condensed ring system containing that ring being substituted by halogen atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C205/00—Compounds containing nitro groups bound to a carbon skeleton
    • C07C205/44—Compounds containing nitro groups bound to a carbon skeleton the carbon skeleton being further substituted by —CHO groups
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C45/00—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C45/00—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds
    • C07C45/45—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by condensation
    • C07C45/46—Friedel-Crafts reactions
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D207/00—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D207/02—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D207/04—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
    • C07D207/08—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon radicals, substituted by hetero atoms, attached to ring carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D207/00—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D207/02—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D207/04—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
    • C07D207/08—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon radicals, substituted by hetero atoms, attached to ring carbon atoms
    • C07D207/09—Radicals substituted by nitrogen atoms, not forming part of a nitro radical
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D207/00—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D207/02—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D207/18—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having one double bond between ring members or between a ring member and a non-ring member
    • C07D207/22—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having one double bond between ring members or between a ring member and a non-ring member with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D207/24—Oxygen or sulfur atoms
    • C07D207/26—2-Pyrrolidones
    • C07D207/273—2-Pyrrolidones with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to other ring carbon atoms
    • C07D207/277—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
    • C07D207/28—2-Pyrrolidone-5- carboxylic acids; Functional derivatives thereof, e.g. esters, nitriles

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Hydrogenated Pyridines (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

Dérivés de trifluorométhyl-3 benzène répondant à la formule :
FR7639033A 1976-12-24 1976-12-24 Derives de trifluoromethyl-3 benzene Granted FR2375167A1 (fr)

Priority Applications (17)

Application Number Priority Date Filing Date Title
FR7639033A FR2375167A1 (fr) 1976-12-24 1976-12-24 Derives de trifluoromethyl-3 benzene
NO774402A NO774402L (no) 1976-12-24 1977-12-21 R fremgangsmaate for fremstilling av metoksy-benzamidderivate
AU31921/77A AU3192177A (en) 1976-12-24 1977-12-22 2-methoxybenzamides
NZ186075A NZ186075A (en) 1976-12-24 1977-12-22 2-methoxybenzamide derivatives, and pharmaceutical compositions containing them
DE19772757406 DE2757406A1 (de) 1976-12-24 1977-12-22 2-methoxy-benzamidderivate, verfahren zu ihrer herstellung und sie enthaltende arzneimittel
DK575877A DK575877A (da) 1976-12-24 1977-12-22 Fremgangsmaade til fremstilling af 2-methoxybenzamider
GB53570/77A GB1556566A (en) 1976-12-24 1977-12-22 2-methoxybenzamides
SE7714659A SE7714659L (sv) 1976-12-24 1977-12-22 Metoxibensamider
FI773911A FI773911A (fi) 1976-12-24 1977-12-22 Metoxibenzamidderivat
ZA00777613A ZA777613B (en) 1976-12-24 1977-12-22 2-methoxybenzamides
IL53680A IL53680A0 (en) 1976-12-24 1977-12-22 Novel 2-methoxybenzamide derivatives their preparation and pharmaceutical compositions containing them
NL7714301A NL7714301A (nl) 1976-12-24 1977-12-23 Werkwijze voor het bereiden van een geneesmiddel, zo gevormd geneesmiddel.
JP15630677A JPS5382771A (en) 1976-12-24 1977-12-23 Methoxybenzamide derivative
BE183809A BE862281R (fr) 1976-12-24 1977-12-23 Derives de methoxy-2 benzamides
LU78773A LU78773A1 (fr) 1976-12-24 1977-12-23 Procede de preparation de methoxy-2-benzamides
ES465366A ES465366A2 (es) 1976-12-24 1977-12-23 Un procedimiento de preparacion de derivados de metoxi-2- benzamidas.
GR55032A GR66082B (fr) 1976-12-24 1977-12-27

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FR7639033A FR2375167A1 (fr) 1976-12-24 1976-12-24 Derives de trifluoromethyl-3 benzene

Publications (2)

Publication Number Publication Date
FR2375167A1 true FR2375167A1 (fr) 1978-07-21
FR2375167B1 FR2375167B1 (fr) 1980-04-30

Family

ID=9181519

Family Applications (1)

Application Number Title Priority Date Filing Date
FR7639033A Granted FR2375167A1 (fr) 1976-12-24 1976-12-24 Derives de trifluoromethyl-3 benzene

Country Status (3)

Country Link
BE (1) BE862281R (fr)
FR (1) FR2375167A1 (fr)
ZA (1) ZA777613B (fr)

Also Published As

Publication number Publication date
BE862281R (fr) 1978-06-23
ZA777613B (en) 1978-10-25
FR2375167B1 (fr) 1980-04-30

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Legal Events

Date Code Title Description
ST Notification of lapse