FI914258A - Antiarrytmiska arylkondenserade och hetarylkondenserade 2,4-diazepin- och 2,4-diazocinderivat och deras framstaellning. - Google Patents
Antiarrytmiska arylkondenserade och hetarylkondenserade 2,4-diazepin- och 2,4-diazocinderivat och deras framstaellning. Download PDFInfo
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- FI914258A FI914258A FI914258A FI914258A FI914258A FI 914258 A FI914258 A FI 914258A FI 914258 A FI914258 A FI 914258A FI 914258 A FI914258 A FI 914258A FI 914258 A FI914258 A FI 914258A
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- alkyl
- och
- hydrogen
- aryl
- hetaryl
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- C07D295/04—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms
- C07D295/12—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by singly or doubly bound nitrogen atoms
- C07D295/125—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by singly or doubly bound nitrogen atoms with the ring nitrogen atoms and the substituent nitrogen atoms attached to the same carbon chain, which is not interrupted by carbocyclic rings
- C07D295/13—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by singly or doubly bound nitrogen atoms with the ring nitrogen atoms and the substituent nitrogen atoms attached to the same carbon chain, which is not interrupted by carbocyclic rings to an acyclic saturated chain
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- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
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- C07C217/06—Compounds containing amino and etherified hydroxy groups bound to the same carbon skeleton having etherified hydroxy groups and amino groups bound to acyclic carbon atoms of the same carbon skeleton the carbon skeleton being acyclic and saturated having only one etherified hydroxy group and one amino group bound to the carbon skeleton, which is not further substituted
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- C07C233/35—Carboxylic acid amides having carbon atoms of carboxamide groups bound to hydrogen atoms or to acyclic carbon atoms having the nitrogen atom of at least one of the carboxamide groups bound to a carbon atom of a hydrocarbon radical substituted by amino groups with the substituted hydrocarbon radical bound to the nitrogen atom of the carboxamide group by an acyclic carbon atom
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- C07C235/32—Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by oxygen atoms having carbon atoms of carboxamide groups bound to acyclic carbon atoms and singly-bound oxygen atoms bound to the same carbon skeleton the carbon skeleton containing six-membered aromatic rings
- C07C235/34—Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by oxygen atoms having carbon atoms of carboxamide groups bound to acyclic carbon atoms and singly-bound oxygen atoms bound to the same carbon skeleton the carbon skeleton containing six-membered aromatic rings having the nitrogen atoms of the carboxamide groups bound to hydrogen atoms or to acyclic carbon atoms
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- C07C311/02—Sulfonamides having sulfur atoms of sulfonamide groups bound to acyclic carbon atoms of an acyclic saturated carbon skeleton
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- C07C311/06—Sulfonamides having sulfur atoms of sulfonamide groups bound to acyclic carbon atoms of an acyclic saturated carbon skeleton having the nitrogen atoms of the sulfonamide groups bound to hydrogen atoms or to acyclic carbon atoms to acyclic carbon atoms of hydrocarbon radicals substituted by carboxyl groups
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- Heart & Thoracic Surgery (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Plural Heterocyclic Compounds (AREA)
- Medicines Containing Antibodies Or Antigens For Use As Internal Diagnostic Agents (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Polyamides (AREA)
- Furan Compounds (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
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Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US58006590A | 1990-09-10 | 1990-09-10 | |
US74385391A | 1991-06-13 | 1991-06-13 |
Publications (2)
Publication Number | Publication Date |
---|---|
FI914258A0 FI914258A0 (fi) | 1991-09-10 |
FI914258A true FI914258A (fi) | 1992-03-11 |
Family
ID=27077939
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
FI914258A FI914258A (fi) | 1990-09-10 | 1991-09-10 | Antiarrytmiska arylkondenserade och hetarylkondenserade 2,4-diazepin- och 2,4-diazocinderivat och deras framstaellning. |
Country Status (17)
Country | Link |
---|---|
EP (1) | EP0475527B1 (ko) |
JP (1) | JPH05339246A (ko) |
AT (1) | ATE163413T1 (ko) |
AU (2) | AU639821B2 (ko) |
CA (1) | CA2050962A1 (ko) |
DE (1) | DE69128949D1 (ko) |
FI (1) | FI914258A (ko) |
HU (2) | HUT64313A (ko) |
IE (1) | IE913175A1 (ko) |
IL (1) | IL99452A (ko) |
MX (1) | MX9100937A (ko) |
MY (1) | MY109430A (ko) |
NO (1) | NO300268B1 (ko) |
NZ (1) | NZ239407A (ko) |
PT (1) | PT98918B (ko) |
RU (1) | RU2114833C1 (ko) |
TW (1) | TW245719B (ko) |
Families Citing this family (14)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US5380721A (en) * | 1990-09-10 | 1995-01-10 | Sterling Winthrop Inc. | Aryl-fused and hetaryl-fused-2,4-diazepine and 2,4-diazocine antiarrhythmic agents |
CA2104060A1 (en) * | 1992-11-10 | 1994-05-11 | Robert Ed Johnson | Aryl-fused and hetaryl-fused-2,4-diazepine and 2,4-diazocine antiarrhythmic agents |
US5716956A (en) * | 1995-06-07 | 1998-02-10 | Bearsden Bearsden Bio, Inc. | Dihydrophthalazine antagonists of excitatory amino acid receptors |
US6048853A (en) * | 1996-01-18 | 2000-04-11 | Bearsden Bio, Inc. | 1-arylphthalazine antagonists of excitatory amino acid receptors |
IL136499A0 (en) | 1997-12-05 | 2001-06-14 | Astrazeneca Uk Ltd Astrazeneca | Pyrrolo-, thieno-, furano- and pyrazolo-[3,4,d] pypyrrolo-, thieno-, furano- and pyrazolo-[3,4,d] pyridazinone compounds, process for their preparatioridaziones compounds, process for their preparation, pharmaceutical compositions containing them, a n, pharmaceutical compositions containing them, a process for prepating the pharmaceutical compositiprocess for preparing the pharmaceutical compositions, and use thereof ons, and use thereof |
DE19824673A1 (de) * | 1998-05-26 | 1999-12-02 | Schering Ag | Neue 2,3-Benzodiazepinderivate, deren Herstellung und Verwendung als Arzneimittel |
HU9803014D0 (en) * | 1998-12-23 | 1999-02-01 | Egyt Gyogyszervegyeszeti Gyar | Novel phtalazine derivatives, process for their production and pharmaceutical compositions containing the same |
DE19920486A1 (de) * | 1999-05-04 | 2000-11-09 | Basf Ag | Metallorganische Katalysatoren für die Polymerisation ungesättigter Verbindungen |
CN101106994A (zh) * | 2005-01-19 | 2008-01-16 | 默克公司 | 用于治疗阿尔茨海默氏病的氨基甲基β-分泌酶抑制剂 |
EP2323991B1 (en) | 2008-08-13 | 2017-05-31 | Boehringer Ingelheim International GmbH | Chymase inhibitors |
WO2014113620A2 (en) | 2013-01-18 | 2014-07-24 | Bristol-Myers Squibb Company | Phthalazinones and isoquinolinones as rock inhibitors |
US9902702B2 (en) | 2014-07-15 | 2018-02-27 | Bristol-Myers Squibb Company | Spirocycloheptanes as inhibitors of rock |
KR101991429B1 (ko) | 2014-12-19 | 2019-06-20 | 주식회사 엘지화학 | 새로운 화합물 및 이를 이용한 고분자 전해질막 |
CN107082764B (zh) * | 2017-05-23 | 2018-11-02 | 上海锐聚恩新药研发有限公司 | 一类多羟基酞嗪酮化合物、其制备方法及应用 |
Family Cites Families (4)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
CH523264A (de) * | 1967-04-13 | 1972-05-31 | Ciba Geigy Ag | Verfahren zur Herstellung von 2,4 Benzdiazepinen |
US3696093A (en) * | 1970-09-30 | 1972-10-03 | Ciba Geigy Corp | 2,4-benzodiazepines |
ATE13884T1 (de) * | 1979-12-24 | 1985-07-15 | Kali Chemie Pharma Gmbh | 2-azidomethyl-1,4-benzodiazepine und deren salze sowie verfahren zu ihrer herstellung und diese verbindungen enthaltende arzneimittel. |
CA2009542C (en) * | 1989-02-10 | 2000-03-14 | Albert A. Carr | Cyclic guanidines as calcium antagonists |
-
1991
- 1991-08-14 TW TW080106443A patent/TW245719B/zh active
- 1991-08-15 NZ NZ239407A patent/NZ239407A/en unknown
- 1991-08-22 AU AU82641/91A patent/AU639821B2/en not_active Ceased
- 1991-09-04 MX MX9100937A patent/MX9100937A/es unknown
- 1991-09-06 AT AT91202290T patent/ATE163413T1/de not_active IP Right Cessation
- 1991-09-06 EP EP91202290A patent/EP0475527B1/en not_active Expired - Lifetime
- 1991-09-06 DE DE69128949T patent/DE69128949D1/de not_active Expired - Lifetime
- 1991-09-09 RU SU5001677A patent/RU2114833C1/ru active
- 1991-09-09 JP JP3229129A patent/JPH05339246A/ja not_active Withdrawn
- 1991-09-09 CA CA002050962A patent/CA2050962A1/en not_active Abandoned
- 1991-09-10 HU HU912918A patent/HUT64313A/hu unknown
- 1991-09-10 NO NO913566A patent/NO300268B1/no unknown
- 1991-09-10 PT PT98918A patent/PT98918B/pt not_active IP Right Cessation
- 1991-09-10 MY MYPI91001641A patent/MY109430A/en unknown
- 1991-09-10 IE IE317591A patent/IE913175A1/en unknown
- 1991-09-10 FI FI914258A patent/FI914258A/fi not_active Application Discontinuation
- 1991-09-11 IL IL9945291A patent/IL99452A/en not_active IP Right Cessation
-
1993
- 1993-04-22 AU AU37069/93A patent/AU649919B2/en not_active Ceased
-
1995
- 1995-06-30 HU HU95P/P00634P patent/HU211316A9/hu unknown
Also Published As
Publication number | Publication date |
---|---|
TW245719B (ko) | 1995-04-21 |
JPH05339246A (ja) | 1993-12-21 |
NO300268B1 (no) | 1997-05-05 |
HU211316A9 (en) | 1995-11-28 |
HU912918D0 (en) | 1992-01-28 |
EP0475527B1 (en) | 1998-02-25 |
EP0475527A3 (en) | 1992-06-17 |
MY109430A (en) | 1997-01-31 |
AU8264191A (en) | 1992-03-12 |
AU639821B2 (en) | 1993-08-05 |
EP0475527A2 (en) | 1992-03-18 |
ATE163413T1 (de) | 1998-03-15 |
AU3706993A (en) | 1993-07-29 |
FI914258A0 (fi) | 1991-09-10 |
RU2114833C1 (ru) | 1998-07-10 |
PT98918B (pt) | 1999-03-31 |
PT98918A (pt) | 1992-07-31 |
DE69128949D1 (de) | 1998-04-02 |
NZ239407A (en) | 1994-06-27 |
NO913566D0 (no) | 1991-09-10 |
IE913175A1 (en) | 1992-03-11 |
MX9100937A (es) | 1992-05-04 |
HUT64313A (en) | 1993-12-28 |
CA2050962A1 (en) | 1992-03-11 |
IL99452A (en) | 1996-12-05 |
IL99452A0 (en) | 1992-08-18 |
NO913566L (no) | 1992-03-11 |
AU649919B2 (en) | 1994-06-02 |
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Legal Events
Date | Code | Title | Description |
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HC | Name/ company changed in application |
Owner name: SANOFI |
|
GB | Transfer or assigment of application |
Owner name: SANOFI |
|
FD | Application lapsed |