FI812469L - Synergistisk foerening av (r s)alfa-fluormetylhistidin och simetidin som saorbildning foerhindrande aemnen - Google Patents

Synergistisk foerening av (r s)alfa-fluormetylhistidin och simetidin som saorbildning foerhindrande aemnen

Info

Publication number
FI812469L
FI812469L FI812469A FI812469A FI812469L FI 812469 L FI812469 L FI 812469L FI 812469 A FI812469 A FI 812469A FI 812469 A FI812469 A FI 812469A FI 812469 L FI812469 L FI 812469L
Authority
FI
Finland
Prior art keywords
simetidin
saorbildning
fluormethylhistidine
foerening
foerhindrande
Prior art date
Application number
FI812469A
Other languages
English (en)
Finnish (fi)
Inventor
Janos Kollonitsch
Original Assignee
Merck & Co Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Merck & Co Inc filed Critical Merck & Co Inc
Publication of FI812469L publication Critical patent/FI812469L/fi

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/4151,2-Diazoles
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/04Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants

Landscapes

  • Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Chemical & Material Sciences (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
FI812469A 1980-08-18 1981-08-10 Synergistisk foerening av (r s)alfa-fluormetylhistidin och simetidin som saorbildning foerhindrande aemnen FI812469L (fi)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US17935880A 1980-08-18 1980-08-18

Publications (1)

Publication Number Publication Date
FI812469L true FI812469L (fi) 1982-02-19

Family

ID=22656255

Family Applications (1)

Application Number Title Priority Date Filing Date
FI812469A FI812469L (fi) 1980-08-18 1981-08-10 Synergistisk foerening av (r s)alfa-fluormetylhistidin och simetidin som saorbildning foerhindrande aemnen

Country Status (8)

Country Link
EP (1) EP0046290B1 (ja)
JP (1) JPS5759812A (ja)
AU (1) AU7398381A (ja)
DD (1) DD200404A5 (ja)
DE (1) DE3168036D1 (ja)
FI (1) FI812469L (ja)
GR (1) GR74627B (ja)
PT (1) PT73517B (ja)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4447443A (en) * 1982-11-15 1984-05-08 Merck & Co., Inc. Anti-inflammatory/analgesic combination of α-fluoromethylhistidine and a selected non-steroidal anti-inflammatory drug (NSAID)
US5030645A (en) * 1990-10-15 1991-07-09 Merck & Co., Inc. Method of treating asthma using (S)-α-fluoromethyl-histidine and esters thereof
FR2822709B1 (fr) * 2001-03-30 2007-01-19 Antialis Composition pharmaceutique anti-allergique comprenant au moins un allergene et au moins un compose antihistaminique
FR2896156A1 (fr) * 2006-01-17 2007-07-20 Gaetan Terrasse Nouvelle utilisation de la tritoqualine en association avec des substances medicamenteuses antagonistes du recepteur h2 a l'histamine,pour le traitement des maladies inflammatoires digestives
US8207292B2 (en) * 2007-02-12 2012-06-26 Michalis Nicolaou Treatment of COPD, gastro-esophageal reflux disease (GERD), food allergies and other gastrointestinal conditions and disorders ameliorated by proper histamine management using a combination of histidine decarboxylase inhibitors, LRA drugs, anti-H1 and/or anti-H2 drugs

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4000302A (en) * 1972-04-20 1976-12-28 Smith Kline & French Laboratories Limited Pharmaceutical compositions and methods of inhibiting H-1 and H-2 histamine receptors
US4215221A (en) * 1977-06-01 1980-07-29 Merck & Co., Inc. Fluorination process

Also Published As

Publication number Publication date
PT73517A (en) 1981-09-01
JPS5759812A (en) 1982-04-10
PT73517B (en) 1983-07-06
AU7398381A (en) 1982-02-25
GR74627B (ja) 1984-06-29
EP0046290A1 (en) 1982-02-24
EP0046290B1 (en) 1985-01-02
DD200404A5 (de) 1983-05-04
JPH0154326B2 (ja) 1989-11-17
DE3168036D1 (en) 1985-02-14

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Legal Events

Date Code Title Description
FD Application lapsed

Owner name: MERCK & CO INC