FI903971A0 - Peptid med bradykinin antagonistverkan. - Google Patents

Peptid med bradykinin antagonistverkan.

Info

Publication number
FI903971A0
FI903971A0 FI903971A FI903971A FI903971A0 FI 903971 A0 FI903971 A0 FI 903971A0 FI 903971 A FI903971 A FI 903971A FI 903971 A FI903971 A FI 903971A FI 903971 A0 FI903971 A0 FI 903971A0
Authority
FI
Finland
Prior art keywords
amino acid
direct bond
bradykinin
peptides
bradykin
Prior art date
Application number
FI903971A
Other languages
English (en)
Other versions
FI102759B (fi
FI102759B1 (fi
Inventor
Stephan Henke
Gerhard Breipohl
Jochen Knolle
Bernward Schoelkens
Hermann Gerhards
Original Assignee
Hoechst Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Hoechst Ag filed Critical Hoechst Ag
Publication of FI903971A0 publication Critical patent/FI903971A0/fi
Application granted granted Critical
Publication of FI102759B publication Critical patent/FI102759B/fi
Publication of FI102759B1 publication Critical patent/FI102759B1/fi

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K7/00Peptides having 5 to 20 amino acids in a fully defined sequence; Derivatives thereof
    • C07K7/04Linear peptides containing only normal peptide links
    • C07K7/06Linear peptides containing only normal peptide links having 5 to 11 amino acids
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K7/00Peptides having 5 to 20 amino acids in a fully defined sequence; Derivatives thereof
    • C07K7/04Linear peptides containing only normal peptide links
    • C07K7/18Kallidins; Bradykinins; Related peptides
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00Medicinal preparations containing peptides

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Biochemistry (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Molecular Biology (AREA)
  • Genetics & Genomics (AREA)
  • Biophysics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Peptides Or Proteins (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)
FI903971A 1989-08-14 1990-08-10 Menetelmä terapeuttisesti aktiivisten nona- ja dekapeptidien valmistamiseksi FI102759B1 (fi)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE3926822A DE3926822A1 (de) 1989-08-14 1989-08-14 Peptide mit bradykinin-antagonistischer wirkung

Publications (3)

Publication Number Publication Date
FI903971A0 true FI903971A0 (fi) 1990-08-10
FI102759B FI102759B (fi) 1999-02-15
FI102759B1 FI102759B1 (fi) 1999-02-15

Family

ID=6387091

Family Applications (1)

Application Number Title Priority Date Filing Date
FI903971A FI102759B1 (fi) 1989-08-14 1990-08-10 Menetelmä terapeuttisesti aktiivisten nona- ja dekapeptidien valmistamiseksi

Country Status (24)

Country Link
EP (1) EP0413277B1 (fi)
JP (1) JP2997519B2 (fi)
KR (1) KR0173976B1 (fi)
CN (1) CN1034577C (fi)
AT (1) ATE114320T1 (fi)
AU (1) AU638735B2 (fi)
CA (1) CA2023194C (fi)
CY (1) CY2029A (fi)
CZ (1) CZ284783B6 (fi)
DD (1) DD297169A5 (fi)
DE (2) DE3926822A1 (fi)
DK (1) DK0413277T3 (fi)
ES (1) ES2065445T3 (fi)
FI (1) FI102759B1 (fi)
HU (1) HU208324B (fi)
IE (1) IE65356B1 (fi)
IL (1) IL95357A (fi)
LT (1) LT3868B (fi)
NO (1) NO178433C (fi)
NZ (1) NZ234861A (fi)
PT (1) PT94982B (fi)
RU (1) RU2081880C1 (fi)
SK (1) SK280787B6 (fi)
ZA (1) ZA906381B (fi)

Families Citing this family (20)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE4013270A1 (de) * 1990-04-26 1991-10-31 Hoechst Ag Peptide mit bradykinin-antagonistischer wirkung
EP0586613A4 (en) * 1991-04-01 1994-08-24 Cortech Inc Bradykinin antagonists
EP0618810B1 (en) * 1991-04-19 2001-07-04 Scios Nova Inc. Bradykinin antagonist peptides
ATE169823T1 (de) 1991-04-19 1998-09-15 Scios Nova Inc Bradykinin typische peptide
US6770741B1 (en) 1991-04-19 2004-08-03 Scios Inc. Bradykinin antagonist peptides
US5380875A (en) * 1991-06-06 1995-01-10 Hitachi Chemical Company, Ltd. Hydroxyproline derivatives and preparative process therefor
WO1993011789A1 (en) 1991-12-12 1993-06-24 Scios Nova Inc. Modified position (7) bradykinin antagonist peptides
TW199863B (fi) * 1991-12-21 1993-02-11 Hoechst Ag
TW258739B (fi) * 1992-04-04 1995-10-01 Hoechst Ag
US5521158A (en) * 1992-10-08 1996-05-28 Scios Nova Inc. Pseudopeptide bradykinin receptor antagonists
US5541286A (en) * 1992-10-08 1996-07-30 Scios Nova Inc. Bradykinin antagonist pseudopeptide derivatives of olefinic aminoalkanoic acids
US5686565A (en) * 1992-10-08 1997-11-11 Scios Inc. Bradykinin antagonist pseudopeptide derivatives of aminoalkanoic acids and related olefins
US5610142A (en) * 1992-10-08 1997-03-11 Scios Inc. Bradykinin antagonist pseudopeptide derivatives of substituted 4-keto-1,3,8-triazaspiro[4.5]decan-3-alkanoic acids
WO1994019372A1 (en) * 1993-02-17 1994-09-01 Scios Nova Inc. Cyclic bradykinin antagonist peptides
US5817756A (en) * 1993-09-09 1998-10-06 Scios Inc. Pseudo- and non-peptide bradykinin receptor antagonists
FR2739553B1 (fr) 1995-10-06 1998-01-02 Oreal Utilisation d'antagonistes de la bradykinine pour stimuler ou induire la pousse des cheveux et/ou stopper leur chute
DE19612067A1 (de) * 1996-03-27 1997-10-02 Hoechst Ag Verwendung von Bradykinin-Antagonisten zur Herstellung von Arzneimitteln zur Behandlung von chronisch fibrogenetischen Lebererkrankungen und akuten Lebererkrankungen
FR2756566B1 (fr) * 1996-12-04 1999-01-08 Fournier Ind & Sante Peptides agonistes du recepteur b2 de la bradykinine, procede de preparation et utilisation en therapeutique
MXPA06014754A (es) * 2004-06-17 2007-06-22 Infinity Pharmaceuticals Inc Compuestos y metodos para inhibir la interaccion de las proteinas bcl con los componentes de enlace.
KR101707887B1 (ko) * 2016-11-22 2017-02-17 홍인석 방향제 시트가 부착된 포장지 제조장치 및 제조방법

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4693993A (en) 1985-06-13 1987-09-15 Stewart John M Bradykinin antagonist peptides
DE3618218A1 (de) 1986-05-30 1987-12-03 Hoechst Ag Aminosaeure-oobt-ester, verfahren zu deren herstellung und deren verwendung
DE3635670A1 (de) 1986-10-21 1988-04-28 Hoechst Ag Synthese von peptid-aminoalkylamiden und peptidhydraziden mittels festphasenmethode
US4923963A (en) * 1987-09-02 1990-05-08 Nova Technology Limited Partnership Bradykinin antagonist peptides
WO1989001780A1 (en) * 1987-09-02 1989-03-09 Stewart John M Bradykinin antagonist peptides

Also Published As

Publication number Publication date
HUT54712A (en) 1991-03-28
IE65356B1 (en) 1995-10-18
AU638735B2 (en) 1993-07-08
DE59007747D1 (de) 1995-01-05
KR910004662A (ko) 1991-03-29
NZ234861A (en) 1992-09-25
EP0413277A1 (de) 1991-02-20
DK0413277T3 (da) 1995-04-18
LT3868B (en) 1996-04-25
CS397990A3 (en) 1992-03-18
LTIP1466A (en) 1995-06-26
CY2029A (en) 1998-02-20
IL95357A0 (en) 1991-06-30
DE3926822A1 (de) 1991-02-21
RU2081880C1 (ru) 1997-06-20
NO178433B (no) 1995-12-18
CZ284783B6 (cs) 1999-03-17
NO903545L (no) 1991-02-15
CN1049505A (zh) 1991-02-27
PT94982A (pt) 1991-04-18
FI102759B (fi) 1999-02-15
CA2023194C (en) 2001-09-11
JP2997519B2 (ja) 2000-01-11
FI102759B1 (fi) 1999-02-15
IE902923A1 (en) 1991-02-27
EP0413277B1 (de) 1994-11-23
PT94982B (pt) 1997-04-30
CN1034577C (zh) 1997-04-16
ZA906381B (en) 1991-05-29
SK280787B6 (sk) 2000-07-11
JPH0386898A (ja) 1991-04-11
HU904989D0 (en) 1991-01-28
NO903545D0 (no) 1990-08-13
ES2065445T3 (es) 1995-02-16
KR0173976B1 (ko) 1999-02-01
NO178433C (no) 1996-03-27
IL95357A (en) 1995-08-31
AU6092490A (en) 1991-02-21
CA2023194A1 (en) 1991-02-15
DD297169A5 (de) 1992-01-02
HU208324B (en) 1993-09-28
ATE114320T1 (de) 1994-12-15

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FI893738A (fi) Menetelmä terapeuttisesti käyttökelpoisen bradykiniiniantagonistin valmistamiseksi
FI903971A0 (fi) Peptid med bradykinin antagonistverkan.
ES2099102T3 (es) Peptidos con accion antagonista de la bradiquinina.

Legal Events

Date Code Title Description
FG Patent granted

Owner name: HOECHST AKTIENGESELLSCHAFT