FR2100973A1 - 5-Aminopyrazoles - with analgesic, antiinflammatory and muscle relaxant activity - Google Patents

5-Aminopyrazoles - with analgesic, antiinflammatory and muscle relaxant activity

Info

Publication number
FR2100973A1
FR2100973A1 FR7128105A FR7128105A FR2100973A1 FR 2100973 A1 FR2100973 A1 FR 2100973A1 FR 7128105 A FR7128105 A FR 7128105A FR 7128105 A FR7128105 A FR 7128105A FR 2100973 A1 FR2100973 A1 FR 2100973A1
Authority
FR
France
Prior art keywords
antiinflammatory
analgesic
aminopyrazoles
muscle relaxant
relaxant activity
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
FR7128105A
Other languages
English (en)
French (fr)
Other versions
FR2100973B1 (OSRAM
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Tanabe Pharma Corp
Original Assignee
Yoshitomi Pharmaceutical Industries Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Yoshitomi Pharmaceutical Industries Ltd filed Critical Yoshitomi Pharmaceutical Industries Ltd
Priority to FR7128105A priority Critical patent/FR2100973A1/fr
Publication of FR2100973A1 publication Critical patent/FR2100973A1/fr
Application granted granted Critical
Publication of FR2100973B1 publication Critical patent/FR2100973B1/fr
Granted legal-status Critical Current

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D231/00Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/14Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D231/38Nitrogen atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D231/00Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/14Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D231/38Nitrogen atoms
    • C07D231/40Acylated on said nitrogen atom

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
FR7128105A 1970-07-30 1971-07-30 5-Aminopyrazoles - with analgesic, antiinflammatory and muscle relaxant activity Granted FR2100973A1 (en)

Priority Applications (1)

Application Number Priority Date Filing Date Title
FR7128105A FR2100973A1 (en) 1970-07-30 1971-07-30 5-Aminopyrazoles - with analgesic, antiinflammatory and muscle relaxant activity

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
JP6707470 1970-07-30
FR7128105A FR2100973A1 (en) 1970-07-30 1971-07-30 5-Aminopyrazoles - with analgesic, antiinflammatory and muscle relaxant activity

Publications (2)

Publication Number Publication Date
FR2100973A1 true FR2100973A1 (en) 1972-03-24
FR2100973B1 FR2100973B1 (OSRAM) 1975-02-07

Family

ID=26216548

Family Applications (1)

Application Number Title Priority Date Filing Date
FR7128105A Granted FR2100973A1 (en) 1970-07-30 1971-07-30 5-Aminopyrazoles - with analgesic, antiinflammatory and muscle relaxant activity

Country Status (1)

Country Link
FR (1) FR2100973A1 (OSRAM)

Cited By (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0068806A3 (en) * 1981-06-26 1983-08-10 Warner-Lambert Company Basic acyl amides of (5-amino-1,3-dialkylpyrazol-4-yl)(aryl)methanones, processes for their production, and pharmaceutical compositions containing such compounds
US6316466B1 (en) 1998-05-05 2001-11-13 Syntex (U.S.A.) Llc Pyrazole derivatives P-38 MAP kinase inhibitors
US6376527B1 (en) 1998-05-05 2002-04-23 Syntex (U.S.A.) Llc Pyrazole derivatives-p38 map kinase inhibitors
US6979693B2 (en) 1998-05-05 2005-12-27 Syntex (U.S.A.) Llc Pyrazole derivatives-p38 MAP kinase inhibitors

Citations (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US2989537A (en) * 1958-05-30 1961-06-20 Ciba Pharm Prod Inc Pyrazolo [2, 3-alpha] imidazolidines
FR2023474A1 (OSRAM) * 1968-11-16 1970-08-21 Bayer Ag

Patent Citations (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US2989537A (en) * 1958-05-30 1961-06-20 Ciba Pharm Prod Inc Pyrazolo [2, 3-alpha] imidazolidines
FR2023474A1 (OSRAM) * 1968-11-16 1970-08-21 Bayer Ag

Cited By (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0068806A3 (en) * 1981-06-26 1983-08-10 Warner-Lambert Company Basic acyl amides of (5-amino-1,3-dialkylpyrazol-4-yl)(aryl)methanones, processes for their production, and pharmaceutical compositions containing such compounds
US6316466B1 (en) 1998-05-05 2001-11-13 Syntex (U.S.A.) Llc Pyrazole derivatives P-38 MAP kinase inhibitors
US6376527B1 (en) 1998-05-05 2002-04-23 Syntex (U.S.A.) Llc Pyrazole derivatives-p38 map kinase inhibitors
US6979693B2 (en) 1998-05-05 2005-12-27 Syntex (U.S.A.) Llc Pyrazole derivatives-p38 MAP kinase inhibitors

Also Published As

Publication number Publication date
FR2100973B1 (OSRAM) 1975-02-07

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Legal Events

Date Code Title Description
ST Notification of lapse