FR2220257A1 - 5,6-Dihydro-(4H)-s-triazolo-(4,3-a) (1,5)benzodiazepines - as antiinflam-matory and analgesic agents without tranquillising effects - Google Patents
5,6-Dihydro-(4H)-s-triazolo-(4,3-a) (1,5)benzodiazepines - as antiinflam-matory and analgesic agents without tranquillising effectsInfo
- Publication number
- FR2220257A1 FR2220257A1 FR7308510A FR7308510A FR2220257A1 FR 2220257 A1 FR2220257 A1 FR 2220257A1 FR 7308510 A FR7308510 A FR 7308510A FR 7308510 A FR7308510 A FR 7308510A FR 2220257 A1 FR2220257 A1 FR 2220257A1
- Authority
- FR
- France
- Prior art keywords
- antiinflam
- tranquillising
- matory
- benzodiazepines
- triazolo
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems
Priority Applications (19)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
FR7308510A FR2220257A1 (en) | 1973-03-09 | 1973-03-09 | 5,6-Dihydro-(4H)-s-triazolo-(4,3-a) (1,5)benzodiazepines - as antiinflam-matory and analgesic agents without tranquillising effects |
IE00393/74A IE38931B1 (en) | 1973-03-09 | 1974-02-26 | Triazolobenzodiazepines |
BE141389A BE811576A (fr) | 1973-03-09 | 1974-02-26 | Nouvelles dihydro-5 |
ZA00741263A ZA741263B (en) | 1973-03-09 | 1974-02-26 | 4h-5,6-dihydro-4,3-a-s-triazolo-1, 5-benzodiazepines and theur preparation |
DE2409308A DE2409308C3 (de) | 1973-03-09 | 1974-02-27 | 5,6-Dihydro- [4 H] (s)triazolo- [43-a] -1,5benzodiazepine, Verfahren zu ihrer Herstellung und sie enthaltende Arzneimittel |
IL44338A IL44338A (en) | 1973-03-09 | 1974-03-04 | 4h-5,6-dihydro-1-phenyl-(4,3-a)-s-triazolo-1,5-benzodiazepines,their preparation and pharmaceutical compositions containing them |
AU66276/74A AU478312B2 (en) | 1973-03-09 | 1974-03-05 | New triazolobenzodiazepines and process for their preparation |
GB1035574A GB1409693A (en) | 1973-03-09 | 1974-03-07 | Triazolobenzodiazepines |
HULI000251 HU168538B (fr) | 1973-03-09 | 1974-03-08 | |
US05/449,477 US4110337A (en) | 1973-03-09 | 1974-03-08 | Triazolobenzodiazepines |
NO740833A NO139048C (no) | 1973-03-09 | 1974-03-08 | Analogifremgangsmaate for fremstilling av nye analgetisk og/eller antiinflammatorisk virksomme (4h)-5,6-dihydro-(4,3-a)-s-triazolo-1,5-benzodiazepiner |
DD177060A DD110497A5 (fr) | 1973-03-09 | 1974-03-08 | |
ES424067A ES424067A1 (es) | 1973-03-09 | 1974-03-08 | Procedimiento de preparacion de dihidro - 5,6 (4h) - (s) - triazolo - (3,3 - a) - benzodiazepinas - 1,5. |
AT195974A AT336024B (de) | 1973-03-09 | 1974-03-08 | Verfahren zur herstellung von neuen 5,6-dihydro-(4 h)- (s)-triazolo-(4,3-a)-1,5-benzodiazepinen |
CH332374A CH589084A5 (fr) | 1973-03-09 | 1974-03-08 | |
DK125874AA DK139099B (da) | 1973-03-09 | 1974-03-08 | Analogifremgangsmåde til fremstilling af 5,6-4H-dihydro-s-triazolo(4,3-a)benzodiazepiner-1,5. |
CA194,513A CA1011333A (en) | 1973-03-09 | 1974-03-08 | (4h)-5,6-dihydro-(4,3-a)-s-triazolo-1,5-benzodiazepines and their process of preparation |
JP49026797A JPS49125395A (fr) | 1973-03-09 | 1974-03-09 | |
NL7403247A NL7403247A (fr) | 1973-03-09 | 1974-03-11 |
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
FR7308510A FR2220257A1 (en) | 1973-03-09 | 1973-03-09 | 5,6-Dihydro-(4H)-s-triazolo-(4,3-a) (1,5)benzodiazepines - as antiinflam-matory and analgesic agents without tranquillising effects |
Publications (2)
Publication Number | Publication Date |
---|---|
FR2220257A1 true FR2220257A1 (en) | 1974-10-04 |
FR2220257B1 FR2220257B1 (fr) | 1976-08-13 |
Family
ID=9116060
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
FR7308510A Granted FR2220257A1 (en) | 1973-03-09 | 1973-03-09 | 5,6-Dihydro-(4H)-s-triazolo-(4,3-a) (1,5)benzodiazepines - as antiinflam-matory and analgesic agents without tranquillising effects |
Country Status (3)
Country | Link |
---|---|
BE (1) | BE811576A (fr) |
FR (1) | FR2220257A1 (fr) |
ZA (1) | ZA741263B (fr) |
Cited By (8)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US6630004B1 (en) | 1997-10-08 | 2003-10-07 | L'oreal S.A. | Oxidation dye composition for keratinous fibers |
EP2705039A2 (fr) * | 2011-05-04 | 2014-03-12 | Constellation Pharmaceuticals, Inc. | Inhibiteurs de bromodomaines et leurs utilisations |
US9249161B2 (en) | 2010-12-02 | 2016-02-02 | Constellation Pharmaceuticals, Inc. | Bromodomain inhibitors and uses thereof |
US9328117B2 (en) | 2011-06-17 | 2016-05-03 | Constellation Pharmaceuticals, Inc. | Bromodomain inhibitors and uses thereof |
US9493483B2 (en) | 2012-06-06 | 2016-11-15 | Constellation Pharmaceuticals, Inc. | Benzo [C] isoxazoloazepine bromodomain inhibitors and uses thereof |
US9522920B2 (en) | 2010-12-02 | 2016-12-20 | Constellation Pharmaceuticals, Inc. | Bromodomain inhibitors and uses thereof |
US9624244B2 (en) | 2012-06-06 | 2017-04-18 | Constellation Pharmaceuticals, Inc. | Benzo [B] isoxazoloazepine bromodomain inhibitors and uses thereof |
US9969747B2 (en) | 2014-06-20 | 2018-05-15 | Constellation Pharmaceuticals, Inc. | Crystalline forms of 2-((4S)-6-(4-chlorophenyl)-1-methyl-4H-benzo[C]isoxazolo[4,5-e]azepin-4-yl)acetamide |
Citations (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
FR2137714A1 (fr) * | 1971-05-11 | 1972-12-29 | Upjohn Co |
-
1973
- 1973-03-09 FR FR7308510A patent/FR2220257A1/fr active Granted
-
1974
- 1974-02-26 BE BE141389A patent/BE811576A/fr not_active IP Right Cessation
- 1974-02-26 ZA ZA00741263A patent/ZA741263B/xx unknown
Patent Citations (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
FR2137714A1 (fr) * | 1971-05-11 | 1972-12-29 | Upjohn Co |
Cited By (11)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US6630004B1 (en) | 1997-10-08 | 2003-10-07 | L'oreal S.A. | Oxidation dye composition for keratinous fibers |
US9249161B2 (en) | 2010-12-02 | 2016-02-02 | Constellation Pharmaceuticals, Inc. | Bromodomain inhibitors and uses thereof |
US9522920B2 (en) | 2010-12-02 | 2016-12-20 | Constellation Pharmaceuticals, Inc. | Bromodomain inhibitors and uses thereof |
EP2705039A2 (fr) * | 2011-05-04 | 2014-03-12 | Constellation Pharmaceuticals, Inc. | Inhibiteurs de bromodomaines et leurs utilisations |
EP2705039A4 (fr) * | 2011-05-04 | 2014-10-08 | Constellation Pharmaceuticals Inc | Inhibiteurs de bromodomaines et leurs utilisations |
US9422292B2 (en) | 2011-05-04 | 2016-08-23 | Constellation Pharmaceuticals, Inc. | Bromodomain inhibitors and uses thereof |
US9328117B2 (en) | 2011-06-17 | 2016-05-03 | Constellation Pharmaceuticals, Inc. | Bromodomain inhibitors and uses thereof |
US9493483B2 (en) | 2012-06-06 | 2016-11-15 | Constellation Pharmaceuticals, Inc. | Benzo [C] isoxazoloazepine bromodomain inhibitors and uses thereof |
US9624244B2 (en) | 2012-06-06 | 2017-04-18 | Constellation Pharmaceuticals, Inc. | Benzo [B] isoxazoloazepine bromodomain inhibitors and uses thereof |
US9925197B2 (en) | 2012-06-06 | 2018-03-27 | Constellation Pharmaceuticals, Inc. | Benzo [C] isoxazoloazepine bromodomain inhibitors and uses thereof |
US9969747B2 (en) | 2014-06-20 | 2018-05-15 | Constellation Pharmaceuticals, Inc. | Crystalline forms of 2-((4S)-6-(4-chlorophenyl)-1-methyl-4H-benzo[C]isoxazolo[4,5-e]azepin-4-yl)acetamide |
Also Published As
Publication number | Publication date |
---|---|
BE811576A (fr) | 1974-06-17 |
FR2220257B1 (fr) | 1976-08-13 |
ZA741263B (en) | 1975-01-29 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
ST | Notification of lapse |