FI901199A7 - Uusia steroidi-dioleja, niitä sisältäviä farmaseuttisia yhdistelmiä ja menetelmä niiden valmistamiseksi - Google Patents

Uusia steroidi-dioleja, niitä sisältäviä farmaseuttisia yhdistelmiä ja menetelmä niiden valmistamiseksi Download PDF

Info

Publication number
FI901199A7
FI901199A7 FI901199A FI901199A FI901199A7 FI 901199 A7 FI901199 A7 FI 901199A7 FI 901199 A FI901199 A FI 901199A FI 901199 A FI901199 A FI 901199A FI 901199 A7 FI901199 A7 FI 901199A7
Authority
FI
Finland
Prior art keywords
preparation
pharmaceutical compositions
compositions containing
novel steroid
diols
Prior art date
Application number
FI901199A
Other languages
English (en)
Finnish (fi)
Swedish (sv)
Other versions
FI901199A0 (fi
Inventor
György Fekete
György Hajos
Csaba Molnar
Laszlo Szporny
Jozef Toth
Arpad Kiraly
Nee Mezei Anna Boor
Janos Csörgei
Krisztina Szekely
Lilla Forgacs
Bulcsu Herenyi
Sandor Holly
Jozsef Szuyog
Original Assignee
Richter Gedeon Vegyeszeti Gyar R T
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Richter Gedeon Vegyeszeti Gyar R T filed Critical Richter Gedeon Vegyeszeti Gyar R T
Publication of FI901199A0 publication Critical patent/FI901199A0/fi
Publication of FI901199A7 publication Critical patent/FI901199A7/fi

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07JSTEROIDS
    • C07J5/00Normal steroids containing carbon, hydrogen, halogen or oxygen, substituted in position 17 beta by a chain of two carbon atoms, e.g. pregnane and substituted in position 21 by only one singly bound oxygen atom, i.e. only one oxygen bound to position 21 by a single bond
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07JSTEROIDS
    • C07J5/00Normal steroids containing carbon, hydrogen, halogen or oxygen, substituted in position 17 beta by a chain of two carbon atoms, e.g. pregnane and substituted in position 21 by only one singly bound oxygen atom, i.e. only one oxygen bound to position 21 by a single bond
    • C07J5/0046Normal steroids containing carbon, hydrogen, halogen or oxygen, substituted in position 17 beta by a chain of two carbon atoms, e.g. pregnane and substituted in position 21 by only one singly bound oxygen atom, i.e. only one oxygen bound to position 21 by a single bond substituted in position 17 alfa
    • C07J5/0061Normal steroids containing carbon, hydrogen, halogen or oxygen, substituted in position 17 beta by a chain of two carbon atoms, e.g. pregnane and substituted in position 21 by only one singly bound oxygen atom, i.e. only one oxygen bound to position 21 by a single bond substituted in position 17 alfa substituted in position 16
    • C07J5/0092Normal steroids containing carbon, hydrogen, halogen or oxygen, substituted in position 17 beta by a chain of two carbon atoms, e.g. pregnane and substituted in position 21 by only one singly bound oxygen atom, i.e. only one oxygen bound to position 21 by a single bond substituted in position 17 alfa substituted in position 16 by an OH group free esterified or etherified
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07JSTEROIDS
    • C07J13/00Normal steroids containing carbon, hydrogen, halogen or oxygen having a carbon-to-carbon double bond from or to position 17
    • C07J13/005Normal steroids containing carbon, hydrogen, halogen or oxygen having a carbon-to-carbon double bond from or to position 17 with double bond in position 16 (17)

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Rheumatology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pain & Pain Management (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Steroid Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
FI901199A 1989-03-09 1990-03-09 Uusia steroidi-dioleja, niitä sisältäviä farmaseuttisia yhdistelmiä ja menetelmä niiden valmistamiseksi FI901199A7 (fi)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
HU891156A HU203562B (en) 1989-03-09 1989-03-09 Process for producing new steroide diols and pharmaceutical compositions containing them

Publications (2)

Publication Number Publication Date
FI901199A0 FI901199A0 (fi) 1990-03-09
FI901199A7 true FI901199A7 (fi) 1990-09-10

Family

ID=10953088

Family Applications (1)

Application Number Title Priority Date Filing Date
FI901199A FI901199A7 (fi) 1989-03-09 1990-03-09 Uusia steroidi-dioleja, niitä sisältäviä farmaseuttisia yhdistelmiä ja menetelmä niiden valmistamiseksi

Country Status (17)

Country Link
US (1) US5082835A (forum.php)
EP (1) EP0387091A3 (forum.php)
JP (1) JPH06104679B2 (forum.php)
KR (1) KR930009445B1 (forum.php)
CN (1) CN1045396A (forum.php)
AR (1) AR244700A1 (forum.php)
AU (1) AU623503B2 (forum.php)
CA (1) CA2011282A1 (forum.php)
EG (1) EG19411A (forum.php)
FI (1) FI901199A7 (forum.php)
HU (1) HU203562B (forum.php)
IL (1) IL93478A (forum.php)
IN (1) IN170846B (forum.php)
NO (1) NO177147C (forum.php)
PH (1) PH26676A (forum.php)
PT (1) PT93375A (forum.php)
ZA (1) ZA901752B (forum.php)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
SE9100341D0 (sv) * 1991-02-04 1991-02-04 Astra Ab Novel steroids
FR2675146A1 (fr) * 1991-04-10 1992-10-16 Roussel Uclaf Nouveaux derives sterouides de la pregna-1,4-diene-3,20-dione, leur preparation, leur application a la preparation de derives 16,17-methylene dioxy substitues et nouveaux intermediaires.
ES2347027T3 (es) 1998-05-22 2010-10-22 The Board Of Trustees Of The Leland Stanford Junior University Moleculas bifuncionales y terapias basadas en las mismas.
EP3827747A1 (en) 2005-04-28 2021-06-02 Otsuka Pharmaceutical Co., Ltd. Pharma-informatics system
US9062126B2 (en) 2005-09-16 2015-06-23 Raptor Pharmaceuticals Inc. Compositions comprising receptor-associated protein (RAP) variants specific for CR-containing proteins and uses thereof
PT3395372T (pt) 2009-02-20 2022-05-05 Enhanx Biopharm Inc Sistema de entrega de medicamentos à base de glutationa
KR101741629B1 (ko) 2009-05-06 2017-05-31 라보라토리 스킨 케어, 인크. 활성제-칼슘 포스페이트 입자 복합체를 포함하는 피부 전달 조성물 및 이들을 이용하는 방법
CN110078785A (zh) * 2019-06-04 2019-08-02 博诺康源(北京)药业科技有限公司 一种布地奈德杂质ep-ze的合成方法

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3167545A (en) * 1959-02-07 1965-01-26 Syntex Corp 16beta-methyl-16alpha, 17 alpha-dihydroxy pregnenes and the 16alpha, 17alpha-cyclic ketals and acetals thereof
US3345362A (en) * 1961-07-27 1967-10-03 Lilly Co Eli Novel pregnenolone acetonides
US4036831A (en) * 1975-10-28 1977-07-19 Steroid Development Company Establishment Trimethyl siloxane steroid intermediates
ATE85620T1 (de) * 1987-08-14 1993-02-15 Upjohn Co Verfahren zur 9-alpha-dehalogenierung von 9-alpha-steroiden.

Also Published As

Publication number Publication date
US5082835A (en) 1992-01-21
JPH06104679B2 (ja) 1994-12-21
AU5110290A (en) 1990-09-13
IN170846B (forum.php) 1992-05-30
ZA901752B (en) 1991-05-29
NO177147C (no) 1995-07-26
PT93375A (pt) 1990-11-07
EP0387091A2 (en) 1990-09-12
CN1045396A (zh) 1990-09-19
AU623503B2 (en) 1992-05-14
NO901103D0 (no) 1990-03-08
JPH02279695A (ja) 1990-11-15
KR900014422A (ko) 1990-10-23
HU203562B (en) 1991-08-28
IL93478A0 (en) 1990-11-29
EG19411A (en) 1995-01-31
AR244700A1 (es) 1993-11-30
NO901103L (no) 1990-09-10
NO177147B (no) 1995-04-18
IL93478A (en) 1994-11-11
FI901199A0 (fi) 1990-03-09
EP0387091A3 (en) 1992-05-06
CA2011282A1 (en) 1990-09-09
PH26676A (en) 1992-09-15
KR930009445B1 (ko) 1993-10-04

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Legal Events

Date Code Title Description
FD Application lapsed
MM Patent lapsed

Owner name: RICHTER GEDEON VEGYESZETI GYAR R.T.