FI93118B - Menetelmä uusien terapeuttisesti käyttökelpoisten 1,4-diatsepiinijohdannaisten valmistamiseksi - Google Patents

Menetelmä uusien terapeuttisesti käyttökelpoisten 1,4-diatsepiinijohdannaisten valmistamiseksi

Info

Publication number
FI93118B
FI93118B FI893250A FI893250A FI93118B FI 93118 B FI93118 B FI 93118B FI 893250 A FI893250 A FI 893250A FI 893250 A FI893250 A FI 893250A FI 93118 B FI93118 B FI 93118B
Authority
FI
Finland
Prior art keywords
preparation
therapeutically useful
new therapeutically
diazepine derivatives
diazepine
Prior art date
Application number
FI893250A
Other languages
English (en)
Swedish (sv)
Other versions
FI93118C (fi
FI893250A0 (fi
FI893250A (fi
Inventor
Hartog Jacobus Antonius Jo Den
Stuivenberg Herman Heinric Van
Wijngaarden Ineke Van
Original Assignee
Duphar Int Res
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Duphar Int Res filed Critical Duphar Int Res
Publication of FI893250A0 publication Critical patent/FI893250A0/fi
Publication of FI893250A publication Critical patent/FI893250A/fi
Application granted granted Critical
Publication of FI93118B publication Critical patent/FI93118B/fi
Publication of FI93118C publication Critical patent/FI93118C/fi

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/55Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole
    • A61K31/551Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole having two nitrogen atoms, e.g. dilazep
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D491/00Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00
    • C07D491/02Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains two hetero rings
    • C07D491/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/04Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D495/00Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
    • C07D495/02Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
    • C07D495/04Ortho-condensed systems
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D495/00Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
    • C07D495/12Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains three hetero rings
    • C07D495/14Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Engineering & Computer Science (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
FI893250A 1988-07-07 1989-07-04 Menetelmä uusien terapeuttisesti käyttökelpoisten 1,4-diatsepiinijohdannaisten valmistamiseksi FI93118C (fi)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
NL8801716 1988-07-07
NL8801716 1988-07-07

Publications (4)

Publication Number Publication Date
FI893250A0 FI893250A0 (fi) 1989-07-04
FI893250A FI893250A (fi) 1990-01-08
FI93118B true FI93118B (fi) 1994-11-15
FI93118C FI93118C (fi) 1995-02-27

Family

ID=19852585

Family Applications (1)

Application Number Title Priority Date Filing Date
FI893250A FI93118C (fi) 1988-07-07 1989-07-04 Menetelmä uusien terapeuttisesti käyttökelpoisten 1,4-diatsepiinijohdannaisten valmistamiseksi

Country Status (16)

Country Link
US (2) US4985423A (fi)
EP (1) EP0350131A3 (fi)
JP (1) JPH0259582A (fi)
KR (1) KR900001696A (fi)
CN (1) CN1028408C (fi)
AU (1) AU626892B2 (fi)
CA (1) CA1315781C (fi)
DK (1) DK330689A (fi)
FI (1) FI93118C (fi)
HU (1) HU204528B (fi)
IL (1) IL90865A (fi)
NO (1) NO170282C (fi)
NZ (1) NZ229815A (fi)
PT (1) PT91052B (fi)
TW (1) TW219896B (fi)
ZA (1) ZA895086B (fi)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB0015904D0 (en) * 2000-06-28 2000-08-23 Hoffmann La Roche Inhibitors of HPV E1 helicase enzyme
DE10312969A1 (de) * 2003-03-24 2004-10-07 Bayer Healthcare Ag Benzofuro-1,4-diazepin-2-on-Derivate
WO2009049362A1 (en) * 2007-10-15 2009-04-23 Monash University A1 adenosine receptor allosteric enhancers
WO2015088565A1 (en) * 2013-12-13 2015-06-18 Sunovion Pharmaceuticals Inc. P2x4 receptor modulating compounds and methods of use thereof

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3910887A (en) * 1972-12-07 1975-10-07 Degussa Azabenzo-1,5-diazepines
US4404137A (en) * 1979-10-16 1983-09-13 Lilly Industries Limited Pyrazolo [3,4-b][1,5]benzodiazepine compounds
GB8409960D0 (en) * 1984-04-17 1984-05-31 Searle & Co Therapeutic method
US5087625A (en) * 1990-10-19 1992-02-11 Boehringer Ingelheim Pharmaceuticals, Inc. Pyridodiazepines and their use in the prevention or treatment of HIV infection

Also Published As

Publication number Publication date
CN1028408C (zh) 1995-05-17
FI93118C (fi) 1995-02-27
FI893250A0 (fi) 1989-07-04
FI893250A (fi) 1990-01-08
US4985423A (en) 1991-01-15
NO892772D0 (no) 1989-07-04
PT91052A (pt) 1990-02-08
NO170282B (no) 1992-06-22
JPH0259582A (ja) 1990-02-28
CA1315781C (en) 1993-04-06
DK330689D0 (da) 1989-07-04
EP0350131A3 (en) 1991-07-10
IL90865A0 (en) 1990-02-09
TW219896B (fi) 1994-02-01
NO170282C (no) 1992-09-30
AU626892B2 (en) 1992-08-13
NO892772L (no) 1990-01-08
DK330689A (da) 1990-01-08
PT91052B (pt) 1995-01-31
AU3795489A (en) 1990-01-11
NZ229815A (en) 1992-03-26
US5140024A (en) 1992-08-18
IL90865A (en) 1994-02-27
KR900001696A (ko) 1990-02-27
ZA895086B (en) 1990-05-30
EP0350131A2 (en) 1990-01-10
HU204528B (en) 1992-01-28
CN1040027A (zh) 1990-02-28

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Legal Events

Date Code Title Description
BB Publication of examined application
MM Patent lapsed
MM Patent lapsed

Owner name: DUPHAR INTERNATIONAL RESEARCH B.V