FI943100A - Ansamysiinijohdannaisia antionkogeenisina ja syövänvastaisina aineina - Google Patents
Ansamysiinijohdannaisia antionkogeenisina ja syövänvastaisina aineina Download PDFInfo
- Publication number
- FI943100A FI943100A FI943100A FI943100A FI943100A FI 943100 A FI943100 A FI 943100A FI 943100 A FI943100 A FI 943100A FI 943100 A FI943100 A FI 943100A FI 943100 A FI943100 A FI 943100A
- Authority
- FI
- Finland
- Prior art keywords
- anthionogenic
- cancer agents
- ansamycin derivatives
- ansamycin
- derivatives
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
- C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
- C07D403/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings directly linked by a ring-member-to-ring-member bond
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D225/00—Heterocyclic compounds containing rings of more than seven members having one nitrogen atom as the only ring hetero atom
- C07D225/04—Heterocyclic compounds containing rings of more than seven members having one nitrogen atom as the only ring hetero atom condensed with carbocyclic rings or ring systems
- C07D225/06—Heterocyclic compounds containing rings of more than seven members having one nitrogen atom as the only ring hetero atom condensed with carbocyclic rings or ring systems condensed with one six-membered ring
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
- C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
- C07D403/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
- C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
- C07D405/12—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a chain containing hetero atoms as chain links
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US8506593A | 1993-06-29 | 1993-06-29 |
Publications (2)
Publication Number | Publication Date |
---|---|
FI943100A0 FI943100A0 (fi) | 1994-06-28 |
FI943100A true FI943100A (fi) | 1994-12-30 |
Family
ID=22189242
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
FI943100A FI943100A (fi) | 1993-06-29 | 1994-06-28 | Ansamysiinijohdannaisia antionkogeenisina ja syövänvastaisina aineina |
Country Status (5)
Country | Link |
---|---|
EP (1) | EP0706516A1 (fi) |
JP (1) | JP2794342B2 (fi) |
CA (1) | CA2166320A1 (fi) |
FI (1) | FI943100A (fi) |
WO (1) | WO1995001342A1 (fi) |
Families Citing this family (17)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
JP2002520369A (ja) | 1998-07-17 | 2002-07-09 | アメリカ合衆国 | 水溶性薬剤およびその製造方法 |
AU769235B2 (en) * | 1999-04-09 | 2004-01-22 | Sloan-Kettering Institute For Cancer Research | Methods and compositions for degradation and/or inhibition of her-family tyrosine kinases |
AU2002217866A1 (en) * | 2000-11-06 | 2002-05-15 | The Government Of The United States Of America, As Represented By The Secretary Of The Department Of Health And Human Services | Geldanamycin derivatives useful for the treatment of cancer |
SI21369A (sl) * | 2001-03-30 | 2004-06-30 | The United States Of America, Represented By The Secretary, | Geldanamicinski derivat in postopek zdravljenja raka z uporabo le-tega |
WO2003013430A2 (en) * | 2001-08-06 | 2003-02-20 | Kosan Biosciences, Inc. | Benzoquinone ansamycins |
EP1923061A1 (en) | 2001-09-24 | 2008-05-21 | Conforma Therapeutic Corporation | Process for preparing 17-Allyl amino geldanamycin (17-AAG) and other ansamycins |
DE60225307T2 (de) * | 2001-09-24 | 2009-03-19 | Conforma Therapeutics Corp., San Diego | Verfahren zur herstellung von 17-allyl-amino-geldanamycin (17-aag) und anderer ansamycine |
ATE433961T1 (de) | 2002-02-08 | 2009-07-15 | Conforma Therapeutics Corp | Ansamycine mit verbesserten pharmakologischen und biologischen eigenschaften |
AU2003277299B2 (en) * | 2002-04-10 | 2009-12-10 | Conforma Therapeutics Corporation | Drug formulations having long and medium chain triglycerides |
US6855705B1 (en) | 2003-11-12 | 2005-02-15 | Kosan Biosciences, Inc. | 11-O-methylgeldanamycin compounds |
US6887993B1 (en) | 2003-11-12 | 2005-05-03 | Kosan Biosciences, Inc. | 11-O-methylgeldanamycin compounds |
US6875863B1 (en) | 2003-11-12 | 2005-04-05 | Kosan Biosciences, Inc. | 11-O-methylgeldanamycin compounds |
CA2545457A1 (en) | 2003-11-12 | 2005-06-23 | Kosan Biosciences, Inc. | 11-o-methylgeldanamycin compounds |
US20060019941A1 (en) * | 2003-12-23 | 2006-01-26 | Infinity Pharmaceuticals, Inc. | Analogs of benzoquinone-containing ansamycins and methods of use thereof |
EP2492261B1 (en) | 2003-12-23 | 2015-02-18 | Infinity Discovery, Inc. | Analogs of benzoquinone-containing ansamycins for the treatment of cancer |
PE20081506A1 (es) * | 2006-12-12 | 2008-12-09 | Infinity Discovery Inc | Formulaciones de ansamicina |
WO2010045442A1 (en) | 2008-10-15 | 2010-04-22 | Infinity Discovery, Inc. | Ansamycin hydroquinone compositions |
Family Cites Families (4)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US3595955A (en) * | 1969-03-26 | 1971-07-27 | Upjohn Co | Geldanamycin and process for producing same |
US3987035A (en) * | 1974-04-05 | 1976-10-19 | University Of Illinois Foundation | Biologically active compounds |
US4261989A (en) * | 1979-02-19 | 1981-04-14 | Kaken Chemical Co. Ltd. | Geldanamycin derivatives and antitumor drug |
JPH06510913A (ja) * | 1992-01-06 | 1994-12-08 | フアイザー・インコーポレイテツド | 4,5‐ジヒドロゲルダナマイシン及びそのヒドロキノンの製造及び使用 |
-
1994
- 1994-06-16 WO PCT/IB1994/000160 patent/WO1995001342A1/en not_active Application Discontinuation
- 1994-06-16 EP EP94916372A patent/EP0706516A1/en not_active Withdrawn
- 1994-06-16 CA CA002166320A patent/CA2166320A1/en not_active Abandoned
- 1994-06-16 JP JP7503379A patent/JP2794342B2/ja not_active Expired - Lifetime
- 1994-06-28 FI FI943100A patent/FI943100A/fi unknown
Also Published As
Publication number | Publication date |
---|---|
JP2794342B2 (ja) | 1998-09-03 |
FI943100A0 (fi) | 1994-06-28 |
WO1995001342A1 (en) | 1995-01-12 |
CA2166320A1 (en) | 1995-01-12 |
JPH08506356A (ja) | 1996-07-09 |
EP0706516A1 (en) | 1996-04-17 |
Similar Documents
Publication | Publication Date | Title |
---|---|---|
FI961599A (fi) | 1N-alkyyli-N-aryylipyrimidiiniamiineja ja niiden johdannaisia | |
ATE162199T1 (de) | Androstenderivate | |
FI941137A (fi) | 2-debentsoyyli-2-asyylitaksolijohdannaisia ja menetelmiä niiden valmistamiseksi | |
EE9700190A (et) | Pürasool-4-üül-bensoüüli derivaadid ja nende kasutamine herbitsiididena | |
FI944310A0 (fi) | Heteroaryyliamino- ja heteroaryylisuolfonamidosubstituoituja 3-bentsyyliaminometyylipiperidiinejä ja vastaavia yhdisteitä | |
FI953479A0 (fi) | 1-aryylipyrimidiinijohdannaiset ja niiden farmaseuttinen käyttö | |
ATA75293A (de) | Indolderivate | |
FI943100A (fi) | Ansamysiinijohdannaisia antionkogeenisina ja syövänvastaisina aineina | |
ITMI920408A1 (it) | Derivati benzopiranici e benzotiopiranici | |
DE69330497D1 (de) | Chinazolin-derivate | |
FI960867A (fi) | Bentsatsepiinijohdannainen, sen farmaseuttinen seos ja välituote | |
DE59308714D1 (de) | Cyclobutan-benzol-derivate | |
FI953021A0 (fi) | 4-bentsoyyli-isoksatsolin johdannaisia ja niiden käyttö herbisideinä | |
FI960076A0 (fi) | Uudet (1-heteroatsolyyli-1-heterosyklyyli) alkaanijohdannaiset ja niiden käyttö hermostoa suojaavina aineina | |
BR9408029A (pt) | Derivados de 3-azabicicloalcanos N-substituídos | |
FI955679A0 (fi) | Piperidiinijohdannaisia, niiden valmistus ja käyttö | |
NO952288D0 (no) | Benzazepinon-derivater | |
DE69313890D1 (de) | 5-Aminoflavon-Derivate | |
EE9800054A (et) | Pürasool-4-üül-bensoüüli derivaadid ja nende kasutamine herbitsiididena | |
FI943513A0 (fi) | Kolekystokiniiniantagonisteina käyttökelpoisia 3-fenyyliureidoatsepin-2-oneja ja -bentsatsepin-2-oneja | |
DE59407726D1 (de) | 3-Aryl-4-hydroxy-3-dihydrofuranon-Derivate | |
ITMI941191A0 (it) | 1-b-metil-2-tiol carbapen derivati | |
FI950303A (fi) | Pyridoindolobentsodiatsepiinit ja johdannaiset antipsykoottisina aineina | |
DE69400388D1 (de) | Cyclohexendiolderivate | |
NO934473D0 (no) | N-substituerte azabicykloheptanderivater |