FR2365554A1 - Nouveaux amino-ethers peptidiques, leur preparation et leur application comme medicaments - Google Patents
Nouveaux amino-ethers peptidiques, leur preparation et leur application comme medicamentsInfo
- Publication number
- FR2365554A1 FR2365554A1 FR7729003A FR7729003A FR2365554A1 FR 2365554 A1 FR2365554 A1 FR 2365554A1 FR 7729003 A FR7729003 A FR 7729003A FR 7729003 A FR7729003 A FR 7729003A FR 2365554 A1 FR2365554 A1 FR 2365554A1
- Authority
- FR
- France
- Prior art keywords
- alkyl
- tetrahydro
- aculeacine
- equinocandine
- alkylene
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Withdrawn
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K7/00—Peptides having 5 to 20 amino acids in a fully defined sequence; Derivatives thereof
- C07K7/50—Cyclic peptides containing at least one abnormal peptide link
- C07K7/54—Cyclic peptides containing at least one abnormal peptide link with at least one abnormal peptide link in the ring
- C07K7/56—Cyclic peptides containing at least one abnormal peptide link with at least one abnormal peptide link in the ring the cyclisation not occurring through 2,4-diamino-butanoic acid
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/10—Antimycotics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K38/00—Medicinal preparations containing peptides
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- General Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- Animal Behavior & Ethology (AREA)
- Communicable Diseases (AREA)
- Oncology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Biochemistry (AREA)
- Biophysics (AREA)
- Genetics & Genomics (AREA)
- Proteomics, Peptides & Aminoacids (AREA)
- Molecular Biology (AREA)
- Peptides Or Proteins (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Abstract
L'invention concerne de nouveaux aminoéthers peptidiques et leur préparation. Les composés de l'invention répondent à la formule :
Applications Claiming Priority (9)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
CH1224776 | 1976-09-28 | ||
CH1245076 | 1976-10-01 | ||
CH1244976 | 1976-10-01 | ||
CH1294276 | 1976-10-13 | ||
CH1294176 | 1976-10-13 | ||
CH1357476 | 1976-10-28 | ||
CH161577 | 1977-02-10 | ||
CH161677 | 1977-02-10 | ||
CH206077 | 1977-02-18 |
Publications (1)
Publication Number | Publication Date |
---|---|
FR2365554A1 true FR2365554A1 (fr) | 1978-04-21 |
Family
ID=27575767
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
FR7729003A Withdrawn FR2365554A1 (fr) | 1976-09-28 | 1977-09-27 | Nouveaux amino-ethers peptidiques, leur preparation et leur application comme medicaments |
Country Status (7)
Country | Link |
---|---|
JP (1) | JPS5356684A (fr) |
AU (1) | AU2912777A (fr) |
BE (1) | BE859067A (fr) |
DE (1) | DE2742435A1 (fr) |
FR (1) | FR2365554A1 (fr) |
IL (1) | IL53000A0 (fr) |
NL (1) | NL7710418A (fr) |
Cited By (7)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
FR2458551A1 (fr) * | 1979-06-08 | 1981-01-02 | Lilly Co Eli | Nouveaux antibiotiques, leur preparation et leur utilisation |
FR2484451A1 (fr) * | 1979-12-13 | 1981-12-18 | Lilly Co Eli | Noyaux peptidiques cycliques et leur preparation |
EP0535967A2 (fr) * | 1991-10-01 | 1993-04-07 | Merck & Co. Inc. | Cyclohexapeptides bisaminés |
WO1994021677A1 (fr) * | 1993-03-16 | 1994-09-29 | Merck & Co., Inc. | Composes d'aza cyclohexapeptide |
WO1996013272A1 (fr) * | 1994-10-31 | 1996-05-09 | Merck & Co., Inc. | Composes d'azacyclohexapeptide |
US5516757A (en) * | 1994-09-16 | 1996-05-14 | Merck & Co., Inc. | Semi-synthetic lipopeptides, compositions containing said lipopeptides, and methods of use |
US5854213A (en) * | 1995-01-26 | 1998-12-29 | Merck & Co., Inc. | Antifungal cyclohexapeptides |
Families Citing this family (37)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US4293489A (en) * | 1979-12-13 | 1981-10-06 | Eli Lilly And Company | Derivatives of A-30912A nucleus |
US4293486A (en) * | 1979-12-13 | 1981-10-06 | Eli Lilly And Company | Derivatives of S31794/F-1 nucleus |
US4287120A (en) * | 1979-12-13 | 1981-09-01 | Eli Lilly And Company | Derivatives of S31794/F-1 nucleus |
US4299763A (en) * | 1979-12-13 | 1981-11-10 | Eli Lilly And Company | A-30912B Nucleus |
US4293491A (en) * | 1979-12-13 | 1981-10-06 | Eli Lilly And Company | Derivatives of A-30912H nucleus |
US4320054A (en) * | 1979-12-13 | 1982-03-16 | Eli Lilly And Company | Derivatives of A-30912H nucleus |
US4293484A (en) * | 1979-12-13 | 1981-10-06 | Eli Lilly And Company | Derivatives of A-30912H nucleus |
US4322338A (en) * | 1979-12-13 | 1982-03-30 | Eli Lilly And Company | Derivatives of A-30912B nucleus |
CA1182812A (fr) * | 1979-12-13 | 1985-02-19 | Bernard J. Abbott | Preparation de derives de noyaux de peptides cycliques |
US4289692A (en) * | 1979-12-13 | 1981-09-15 | Eli Lilly And Company | Derivatives of A-30912D nucleus |
US4293490A (en) * | 1979-12-13 | 1981-10-06 | Eli Lilly And Company | A-30912H Nuclei |
US4320052A (en) * | 1979-12-13 | 1982-03-16 | Eli Lilly And Company | Derivatives of A-30912A nucleus |
FR2476074A1 (fr) * | 1979-12-13 | 1981-08-21 | Lilly Co Eli | Derives de noyaux peptidiques cycliques, leur preparation et leur utilisation comme agents antifongiques |
US4297277A (en) * | 1979-12-13 | 1981-10-27 | Eli Lilly And Company | Derivatives of A-30912B nucleus |
US4304716A (en) * | 1979-12-13 | 1981-12-08 | Eli Lilly And Company | S 31794/F-1 Nucleus |
US4293483A (en) * | 1979-12-13 | 1981-10-06 | Eli Lilly And Company | Derivatives of A-30912A nucleus |
US4293487A (en) * | 1979-12-13 | 1981-10-06 | Eli Lilly And Company | Derivatives of A-30912D nucleus |
US4320053A (en) * | 1979-12-13 | 1982-03-16 | Eli Lilly And Company | Derivatives of A-30912D nucleus |
US4293482A (en) * | 1979-12-13 | 1981-10-06 | Eli Lilly And Company | A-30912A Nucleus |
US4293485A (en) * | 1979-12-13 | 1981-10-06 | Eli Lilly And Company | Derivatives of S31794/F-1 nucleus |
US4299762A (en) * | 1979-12-13 | 1981-11-10 | Eli Lilly And Company | A-30912D Nucleus |
US4293488A (en) * | 1979-12-13 | 1981-10-06 | Eli Lilly And Company | Derivatives of A-30912B nucleus |
US5166135A (en) * | 1988-09-12 | 1992-11-24 | Merck & Company, Inc. | Method for the control of pneumocystis carinii |
US5021341A (en) * | 1990-03-12 | 1991-06-04 | Merck & Co., Inc. | Antibiotic agent produced by the cultivation of Zalerion microorganism in the presence of mannitol |
US5049546A (en) * | 1990-03-19 | 1991-09-17 | Merck & Co., Inc. | Antibiotic agents |
US5021403A (en) * | 1990-03-19 | 1991-06-04 | Merck & Co., Inc. | Antibiotic agents |
US5939384A (en) * | 1991-10-01 | 1999-08-17 | Merck & Co., Inc. | Cyclohexapeptidyl propanolamine compounds |
US5399552A (en) * | 1991-10-17 | 1995-03-21 | Merck & Co, Inc | Antibiotic peptides bearing aminoalkylthioether moieties |
US5914313A (en) * | 1991-10-17 | 1999-06-22 | Merck & Co., Inc. | 1- 4-hydroxy-5-aminoethyloxy-N2 -(10,12-dimethyl-1-oxotetradecyl)ornithine!-5-(3-hydroxyglutamine)-6-(3-hydroxyproline)echinocandin B, other aminoalkyl derivatives and salts thereof |
US5874403A (en) * | 1992-10-15 | 1999-02-23 | Merck & Co., Inc. | Amino acid conjugates of cyclohexapeptidyl amines |
AU5354094A (en) * | 1992-10-16 | 1994-05-09 | Merck & Co., Inc. | An improved process for cyclohexapeptidyl bisamine compounds |
US6268338B1 (en) | 1993-04-30 | 2001-07-31 | Merck & Co., Inc. | Cyclohexapeptidyl amine compounds |
US5948753A (en) * | 1993-05-04 | 1999-09-07 | Merck & Co., Inc. | Cyclohexapeptidyl propanolamine compounds |
WO1994025045A1 (fr) * | 1993-05-04 | 1994-11-10 | Merck & Co., Inc. | Ethers d'aminoalkyle de cyclohexapeptidyle |
WO1995008341A1 (fr) * | 1993-09-22 | 1995-03-30 | Merck & Co., Inc. | Composes antifongiques et anti-pneumocystose, compositions les contenant et procedes d'utilisation |
DE69513408T2 (de) * | 1994-08-23 | 2000-06-08 | Merck & Co Inc | Ein verbessertes verfahren für die herstellung von seitenketten-derivaten von cyclohexapeptidyl-lipopeptiden |
WO2016201283A1 (fr) | 2015-06-12 | 2016-12-15 | Cidara Therapeutics, Inc. | Agents antifongiques |
Citations (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
FR2340947A1 (fr) * | 1976-02-12 | 1977-09-09 | Sandoz Sa | Nouveaux derives de la tetrahydro-equinocandine b, leur preparation et leur application comme medicaments |
-
1977
- 1977-09-21 DE DE19772742435 patent/DE2742435A1/de active Pending
- 1977-09-23 NL NL7710418A patent/NL7710418A/xx not_active Application Discontinuation
- 1977-09-26 BE BE181214A patent/BE859067A/fr unknown
- 1977-09-26 AU AU29127/77A patent/AU2912777A/en active Pending
- 1977-09-26 IL IL53000A patent/IL53000A0/xx unknown
- 1977-09-27 FR FR7729003A patent/FR2365554A1/fr not_active Withdrawn
- 1977-09-27 JP JP11601777A patent/JPS5356684A/ja active Pending
Patent Citations (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
FR2340947A1 (fr) * | 1976-02-12 | 1977-09-09 | Sandoz Sa | Nouveaux derives de la tetrahydro-equinocandine b, leur preparation et leur application comme medicaments |
Cited By (12)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
FR2458551A1 (fr) * | 1979-06-08 | 1981-01-02 | Lilly Co Eli | Nouveaux antibiotiques, leur preparation et leur utilisation |
FR2484451A1 (fr) * | 1979-12-13 | 1981-12-18 | Lilly Co Eli | Noyaux peptidiques cycliques et leur preparation |
EP0535967A2 (fr) * | 1991-10-01 | 1993-04-07 | Merck & Co. Inc. | Cyclohexapeptides bisaminés |
EP0535967A3 (fr) * | 1991-10-01 | 1994-04-06 | Merck & Co Inc | |
WO1994021677A1 (fr) * | 1993-03-16 | 1994-09-29 | Merck & Co., Inc. | Composes d'aza cyclohexapeptide |
EP0620232A1 (fr) * | 1993-03-16 | 1994-10-19 | Merck & Co. Inc. | Aza-cyclohexapeptides |
US5792746A (en) * | 1993-03-16 | 1998-08-11 | Merck & Co., Inc. | Aza cyclohexapeptide compounds |
CN1098274C (zh) * | 1993-03-16 | 2003-01-08 | 麦克公司 | 氮杂环己肽化合物 |
US5516757A (en) * | 1994-09-16 | 1996-05-14 | Merck & Co., Inc. | Semi-synthetic lipopeptides, compositions containing said lipopeptides, and methods of use |
WO1996013272A1 (fr) * | 1994-10-31 | 1996-05-09 | Merck & Co., Inc. | Composes d'azacyclohexapeptide |
US5516756A (en) * | 1994-10-31 | 1996-05-14 | Merck & Co., Inc. | Aza cyclohexapeptide compounds |
US5854213A (en) * | 1995-01-26 | 1998-12-29 | Merck & Co., Inc. | Antifungal cyclohexapeptides |
Also Published As
Publication number | Publication date |
---|---|
NL7710418A (nl) | 1978-03-30 |
DE2742435A1 (de) | 1978-04-06 |
BE859067A (fr) | 1978-03-28 |
JPS5356684A (en) | 1978-05-23 |
IL53000A0 (en) | 1977-11-30 |
AU2912777A (en) | 1979-04-05 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
RE | Withdrawal of published application |