FI49302C - Menetelmä sepelvaltimoa laajentavien N6-bentsyyli-adenosiini-johdannai sten valmistamiseksi. - Google Patents
Menetelmä sepelvaltimoa laajentavien N6-bentsyyli-adenosiini-johdannai sten valmistamiseksi.Info
- Publication number
- FI49302C FI49302C FI673279A FI327967A FI49302C FI 49302 C FI49302 C FI 49302C FI 673279 A FI673279 A FI 673279A FI 327967 A FI327967 A FI 327967A FI 49302 C FI49302 C FI 49302C
- Authority
- FI
- Finland
- Prior art keywords
- benzyl
- preparation
- adenosine derivatives
- coronary dilating
- dilating
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
- C07H19/00—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof
- C07H19/02—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof sharing nitrogen
- C07H19/04—Heterocyclic radicals containing only nitrogen atoms as ring hetero atom
- C07H19/16—Purine radicals
-
- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
- Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
- Y02P20/00—Technologies relating to chemical industry
- Y02P20/50—Improvements relating to the production of bulk chemicals
- Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
DEB0090219 | 1966-12-09 | ||
DEB0093416 | 1967-07-11 |
Publications (2)
Publication Number | Publication Date |
---|---|
FI49302B FI49302B (fi) | 1975-01-31 |
FI49302C true FI49302C (fi) | 1975-05-12 |
Family
ID=25968244
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
FI673279A FI49302C (fi) | 1966-12-09 | 1967-12-07 | Menetelmä sepelvaltimoa laajentavien N6-bentsyyli-adenosiini-johdannai sten valmistamiseksi. |
Country Status (8)
Country | Link |
---|---|
US (1) | US3506643A (fi) |
AT (2) | AT277475B (fi) |
CH (2) | CH509326A (fi) |
FI (1) | FI49302C (fi) |
FR (2) | FR1550512A (fi) |
GB (1) | GB1145789A (fi) |
NL (1) | NL130339C (fi) |
SE (1) | SE323383B (fi) |
Families Citing this family (23)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
DE2007273A1 (de) * | 1970-02-18 | 1971-08-26 | Boehnnger Mannheim GmbH, 6800 Mann heim Waldhof | N(6) Aralkyl adenosin Derivate und Verfahren zur Herstellung derselben |
DE2244328A1 (de) * | 1972-09-09 | 1974-03-21 | Boehringer Mannheim Gmbh | Neue n(6)-disubstituierte adenosinderivate und verfahren zur herstellung derselben |
US4514405A (en) * | 1981-09-17 | 1985-04-30 | Merck Patent Gesellschaft Mit Beschrankter Haftung | Use of adenosine derivatives as anticonvulsants |
US5284834A (en) * | 1985-03-29 | 1994-02-08 | The United States Of America As Represented By The Secretary Of The Department Of Health And Human Services | Adenosine functionalized congeners as cardiovascular treating agents for animals and methods for using same |
JPS63208525A (ja) * | 1987-02-25 | 1988-08-30 | Kikkoman Corp | 心不全治療剤 |
AU4772493A (en) * | 1992-07-15 | 1994-02-14 | United States Of America, Represented By The Secretary, Department Of Health And Human Services, The | Sulfo-derivatives of adenosine |
US20030187261A1 (en) * | 2000-01-07 | 2003-10-02 | Libor Havlicek | Purine derivatives, process for their preparation and use thereof |
CZ294538B6 (cs) * | 2002-12-30 | 2005-01-12 | Ústav Experimentální Botaniky Akademie Vědčeské Re | Substituční deriváty N6-benzyladenosinu, způsob jejich přípravy, jejich použití pro přípravu léčiv, kosmetických přípravků a růstových regulátorů, farmaceutické přípravky, kosmetické přípravky a růstové regulátory tyto sloučeniny obsahující |
US20070161582A1 (en) * | 2003-08-08 | 2007-07-12 | Dusan Mijikovic | Pharmaceutical compositions and methods for metabolic modulation |
JP5677425B2 (ja) | 2009-06-29 | 2015-02-25 | インサイト・コーポレイションIncyte Corporation | Pi3k阻害剤としてのピリミジノン |
WO2011075643A1 (en) * | 2009-12-18 | 2011-06-23 | Incyte Corporation | Substituted heteroaryl fused derivatives as pi3k inhibitors |
US8680108B2 (en) * | 2009-12-18 | 2014-03-25 | Incyte Corporation | Substituted fused aryl and heteroaryl derivatives as PI3K inhibitors |
CA2796311A1 (en) | 2010-04-14 | 2011-10-20 | Incyte Corporation | Fused derivatives as pi3k.delta. inhibitors |
WO2011163195A1 (en) | 2010-06-21 | 2011-12-29 | Incyte Corporation | Fused pyrrole derivatives as pi3k inhibitors |
EP2655374B1 (en) | 2010-12-20 | 2019-10-23 | Incyte Holdings Corporation | N-(1-(substituted-phenyl)ethyl)-9h-purin-6-amines as pi3k inhibitors |
WO2012125629A1 (en) | 2011-03-14 | 2012-09-20 | Incyte Corporation | Substituted diamino-pyrimidine and diamino-pyridine derivatives as pi3k inhibitors |
US9126948B2 (en) | 2011-03-25 | 2015-09-08 | Incyte Holdings Corporation | Pyrimidine-4,6-diamine derivatives as PI3K inhibitors |
KR102507287B1 (ko) | 2011-09-02 | 2023-03-07 | 인사이트 홀딩스 코포레이션 | Pi3k 억제제로서 헤테로시클릴아민 |
AR090548A1 (es) | 2012-04-02 | 2014-11-19 | Incyte Corp | Azaheterociclobencilaminas biciclicas como inhibidores de pi3k |
US10077277B2 (en) | 2014-06-11 | 2018-09-18 | Incyte Corporation | Bicyclic heteroarylaminoalkyl phenyl derivatives as PI3K inhibitors |
PE20180129A1 (es) | 2015-02-27 | 2018-01-18 | Incyte Corp | Sales de inhibidor de pi3k y procesos de preparacion |
US9988401B2 (en) | 2015-05-11 | 2018-06-05 | Incyte Corporation | Crystalline forms of a PI3K inhibitor |
US9732097B2 (en) | 2015-05-11 | 2017-08-15 | Incyte Corporation | Process for the synthesis of a phosphoinositide 3-kinase inhibitor |
Family Cites Families (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US3014900A (en) * | 1959-01-26 | 1961-12-26 | Upjohn Co | Process for the preparation of ketosidopurines |
-
1967
- 1967-10-18 US US676032A patent/US3506643A/en not_active Expired - Lifetime
- 1967-12-06 CH CH588170A patent/CH509326A/de not_active IP Right Cessation
- 1967-12-06 CH CH1707167A patent/CH491119A/de not_active IP Right Cessation
- 1967-12-07 FI FI673279A patent/FI49302C/fi active
- 1967-12-07 GB GB55647/66A patent/GB1145789A/en not_active Expired
- 1967-12-07 AT AT06861/68A patent/AT277475B/de active
- 1967-12-07 AT AT1110667A patent/AT276640B/de active
- 1967-12-08 NL NL6716737A patent/NL130339C/xx active
- 1967-12-08 SE SE16895/67A patent/SE323383B/xx unknown
- 1967-12-08 FR FR131524A patent/FR1550512A/fr not_active Expired
-
1968
- 1968-03-08 FR FR142941A patent/FR7285M/fr not_active Expired
Also Published As
Publication number | Publication date |
---|---|
NL130339C (fi) | 1970-12-15 |
AT276640B (de) | 1969-11-25 |
NL6716737A (fi) | 1968-06-10 |
SE323383B (fi) | 1970-05-04 |
FR7285M (fi) | 1969-09-22 |
GB1145789A (en) | 1969-03-19 |
AT277475B (de) | 1969-12-29 |
CH491119A (de) | 1970-05-31 |
US3506643A (en) | 1970-04-14 |
CH509326A (de) | 1971-06-30 |
FI49302B (fi) | 1975-01-31 |
FR1550512A (fi) | 1968-12-20 |
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