FI58636C - Foerfarande foer framstaellning av butyrofenonderivat - Google Patents

Foerfarande foer framstaellning av butyrofenonderivat Download PDF

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Publication number
FI58636C
FI58636C FI82473A FI82473A FI58636C FI 58636 C FI58636 C FI 58636C FI 82473 A FI82473 A FI 82473A FI 82473 A FI82473 A FI 82473A FI 58636 C FI58636 C FI 58636C
Authority
FI
Finland
Prior art keywords
group
yield
fluorobutyrophenone
formula
piperidin
Prior art date
Application number
FI82473A
Other languages
English (en)
Finnish (fi)
Other versions
FI58636B (fi
Inventor
Kikuo Sasajima
Masaru Nakao
Isamu Maruyama
Keiichi Ono
Shigenari Katayama
Masaharu Takayama
Junki Katsube
Shigeho Inaba
Hisao Yamamoto
Original Assignee
Sumitomo Chemical Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from JP47027610A external-priority patent/JPS5755714B2/ja
Priority claimed from JP47057249A external-priority patent/JPS4914476A/ja
Application filed by Sumitomo Chemical Co filed Critical Sumitomo Chemical Co
Application granted granted Critical
Publication of FI58636B publication Critical patent/FI58636B/fi
Priority to FI803812A priority Critical patent/FI803812L/fi
Publication of FI58636C publication Critical patent/FI58636C/fi

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D295/00—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms
    • C07D295/04—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms
    • C07D295/10—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by doubly bound oxygen or sulphur atoms
    • C07D295/104—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by doubly bound oxygen or sulphur atoms with the ring nitrogen atoms and the doubly bound oxygen or sulfur atoms attached to the same carbon chain, which is not interrupted by carbocyclic rings
    • C07D295/108—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by doubly bound oxygen or sulphur atoms with the ring nitrogen atoms and the doubly bound oxygen or sulfur atoms attached to the same carbon chain, which is not interrupted by carbocyclic rings to an acyclic saturated chain
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C45/00—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds
    • C07C45/45—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by condensation
    • C07C45/46—Friedel-Crafts reactions
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C49/00—Ketones; Ketenes; Dimeric ketenes; Ketonic chelates
    • C07C49/76—Ketones containing a keto group bound to a six-membered aromatic ring
    • C07C49/80—Ketones containing a keto group bound to a six-membered aromatic ring containing halogen
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D211/00—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
    • C07D211/04—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D211/06—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
    • C07D211/36—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D211/40—Oxygen atoms
    • C07D211/44—Oxygen atoms attached in position 4
    • C07D211/52—Oxygen atoms attached in position 4 having an aryl radical as the second substituent in position 4
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D217/00—Heterocyclic compounds containing isoquinoline or hydrogenated isoquinoline ring systems
    • C07D217/02—Heterocyclic compounds containing isoquinoline or hydrogenated isoquinoline ring systems with only hydrogen atoms or radicals containing only carbon and hydrogen atoms, directly attached to carbon atoms of the nitrogen-containing ring; Alkylene-bis-isoquinolines
    • C07D217/04—Heterocyclic compounds containing isoquinoline or hydrogenated isoquinoline ring systems with only hydrogen atoms or radicals containing only carbon and hydrogen atoms, directly attached to carbon atoms of the nitrogen-containing ring; Alkylene-bis-isoquinolines with hydrocarbon or substituted hydrocarbon radicals attached to the ring nitrogen atom
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D317/00—Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms
    • C07D317/08—Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms having the hetero atoms in positions 1 and 3
    • C07D317/10—Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms having the hetero atoms in positions 1 and 3 not condensed with other rings
    • C07D317/14—Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms having the hetero atoms in positions 1 and 3 not condensed with other rings with substituted hydrocarbon radicals attached to ring carbon atoms
    • C07D317/16—Radicals substituted by halogen atoms or nitro radicals

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pyridine Compounds (AREA)
  • Hydrogenated Pyridines (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
FI82473A 1972-03-18 1973-03-16 Foerfarande foer framstaellning av butyrofenonderivat FI58636C (fi)

Priority Applications (1)

Application Number Priority Date Filing Date Title
FI803812A FI803812L (fi) 1972-03-18 1980-12-08 Foerfarande foer framstaellning av butyrofenonderivat

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
JP47027610A JPS5755714B2 (it) 1972-03-18 1972-03-18
JP2761072 1972-03-18
JP47057249A JPS4914476A (it) 1972-06-07 1972-06-07
JP5724972 1972-06-07

Publications (2)

Publication Number Publication Date
FI58636B FI58636B (fi) 1980-11-28
FI58636C true FI58636C (fi) 1981-03-10

Family

ID=26365557

Family Applications (1)

Application Number Title Priority Date Filing Date
FI82473A FI58636C (fi) 1972-03-18 1973-03-16 Foerfarande foer framstaellning av butyrofenonderivat

Country Status (10)

Country Link
AU (1) AU470114B2 (it)
CA (1) CA1024984A (it)
CH (2) CH599939A5 (it)
FI (1) FI58636C (it)
FR (1) FR2183683B1 (it)
GB (1) GB1423576A (it)
HU (1) HU167671B (it)
NL (1) NL7303854A (it)
NO (2) NO144068C (it)
SE (1) SE419441B (it)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS595587B2 (ja) * 1974-04-18 1984-02-06 住友化学工業株式会社 シンキナブチロフエノンユウドウタイ オヨビ ソノエン ノ セイホウ
JPS5116677A (ja) * 1974-07-29 1976-02-10 Sumitomo Chemical Co Shinkinabuchirofuenonjudotai oyobi sonosanfukaennoseiho
FR2530632A1 (fr) * 1982-07-26 1984-01-27 Bouchara Emile Nouveaux derives substitues du 2,5-diamino 1,4-diazole, leurs procedes de preparation et les compositions pharmaceutiques en renfermant
US4569933A (en) * 1984-04-13 1986-02-11 Cornu Pierre Jean Antihypertensive substituted derivatives of 2,5-diamino 1,4-diazole

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB1304599A (it) * 1969-07-16 1973-01-24
SE381656B (sv) * 1970-02-06 1975-12-15 Sumitomo Chemical Co Sett for framstellning av 1,2,3,4-tetrahydroisokinolinderivat
DE2110534C3 (de) * 1970-03-06 1979-03-08 Sumitomo Chemical Co., Ltd., Osaka (Japan) γ-Piperazinobutyrophenonderivate, Verfahren zu ihrer Herstellung und Arzneipräparate
US3799932A (en) * 1970-03-20 1974-03-26 Sumitomo Chemical Co Gamma-piperidinobutyrophenones

Also Published As

Publication number Publication date
NO144069C (no) 1981-06-17
AU5346873A (en) 1974-09-19
AU470114B2 (en) 1976-03-04
NO144068C (no) 1981-06-17
CH599939A5 (it) 1978-06-15
NO144068B (no) 1981-03-09
CA1024984A (en) 1978-01-24
NL7303854A (it) 1973-09-20
FI58636B (fi) 1980-11-28
SE419441B (sv) 1981-08-03
CH589626A5 (it) 1977-07-15
HU167671B (it) 1975-11-28
GB1423576A (en) 1976-02-04
FR2183683A1 (it) 1973-12-21
FR2183683B1 (it) 1976-12-31
NO144069B (no) 1981-03-09

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FI58636C (fi) Foerfarande foer framstaellning av butyrofenonderivat