FR2368490A1 - Nouveaux derives de l'acide clavulanique, leur preparation et compositions pharmaceutiques en contenant - Google Patents

Nouveaux derives de l'acide clavulanique, leur preparation et compositions pharmaceutiques en contenant

Info

Publication number
FR2368490A1
FR2368490A1 FR7732041A FR7732041A FR2368490A1 FR 2368490 A1 FR2368490 A1 FR 2368490A1 FR 7732041 A FR7732041 A FR 7732041A FR 7732041 A FR7732041 A FR 7732041A FR 2368490 A1 FR2368490 A1 FR 2368490A1
Authority
FR
France
Prior art keywords
beta
antibiotics
clavulanic acid
useful
lactamase inhibitors
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
FR7732041A
Other languages
English (en)
Other versions
FR2368490B1 (fr
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Laboratoire Glaxo Wellcome SA
Glaxo Laboratories Ltd
Original Assignee
Laboratoires Glaxo SA
Glaxo Laboratories Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from GB44145/76A external-priority patent/GB1594934A/en
Application filed by Laboratoires Glaxo SA, Glaxo Laboratories Ltd filed Critical Laboratoires Glaxo SA
Publication of FR2368490A1 publication Critical patent/FR2368490A1/fr
Application granted granted Critical
Publication of FR2368490B1 publication Critical patent/FR2368490B1/fr
Granted legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D503/00—Heterocyclic compounds containing 4-oxa-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. oxapenicillins, clavulanic acid derivatives; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Cephalosporin Compounds (AREA)

Abstract

L'invention concerne des dérivés de l'acide clavulamique. Les composés conformes à l'invention répondent à la formule de structure générale suivante :
FR7732041A 1976-10-25 1977-10-25 Nouveaux derives de l'acide clavulanique, leur preparation et compositions pharmaceutiques en contenant Granted FR2368490A1 (fr)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GB44145/76A GB1594934A (en) 1976-10-25 1976-10-25 Clavulanic acid derivatives
GB2267977 1977-05-30

Publications (2)

Publication Number Publication Date
FR2368490A1 true FR2368490A1 (fr) 1978-05-19
FR2368490B1 FR2368490B1 (fr) 1981-02-06

Family

ID=26256057

Family Applications (1)

Application Number Title Priority Date Filing Date
FR7732041A Granted FR2368490A1 (fr) 1976-10-25 1977-10-25 Nouveaux derives de l'acide clavulanique, leur preparation et compositions pharmaceutiques en contenant

Country Status (12)

Country Link
JP (1) JPS53116395A (fr)
AT (1) AT363181B (fr)
AU (1) AU517920B2 (fr)
DE (1) DE2747599A1 (fr)
DK (1) DK471577A (fr)
ES (1) ES463484A1 (fr)
FI (1) FI773157A (fr)
FR (1) FR2368490A1 (fr)
IT (1) IT1091113B (fr)
NL (1) NL7711640A (fr)
NZ (1) NZ185511A (fr)
SE (1) SE7711961L (fr)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DK330880A (da) * 1979-08-03 1981-02-04 Beecham Group Ltd Fremgangsmaade til fremstilling af clavulansyrederivater
US4343807A (en) 1979-09-27 1982-08-10 Beecham Group Limited Derivatives of clavulanic acid, a process for their preparation and their use
ZA805850B (en) 1979-09-27 1981-09-30 Beecham Group Ltd Derivatives of clavulanic acid, a process for their preparation and their use
EP0068609A1 (fr) * 1981-06-11 1983-01-05 Beecham Group Plc Dérivés de l'acide clavulanique, un procédé pour leur préparation et leur application
EP0068617A1 (fr) * 1981-06-12 1983-01-05 Beecham Group Plc Dérivés de l'acide clavulanique, un procédé pour leur préparation et leur application
GB8521516D0 (en) * 1985-08-29 1985-10-02 Beecham Group Plc Compounds

Citations (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2288520A1 (fr) * 1974-10-22 1976-05-21 Beecham Group Ltd Derives des azetidinones a activite antibacterienne

Family Cites Families (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB1501643A (en) * 1974-10-28 1978-02-22 Beecham Group Ltd Antibacterial substituted azetidinones
IE42370B1 (en) * 1974-12-18 1980-07-30 Beecham Group Ltd Isoclavulanic acid derivatives
PT64897B (en) * 1975-04-14 1977-08-18 Beecham Group Ltd Process for the preparation of novel antibacterial agents
GB1542405A (en) * 1975-04-15 1979-03-21 Beecham Group Ltd Clavulanic acid derivatives
GB1493197A (en) * 1975-07-04 1977-11-23 Beecham Group Ltd Amides of clavulanic acid
IL50080A (en) * 1975-07-29 1979-07-25 Beecham Group Ltd 4-oxa-1-azabicyclo(3.2.0)heptan-7-one-2-car boxylic acid derivatives and their preparation
AU503489B2 (en) * 1975-10-13 1979-09-06 Beecham Group Limited Substituted aminodeoxy clavulanic acid
GB1547169A (en) * 1975-10-13 1979-06-06 Beecham Group Ltd Clavulanic acid derivatives
GB1504426A (en) * 1975-10-13 1978-03-22 Beecham Group Ltd Clavulanic acid derivatives

Patent Citations (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2288520A1 (fr) * 1974-10-22 1976-05-21 Beecham Group Ltd Derives des azetidinones a activite antibacterienne

Also Published As

Publication number Publication date
SE7711961L (sv) 1978-06-15
FR2368490B1 (fr) 1981-02-06
IT1091113B (it) 1985-06-26
DE2747599A1 (de) 1978-04-27
DK471577A (da) 1978-04-26
FI773157A (fi) 1978-04-26
JPS53116395A (en) 1978-10-11
NZ185511A (en) 1980-12-19
AU3002177A (en) 1979-06-07
AT363181B (de) 1981-07-10
ES463484A1 (es) 1978-11-16
ATA758877A (de) 1980-12-15
NL7711640A (nl) 1978-04-27
AU517920B2 (en) 1981-09-03

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Legal Events

Date Code Title Description
TP Transmission of property
ST Notification of lapse