FI871123A - Pyrazolo/3,4-d/pyrimidinderivat, deras framstaellning och anvaendning. - Google Patents
Pyrazolo/3,4-d/pyrimidinderivat, deras framstaellning och anvaendning. Download PDFInfo
- Publication number
- FI871123A FI871123A FI871123A FI871123A FI871123A FI 871123 A FI871123 A FI 871123A FI 871123 A FI871123 A FI 871123A FI 871123 A FI871123 A FI 871123A FI 871123 A FI871123 A FI 871123A
- Authority
- FI
- Finland
- Prior art keywords
- pyrimidinderivat
- pyrazolo
- deras framstaellning
- framstaellning och
- och anvaendning
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
Landscapes
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Health & Medical Sciences (AREA)
- Neurosurgery (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Biomedical Technology (AREA)
- Neurology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Life Sciences & Earth Sciences (AREA)
- Hospice & Palliative Care (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Pharmacology & Pharmacy (AREA)
- Psychiatry (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
JP5792086 | 1986-03-14 | ||
JP62014627A JPS6310788A (ja) | 1986-03-14 | 1987-01-23 | 3−アミノピラゾロ〔3,4−d〕ピリミジン誘導体 |
Publications (2)
Publication Number | Publication Date |
---|---|
FI871123A0 FI871123A0 (fi) | 1987-03-13 |
FI871123A true FI871123A (fi) | 1987-09-15 |
Family
ID=26350608
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
FI871123A FI871123A (fi) | 1986-03-14 | 1987-03-13 | Pyrazolo/3,4-d/pyrimidinderivat, deras framstaellning och anvaendning. |
Country Status (8)
Country | Link |
---|---|
US (1) | US4824848A (hu) |
EP (1) | EP0237289A3 (hu) |
CN (1) | CN87101864A (hu) |
DK (1) | DK122587A (hu) |
FI (1) | FI871123A (hu) |
HU (1) | HU197749B (hu) |
NO (1) | NO164542C (hu) |
PT (1) | PT84478B (hu) |
Families Citing this family (15)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
EP0353941A3 (en) * | 1988-08-02 | 1991-05-02 | Takeda Chemical Industries, Ltd. | Medicament for psoriasis containing derivatives of 3-aminopyrazolo [3,4-d]pyrimidine |
JP3116230B2 (ja) * | 1989-02-15 | 2000-12-11 | 武田薬品工業株式会社 | 三環式縮合ピリミジン誘導体 |
DE4035599A1 (de) * | 1990-11-06 | 1992-05-07 | Dresden Arzneimittel | Neue 5-(phenoxyalkanoylamino)-uracile, verfahren zu ihrer herstellung und ihre verwendung als arzneimittel |
SE9701398D0 (sv) * | 1997-04-15 | 1997-04-15 | Astra Pharma Prod | Novel compounds |
GEP20094679B (en) | 2004-03-15 | 2009-05-10 | Takeda Pharmaceuticals Co | Dipeptidyl peptidase inhibitors |
US9255099B2 (en) | 2006-06-06 | 2016-02-09 | Intra-Cellular Therapies, Inc. | Pyrazolo[3,4-D]pyrimidine-4,6(5H,7H)-diones as phosphodiesterase 1 inhibitors |
CN101969774A (zh) * | 2007-12-06 | 2011-02-09 | 细胞内治疗公司 | 有机化合物 |
MX2011005935A (es) | 2008-12-06 | 2011-12-16 | Intra Cellular Therapies Inc | Compuestos organicos. |
CN102223799A (zh) | 2008-12-06 | 2011-10-19 | 细胞内治疗公司 | 有机化合物 |
EA201170772A1 (ru) * | 2008-12-06 | 2012-03-30 | Интра-Селлулар Терапиз, Инк. | Органические соединения |
JP5894148B2 (ja) | 2010-05-31 | 2016-03-23 | イントラ−セルラー・セラピーズ・インコーポレイテッドIntra−Cellular Therapies, Inc. | 有機化合物 |
EP2575817A4 (en) | 2010-05-31 | 2014-01-08 | Intra Cellular Therapies Inc | ORGANIC CONNECTIONS |
DK3415517T3 (da) | 2012-09-28 | 2022-05-30 | Takeda Pharmaceuticals Co | Krystallinsk form af 1-(4-1-(2,6-difluorbenzyl)-5-dimethylaminomethyl-3-(6- methoxypyridazin-3-yl)-2,4-dioxo-1,2,3,4-tetrahydrothieno(2,3-d)-pyrimidin- 6yl)phenyl)-3-methoxyurea |
US9546175B2 (en) | 2014-08-07 | 2017-01-17 | Intra-Cellular Therapies, Inc. | Organic compounds |
RU2595038C1 (ru) | 2015-04-03 | 2016-08-20 | Виктор Вениаминович Тец | Лекарственное средство с противовирусной активностью (варианты) |
Family Cites Families (4)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US3098075A (en) * | 1956-02-10 | 1963-07-16 | Ciba Geigy Corp | New pyrazolo-pyrimidines |
DE1186466B (de) * | 1962-07-18 | 1965-02-04 | Robugen Gmbh | Verfahren zur Herstellung von 4, 6-Dioxo-4, 5, 6, 7-tetrahydro-pyrazolo [3, 4-d] pyrimidinen |
JPS5761757B2 (hu) * | 1974-01-05 | 1982-12-25 | Hisamitsu Pharmaceutical Co | |
US4603203A (en) * | 1983-12-14 | 1986-07-29 | Takeda Chemical Industries, Ltd. | 3-aminopyrazolo[3,4-d]pyrimidine derivatives and production thereof |
-
1987
- 1987-03-06 EP EP87301950A patent/EP0237289A3/en not_active Withdrawn
- 1987-03-10 DK DK122587A patent/DK122587A/da not_active Application Discontinuation
- 1987-03-12 NO NO871024A patent/NO164542C/no unknown
- 1987-03-13 PT PT84478A patent/PT84478B/pt not_active IP Right Cessation
- 1987-03-13 FI FI871123A patent/FI871123A/fi not_active Application Discontinuation
- 1987-03-13 HU HU871116A patent/HU197749B/hu not_active IP Right Cessation
- 1987-03-13 CN CN198787101864A patent/CN87101864A/zh active Pending
- 1987-03-13 US US07/025,622 patent/US4824848A/en not_active Expired - Fee Related
Also Published As
Publication number | Publication date |
---|---|
EP0237289A3 (en) | 1988-07-27 |
NO871024L (no) | 1987-09-15 |
EP0237289A2 (en) | 1987-09-16 |
US4824848A (en) | 1989-04-25 |
HUT45529A (en) | 1988-07-28 |
HU197749B (en) | 1989-05-29 |
DK122587A (da) | 1987-09-15 |
PT84478A (en) | 1987-04-01 |
NO164542C (no) | 1990-10-17 |
NO871024D0 (no) | 1987-03-12 |
PT84478B (pt) | 1989-11-10 |
DK122587D0 (da) | 1987-03-10 |
FI871123A0 (fi) | 1987-03-13 |
CN87101864A (zh) | 1987-11-18 |
NO164542B (no) | 1990-07-09 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
FD | Application lapsed |
Owner name: TAKEDA CHEMICAL INDUSTRIES, LTD. |