ES8203901A1 - Un procedimiento para la preparacion de benzamidas. - Google Patents
Un procedimiento para la preparacion de benzamidas.Info
- Publication number
- ES8203901A1 ES8203901A1 ES498945A ES498945A ES8203901A1 ES 8203901 A1 ES8203901 A1 ES 8203901A1 ES 498945 A ES498945 A ES 498945A ES 498945 A ES498945 A ES 498945A ES 8203901 A1 ES8203901 A1 ES 8203901A1
- Authority
- ES
- Spain
- Prior art keywords
- alkyl
- hydrogen
- phenyl
- active compounds
- pharmaceutically active
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
- C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
- C07D513/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/535—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one oxygen as the ring hetero atoms, e.g. 1,2-oxazines
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/54—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one sulfur as the ring hetero atoms, e.g. sulthiame
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/60—Salicylic acid; Derivatives thereof
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D265/00—Heterocyclic compounds containing six-membered rings having one nitrogen atom and one oxygen atom as the only ring hetero atoms
- C07D265/28—1,4-Oxazines; Hydrogenated 1,4-oxazines
- C07D265/30—1,4-Oxazines; Hydrogenated 1,4-oxazines not condensed with other rings
- C07D265/32—1,4-Oxazines; Hydrogenated 1,4-oxazines not condensed with other rings with oxygen atoms directly attached to ring carbon atoms
- C07D265/33—Two oxygen atoms, in positions 3 and 5
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D279/00—Heterocyclic compounds containing six-membered rings having one nitrogen atom and one sulfur atom as the only ring hetero atoms
- C07D279/10—1,4-Thiazines; Hydrogenated 1,4-thiazines
- C07D279/12—1,4-Thiazines; Hydrogenated 1,4-thiazines not condensed with other rings
Abstract
PROCEDIMIENTO PARA LA OBTENCION DE BENZAMIDAS, SUS N-OXIDOS Y SUS SALES FISIOLOGICAMENTE COMPATIBLES, DE FORMULA (I), EN AL R1 ES ALCOXI C1-6; R5 ES HIDROGENO O ALQUILO C1-4; X ES OXIGENO, AZUFRE O SULFOXIDO; P Y R VALEN 1 O 2, Y R2 R3 Y R4 PUEDEN SER VARIOS TIPOS DE RADICALES. CONSISTE EN LA REACCION DE UN COMPUESTO DE FORMULA (II) O UN DERIVADO REACTIVO DEL MISMO, CON UN COMPUESTO DE FORMULA (III), EN LAS QUE TODOS LOS SIMBOLOS TIENEN EL MISMO SIGNIFICADO QUE EN LA FORMULA (I). LA REACCION SE LLEVA A CABO EN UN DISOLVENTE INERTE Y, SI ES NECESARIO, EN PRESENCIA DE UN AGENTE ACEPTOR DE ACIDO.
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
GB8003154 | 1980-01-30 | ||
GB8028864 | 1980-09-06 |
Publications (2)
Publication Number | Publication Date |
---|---|
ES8203901A1 true ES8203901A1 (es) | 1982-04-16 |
ES498945A0 ES498945A0 (es) | 1982-04-16 |
Family
ID=26274343
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
ES498945A Granted ES498945A0 (es) | 1980-01-30 | 1981-01-29 | Un procedimiento para la preparacion de benzamidas. |
Country Status (9)
Country | Link |
---|---|
US (1) | US4346089A (es) |
EP (1) | EP0034015B1 (es) |
AU (1) | AU545186B2 (es) |
DE (1) | DE3174163D1 (es) |
DK (1) | DK40781A (es) |
ES (1) | ES498945A0 (es) |
GR (1) | GR75278B (es) |
IL (1) | IL61972A0 (es) |
MX (1) | MX6807E (es) |
Families Citing this family (8)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
FR2440946A2 (fr) * | 1978-01-20 | 1980-06-06 | Ile De France | Nouveaux benzamides heterocycliques substitues, leurs procedes de preparation et leur application comme modificateurs du comportement |
EP0057536A1 (en) * | 1981-01-26 | 1982-08-11 | Beecham Group Plc | Pharmaceutically active compounds |
CA1183847A (en) * | 1981-10-01 | 1985-03-12 | Georges Van Daele | N-(3-hydroxy-4-piperidinyl)benzamide derivatives |
GB8518236D0 (en) * | 1985-07-19 | 1985-08-29 | Beecham Group Plc | Compounds |
FR2676448B1 (fr) * | 1991-05-14 | 1995-01-20 | Adir | Nouveaux derives amidiques de 1-amino octahydropyrido [2,1-c] [1,4] oxazine, leurs procedes de preparation et les compositions pharmaceutiques qui les contiennent. |
US5508272A (en) * | 1993-06-15 | 1996-04-16 | Bristol-Myers Squibb Company | Compounds containing a fused bicycle ring and processes therefor |
US5616775A (en) * | 1994-05-05 | 1997-04-01 | Bristol-Myers Squibb Co. | Process for preparing homocystein analogs useful as intermediates for compounds containing a fused bicyclic ring |
US7342010B2 (en) * | 2004-11-15 | 2008-03-11 | Board Of Trustees Of Michigan State University | 2-thiaquinolizidines and process for the preparation thereof |
Family Cites Families (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
GB1593146A (en) * | 1976-11-05 | 1981-07-15 | Beecham Group Ltd | Octahydro-quinolizinyl benzamide derivatives |
GB1561023A (en) * | 1977-04-22 | 1980-02-13 | Beecham Group Ltd | 2-methoxy - 5 - chloro aniline derivatives |
-
1981
- 1981-01-23 IL IL61972A patent/IL61972A0/xx unknown
- 1981-01-28 AU AU66682/81A patent/AU545186B2/en not_active Ceased
- 1981-01-28 EP EP81300362A patent/EP0034015B1/en not_active Expired
- 1981-01-28 US US06/229,191 patent/US4346089A/en not_active Expired - Fee Related
- 1981-01-28 DE DE8181300362T patent/DE3174163D1/de not_active Expired
- 1981-01-29 ES ES498945A patent/ES498945A0/es active Granted
- 1981-01-29 DK DK40781A patent/DK40781A/da unknown
- 1981-01-29 GR GR63996A patent/GR75278B/el unknown
- 1981-01-29 MX MX819288U patent/MX6807E/es unknown
Also Published As
Publication number | Publication date |
---|---|
EP0034015A2 (en) | 1981-08-19 |
EP0034015A3 (en) | 1981-10-14 |
IL61972A0 (en) | 1981-02-27 |
DK40781A (da) | 1981-07-31 |
GR75278B (es) | 1984-07-13 |
AU6668281A (en) | 1981-08-06 |
MX6807E (es) | 1986-07-30 |
US4346089A (en) | 1982-08-24 |
EP0034015B1 (en) | 1986-03-26 |
ES498945A0 (es) | 1982-04-16 |
DE3174163D1 (en) | 1986-04-30 |
AU545186B2 (en) | 1985-07-04 |
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