FR2366295A1 - Composes bactericides de la rifamycine - Google Patents
Composes bactericides de la rifamycineInfo
- Publication number
- FR2366295A1 FR2366295A1 FR7726221A FR7726221A FR2366295A1 FR 2366295 A1 FR2366295 A1 FR 2366295A1 FR 7726221 A FR7726221 A FR 7726221A FR 7726221 A FR7726221 A FR 7726221A FR 2366295 A1 FR2366295 A1 FR 2366295A1
- Authority
- FR
- France
- Prior art keywords
- rifamycin
- bactericidal compounds
- compounds
- bactericidal
- desoxo
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
- 230000000844 anti-bacterial effect Effects 0.000 title abstract 2
- HJYYPODYNSCCOU-ODRIEIDWSA-N rifamycin SV Chemical compound OC1=C(C(O)=C2C)C3=C(O)C=C1NC(=O)\C(C)=C/C=C/[C@H](C)[C@H](O)[C@@H](C)[C@@H](O)[C@@H](C)[C@H](OC(C)=O)[C@H](C)[C@@H](OC)\C=C\O[C@@]1(C)OC2=C3C1=O HJYYPODYNSCCOU-ODRIEIDWSA-N 0.000 title abstract 2
- 229930189077 Rifamycin Natural products 0.000 title 1
- 150000001875 compounds Chemical class 0.000 title 1
- 229960003292 rifamycin Drugs 0.000 title 1
- BTVYFIMKUHNOBZ-ZDHWWVNNSA-N Rifamycin S Natural products COC1C=COC2(C)Oc3c(C)c(O)c4C(=O)C(=CC(=O)c4c3C2=O)NC(=O)C(=C/C=C/C(C)C(O)C(C)C(O)C(C)C(OC(=O)C)C1C)C BTVYFIMKUHNOBZ-ZDHWWVNNSA-N 0.000 abstract 1
- 125000002485 formyl group Chemical class [H]C(*)=O 0.000 abstract 1
- 239000000843 powder Substances 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D498/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D498/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
- C07D498/08—Bridged systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
- A61P31/06—Antibacterial agents for tuberculosis
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D498/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D498/12—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms in which the condensed system contains three hetero rings
- C07D498/18—Bridged systems
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Pharmacology & Pharmacy (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Communicable Diseases (AREA)
- Veterinary Medicine (AREA)
- Oncology (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Pulmonology (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| IT520976 | 1976-09-30 |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| FR2366295A1 true FR2366295A1 (fr) | 1978-04-28 |
| FR2366295B1 FR2366295B1 (OSRAM) | 1982-11-19 |
Family
ID=11119379
Family Applications (3)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| FR7726221A Granted FR2366295A1 (fr) | 1976-09-30 | 1977-08-29 | Composes bactericides de la rifamycine |
| FR7726223A Granted FR2366294A1 (fr) | 1976-09-30 | 1977-08-29 | Composes de la rifamycine ayant une activite anti-bacterienne |
| FR7726222A Granted FR2366296A1 (fr) | 1976-09-30 | 1977-08-29 | Composes antibiotiques de rifamycine |
Family Applications After (2)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| FR7726223A Granted FR2366294A1 (fr) | 1976-09-30 | 1977-08-29 | Composes de la rifamycine ayant une activite anti-bacterienne |
| FR7726222A Granted FR2366296A1 (fr) | 1976-09-30 | 1977-08-29 | Composes antibiotiques de rifamycine |
Country Status (12)
| Country | Link |
|---|---|
| US (3) | US4164499A (OSRAM) |
| JP (3) | JPS5350200A (OSRAM) |
| AT (2) | AT352279B (OSRAM) |
| CA (2) | CA1081218A (OSRAM) |
| CH (3) | CH629496A5 (OSRAM) |
| DE (3) | DE2739624A1 (OSRAM) |
| DK (2) | DK345977A (OSRAM) |
| ES (2) | ES462294A1 (OSRAM) |
| FR (3) | FR2366295A1 (OSRAM) |
| GB (3) | GB1550769A (OSRAM) |
| NL (2) | NL7710625A (OSRAM) |
| SE (2) | SE7708841L (OSRAM) |
Cited By (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| FR2426690A2 (fr) * | 1978-06-09 | 1979-12-21 | Archifar Lab Chim Farm | Composes de rifamycine |
Families Citing this family (12)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| BE886395A (fr) * | 1980-02-13 | 1981-03-16 | Erba Farmitalia | Derives de rifamycine |
| IT1154655B (it) * | 1980-05-22 | 1987-01-21 | Alfa Farmaceutici Spa | Derivati imidazo-rifamicinici metodi per la loro preparazione e loro uso come sostanza ad azione antibatterica |
| EP0049683A3 (de) * | 1980-09-25 | 1982-09-01 | Ciba-Geigy Ag | Imidazo-Rifamycine, Verfahren zu ihrer Herstellung, diese enthaltende pharmazeutische Präparate sowie ihre Verwendung |
| IT1201963B (it) * | 1983-03-24 | 1989-02-02 | Prodotti Antibiotici Spa | Derivati delle rifamicine e procedimento per la loro preparazione |
| US5362726A (en) * | 1993-02-12 | 1994-11-08 | Healthsearch, Inc. | Compound and method of treatment for falciparum malaria |
| US7122525B2 (en) * | 2001-11-21 | 2006-10-17 | Activbiotics, Inc. | Targeted therapeutics and uses thereof |
| PT102807A (pt) * | 2002-07-09 | 2004-01-30 | Inst Nac De Engenharia E Tecno | Derivados n-substituidos de rifabutina uteis como agentes antimicrobianos, processo para a sua preparacao e sua utilizacao como medicamentos |
| US7820652B2 (en) * | 2003-09-24 | 2010-10-26 | Activbiotics Pharma, Llc | Regimen for the administration of rifamycin-class antibiotics |
| US7265107B2 (en) * | 2004-03-10 | 2007-09-04 | Cumbre Pharmaceuticals Inc. | Rifamycin C-11 oxime cyclo derivatives effective against drug-resistant microbes |
| US7256187B2 (en) * | 2004-03-10 | 2007-08-14 | Cumbre Pharmaceuticals Inc. | Rifamycin C-11 oxime derivatives effective against drug-resistant microbes |
| US7678791B2 (en) * | 2006-07-12 | 2010-03-16 | Cumbre Ip Ventures, L.P. | Nitroheteroaryl-containing rifamycin derivatives |
| WO2009064792A1 (en) * | 2007-11-16 | 2009-05-22 | Cumbre Pharmaceuticals Inc. | Quinolone carboxylic acid-substituted rifamycin derivatives |
Family Cites Families (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CH512510A (de) * | 1965-08-24 | 1971-09-15 | Ciba Geigy Ag | Verfahren zur Herstellung von in 3-Stellung durch eine unsubstituierte oder substituierte Aminogruppe substituierten Derivaten von Rifamycin-S und Rifamycin-SV |
| CH536851A (de) * | 1966-10-25 | 1973-05-15 | Ciba Geigy Ag | Verfahren zur Herstellung neuer antibiotisch wirksamer Verbindungen der Rifamycinreihen |
| IT1048565B (it) * | 1975-05-15 | 1980-12-20 | Archifar Ind Chim Trentino | Amine aromatiche |
| IT1056271B (it) * | 1975-05-20 | 1982-01-30 | Archifar Ind Chim Trentino | Prodotti derivati dalle amine aromatiche |
| IT1056272B (it) * | 1975-06-13 | 1982-01-30 | Archifar Ind Chim Trentino | Prodotti derivati dalle amine aromatiche |
-
1977
- 1977-08-02 DK DK345977A patent/DK345977A/da unknown
- 1977-08-03 CH CH952877A patent/CH629496A5/it not_active IP Right Cessation
- 1977-08-03 SE SE7708841A patent/SE7708841L/xx unknown
- 1977-08-03 CH CH953077A patent/CH629498A5/it not_active IP Right Cessation
- 1977-08-03 CH CH952977A patent/CH629497A5/it not_active IP Right Cessation
- 1977-08-09 SE SE7709001A patent/SE7709001L/xx not_active Application Discontinuation
- 1977-08-09 GB GB33315/77A patent/GB1550769A/en not_active Expired
- 1977-08-09 GB GB33316/77A patent/GB1560265A/en not_active Expired
- 1977-08-11 DK DK357477A patent/DK357477A/da unknown
- 1977-08-12 US US05/825,165 patent/US4164499A/en not_active Expired - Lifetime
- 1977-08-12 US US05/825,163 patent/US4175077A/en not_active Expired - Lifetime
- 1977-08-12 US US05/825,166 patent/US4165317A/en not_active Expired - Lifetime
- 1977-08-15 CA CA284,850A patent/CA1081218A/en not_active Expired
- 1977-08-15 GB GB34102/77A patent/GB1557090A/en not_active Expired
- 1977-08-16 CA CA284,958A patent/CA1083144A/en not_active Expired
- 1977-08-29 FR FR7726221A patent/FR2366295A1/fr active Granted
- 1977-08-29 FR FR7726223A patent/FR2366294A1/fr active Granted
- 1977-08-29 FR FR7726222A patent/FR2366296A1/fr active Granted
- 1977-09-02 DE DE19772739624 patent/DE2739624A1/de not_active Withdrawn
- 1977-09-02 DE DE19772739623 patent/DE2739623A1/de not_active Withdrawn
- 1977-09-02 DE DE19772739671 patent/DE2739671A1/de not_active Withdrawn
- 1977-09-09 AT AT649177A patent/AT352279B/de not_active IP Right Cessation
- 1977-09-09 AT AT649077A patent/AT352278B/de not_active IP Right Cessation
- 1977-09-12 ES ES462294A patent/ES462294A1/es not_active Expired
- 1977-09-12 ES ES462293A patent/ES462293A1/es not_active Expired
- 1977-09-21 JP JP11276477A patent/JPS5350200A/ja active Granted
- 1977-09-21 JP JP11276377A patent/JPS5350199A/ja active Granted
- 1977-09-21 JP JP11276277A patent/JPS5350198A/ja active Pending
- 1977-09-28 NL NL7710625A patent/NL7710625A/xx not_active Application Discontinuation
- 1977-09-28 NL NL7710627A patent/NL7710627A/xx not_active Application Discontinuation
Cited By (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| FR2426690A2 (fr) * | 1978-06-09 | 1979-12-21 | Archifar Lab Chim Farm | Composes de rifamycine |
Also Published As
Similar Documents
| Publication | Publication Date | Title |
|---|---|---|
| FR2366295A1 (fr) | Composes bactericides de la rifamycine | |
| BG29121A3 (en) | Herbicide means | |
| GB1290411A (OSRAM) | ||
| IT1212143B (it) | Composizione ad attivita'tricogena. | |
| ES467061A1 (es) | Un procedimiento para la preparacion de un compuesto de tia-diazolilbenzamida. | |
| ES8505955A1 (es) | Un procedimiento para preparar nuevas 5-acil-2-(1h)-piridinonas. | |
| ES438571A1 (es) | Metodo de producir compuestos de bencilidensimicarbazida. | |
| GB1404553A (en) | Fish feeds | |
| ES434045A1 (es) | Un procedimiento para la preparacion de compuestos de qui- noxalin-1, 4-dioxido. | |
| FR2366292A1 (fr) | Nouveaux composes tetracycliques derives de diazepine-1,4 a activite biologique | |
| ES384875A1 (es) | Procedimiento para la preparacion de un medio herbicida se-lectivo basado en la n (p - terciobutilfenil) - n'n' - dime-til urea. | |
| GB1497093A (en) | Toothbrush | |
| IE40173L (en) | 3, 4 - dihydro - 1, 2, 4 - triazines; herbicides | |
| BG31468A3 (en) | Mikrobicidnoe sredstvo | |
| SU681800A1 (ru) | 5',3',4-Тринитро-5-амино-2,2'-битиофен, проявляющий антимикробную активность | |
| ES448047A1 (es) | Mejoras introducidas en un procedimiento para la preparacionde 1,1-dioxido de 3,3,4-tetraclorotetrahidrotiofeno. | |
| SU701101A1 (ru) | Производные 2-х-бензилиденгидразино-4-фенил-5n-r- сульфамоилфенилазотиазола, обладающие акарицидной активностью | |
| SU674416A1 (ru) | 2-(o-оксибензилиденгидразино)-4-n-нитрофенил-5-n- ацетилсульфамоилфенилазоселеназол, обладающий бактерицидной и фунгицидной активностью | |
| SU1455632A1 (ru) | О,о-диэтил-n-(1-пропилтио-2-гидрокси-2-метилпропилиден)-амидотиофосфат, обладающий бактерицидной активностью | |
| FR2405649A1 (fr) | Produit antiparasitaire a base de 1,3-benzodithiole-2-thione | |
| SU694028A1 (ru) | Селенсодержащие гидразоны о-нитрокоричного альдегида, обладающие психотропной активностью | |
| IT7826303A0 (it) | Nuovo farmaco ad attivita'antibatterica. | |
| ES477539A1 (es) | Procedimiento de produccion de compuestos de la rifamicina. | |
| ES444322A1 (es) | Procedimiento de preparacion de derivados fenolicos de men- teno. | |
| SU1607351A1 (ru) | 3-БЕНЗОИЛ-1-ФЕНИЛ-1Н-ПИРАЗОЛО[3,4-b]ХИНОКСАЛИН, ПРОЯВЛЯЮЩИЙ ПРОТИВОСТАФИЛОКОККОВУЮ АКТИВНОСТЬ |
Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| TP | Transmission of property | ||
| TP | Transmission of property | ||
| ST | Notification of lapse |