FI73988B - Foerfarande foer framstaellning av nya kardiotoniskt verkande pyridinyl-2-pyrimidinaminderivat. - Google Patents

Foerfarande foer framstaellning av nya kardiotoniskt verkande pyridinyl-2-pyrimidinaminderivat.

Info

Publication number
FI73988B
FI73988B FI851112A FI851112A FI73988B FI 73988 B FI73988 B FI 73988B FI 851112 A FI851112 A FI 851112A FI 851112 A FI851112 A FI 851112A FI 73988 B FI73988 B FI 73988B
Authority
FI
Finland
Prior art keywords
pyrimidinaminderivat
kardiotoniskt
verkande
nya
pyridinyl
Prior art date
Application number
FI851112A
Other languages
English (en)
Other versions
FI851112A0 (fi
FI73988C (fi
FI851112L (fi
Inventor
George Yohe Lesher
Baldev Singh
Original Assignee
Sterling Drug Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Sterling Drug Inc filed Critical Sterling Drug Inc
Publication of FI851112A0 publication Critical patent/FI851112A0/fi
Publication of FI851112L publication Critical patent/FI851112L/fi
Publication of FI73988B publication Critical patent/FI73988B/fi
Application granted granted Critical
Publication of FI73988C publication Critical patent/FI73988C/fi

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/04Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pyridine Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
FI851112A 1983-07-25 1985-03-20 Foerfarande foer framstaellning av nya kardiotoniskt verkande pyridinyl-2-pyrimidinaminderivat. FI73988C (fi)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
US51682083 1983-07-25
US06/516,820 US4512993A (en) 1983-07-25 1983-07-25 4(Or 5)-(pyridinyl)-2-pyrimidinamines and cardiotonic use thereof
US8401051 1984-06-29
PCT/US1984/001051 WO1985000604A1 (en) 1983-07-25 1984-06-29 Pyridinyl-2-pyrimidinamines useful as cardiotonics and preparation thereof

Publications (4)

Publication Number Publication Date
FI851112A0 FI851112A0 (fi) 1985-03-20
FI851112L FI851112L (fi) 1985-03-20
FI73988B true FI73988B (fi) 1987-08-31
FI73988C FI73988C (fi) 1987-12-10

Family

ID=24057230

Family Applications (1)

Application Number Title Priority Date Filing Date
FI851112A FI73988C (fi) 1983-07-25 1985-03-20 Foerfarande foer framstaellning av nya kardiotoniskt verkande pyridinyl-2-pyrimidinaminderivat.

Country Status (14)

Country Link
US (1) US4512993A (fi)
EP (1) EP0150206A4 (fi)
JP (1) JPS60501952A (fi)
KR (1) KR850001192A (fi)
AU (1) AU561765B2 (fi)
DK (1) DK127385D0 (fi)
FI (1) FI73988C (fi)
IL (1) IL72307A (fi)
IT (1) IT1176419B (fi)
NO (1) NO851066L (fi)
NZ (1) NZ208818A (fi)
PH (1) PH20211A (fi)
WO (1) WO1985000604A1 (fi)
ZA (1) ZA845263B (fi)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4876252A (en) * 1986-01-13 1989-10-24 American Cyanamid Company 4,5,6-substituted-N-(substituted-phenyl)-2-pyrimidinamines
US4788195A (en) * 1986-01-13 1988-11-29 American Cyanamid Company 4,5,6-substituted-N-(substituted-phenyl)-2-pyrimidinamines
ES2087056T3 (es) * 1986-01-13 1996-07-16 American Cyanamid Co 2-pirimidinaminas sustituidas en las posiciones 4, 5 y 6.
US5952331A (en) * 1996-05-23 1999-09-14 Syntex (Usa) Inc. Aryl pyrimidine derivatives
US5958934A (en) * 1996-05-23 1999-09-28 Syntex (U.S.A.) Inc. Aryl pyrimidine derivatives and uses thereof
TW440563B (en) * 1996-05-23 2001-06-16 Hoffmann La Roche Aryl pyrimidine derivatives and a pharmaceutical composition thereof
USRE43932E1 (en) 1997-07-18 2013-01-15 Novartis Ag Crystal modification of a N-phenyl-2-pyrimidineamine derivative, processes for its manufacture and its use
CO4940418A1 (es) 1997-07-18 2000-07-24 Novartis Ag Modificacion de cristal de un derivado de n-fenil-2- pirimidinamina, procesos para su fabricacion y su uso
WO2009007187A1 (de) * 2007-07-09 2009-01-15 Basf Se Substituierte 5-hetarylpyrimidine

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US30024A (en) * 1860-09-11 Chaeles b
US4086233A (en) * 1976-07-23 1978-04-25 Sterling Drug Inc. 4-(Substituted-amino)-2-(pyridinyl) pyrimidine derivatives
US4018770A (en) 1975-03-03 1977-04-19 Sterling Drug Inc. N-(2-(pyridinyl)-4-pyrimidinyl)-aminomethylenemalonates and analogs

Also Published As

Publication number Publication date
AU561765B2 (en) 1987-05-14
PH20211A (en) 1986-10-20
IT8421939A1 (it) 1986-01-18
KR850001192A (ko) 1985-03-16
DK127385A (da) 1985-03-21
DK127385D0 (da) 1985-03-21
EP0150206A4 (en) 1986-03-18
IT8421939A0 (it) 1984-07-18
FI851112A0 (fi) 1985-03-20
NO851066L (no) 1985-03-18
IL72307A (en) 1987-12-20
ZA845263B (en) 1985-02-27
FI73988C (fi) 1987-12-10
EP0150206A1 (en) 1985-08-07
IL72307A0 (en) 1984-11-30
IT1176419B (it) 1987-08-18
FI851112L (fi) 1985-03-20
WO1985000604A1 (en) 1985-02-14
JPS60501952A (ja) 1985-11-14
US4512993A (en) 1985-04-23
AU3153084A (en) 1985-03-04
NZ208818A (en) 1988-02-12

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Legal Events

Date Code Title Description
MM Patent lapsed

Owner name: STERLING DRUG INC