FI104721B - Menetelmä kiraalisen etyyli-(5-amino-1,2-dihydro-2-metyyli-3-fenyylipyrido[3,4-b]pyratsin-7-yyli)karbamaatin valmistamiseksi - Google Patents

Menetelmä kiraalisen etyyli-(5-amino-1,2-dihydro-2-metyyli-3-fenyylipyrido[3,4-b]pyratsin-7-yyli)karbamaatin valmistamiseksi Download PDF

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Publication number
FI104721B
FI104721B FI943706A FI943706A FI104721B FI 104721 B FI104721 B FI 104721B FI 943706 A FI943706 A FI 943706A FI 943706 A FI943706 A FI 943706A FI 104721 B FI104721 B FI 104721B
Authority
FI
Finland
Prior art keywords
amino
carbamate
ethyl
methyl
nitro
Prior art date
Application number
FI943706A
Other languages
English (en)
Finnish (fi)
Swedish (sv)
Other versions
FI943706A (fi
FI943706A0 (fi
Inventor
Om Prakash Goel
Sham Shridhar Nikam
Original Assignee
Warner Lambert Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Warner Lambert Co filed Critical Warner Lambert Co
Publication of FI943706A publication Critical patent/FI943706A/fi
Publication of FI943706A0 publication Critical patent/FI943706A0/fi
Application granted granted Critical
Publication of FI104721B publication Critical patent/FI104721B/fi

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
    • C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D213/72—Nitrogen atoms
    • C07D213/75—Amino or imino radicals, acylated by carboxylic or carbonic acids, or by sulfur or nitrogen analogues thereof, e.g. carbamates
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Pyridine Compounds (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
FI943706A 1992-02-13 1994-08-10 Menetelmä kiraalisen etyyli-(5-amino-1,2-dihydro-2-metyyli-3-fenyylipyrido[3,4-b]pyratsin-7-yyli)karbamaatin valmistamiseksi FI104721B (fi)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
US83662492A 1992-02-13 1992-02-13
US83662492 1992-02-13
US9300467 1993-01-19
PCT/US1993/000467 WO1993016078A1 (fr) 1992-02-13 1993-01-19 PROCEDE DE PREPARATION DE (5-AMINO-1,2-DIHYDRO-2-METHYL-3-PHENYLPYRIDO[3,4-b]PYRAZIN-7-YL)CARBAMATE D'ETHYLE CHIRAL

Publications (3)

Publication Number Publication Date
FI943706A FI943706A (fi) 1994-08-10
FI943706A0 FI943706A0 (fi) 1994-08-10
FI104721B true FI104721B (fi) 2000-03-31

Family

ID=25272357

Family Applications (1)

Application Number Title Priority Date Filing Date
FI943706A FI104721B (fi) 1992-02-13 1994-08-10 Menetelmä kiraalisen etyyli-(5-amino-1,2-dihydro-2-metyyli-3-fenyylipyrido[3,4-b]pyratsin-7-yyli)karbamaatin valmistamiseksi

Country Status (12)

Country Link
US (1) US5484930A (fr)
EP (1) EP0625980A1 (fr)
JP (1) JP3208142B2 (fr)
KR (1) KR100261403B1 (fr)
AU (1) AU666705B2 (fr)
CA (1) CA2127456A1 (fr)
FI (1) FI104721B (fr)
HU (1) HU219636B (fr)
MX (1) MX9300782A (fr)
NO (1) NO302297B1 (fr)
NZ (1) NZ249022A (fr)
WO (1) WO1993016078A1 (fr)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN104211663B (zh) * 2014-08-11 2017-01-11 杭州偶联医药科技有限公司 一种(s)-n-甲氧基-甲基-2-(四氢吡咯基)丙酰胺及其制备方法和应用
CN107617194B (zh) 2016-07-14 2020-01-21 雷仁贸易有限公司 多工蹲立健身器
KR101875338B1 (ko) * 2017-10-23 2018-07-05 이현석 무릎관절을 보호하는 안전 스쿼트 운동기구

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4743585A (en) * 1986-11-21 1988-05-10 Warner-Lambert Company Renin inhibitors
US4866059A (en) * 1988-04-04 1989-09-12 Warner-Lambert Company '(2S)-(5-amino-1,2-dihydro-2-methyl-3-phenylpyrido(3,4-b)pyrazin-7-yl)-carbamic acid, ethyl ester
US5036053A (en) * 1988-05-27 1991-07-30 Warner-Lambert Company Diol-containing renin inhibitors
US5087634A (en) * 1990-10-31 1992-02-11 G. D. Searle & Co. N-substituted imidazol-2-one compounds for treatment of circulatory disorders
US5095017A (en) * 1991-05-22 1992-03-10 Southern Research Institute 1,2-dihydropyrido(3,4,-b)pyrazines as fungicides

Also Published As

Publication number Publication date
NZ249022A (en) 1996-06-25
EP0625980A1 (fr) 1994-11-30
MX9300782A (es) 1993-09-01
FI943706A (fi) 1994-08-10
FI943706A0 (fi) 1994-08-10
US5484930A (en) 1996-01-16
CA2127456A1 (fr) 1993-08-19
WO1993016078A1 (fr) 1993-08-19
KR100261403B1 (ko) 2000-07-01
AU3479093A (en) 1993-09-03
JPH07503956A (ja) 1995-04-27
HU9402350D0 (en) 1994-10-28
AU666705B2 (en) 1996-02-22
NO942964L (no) 1994-08-10
KR950700295A (ko) 1995-01-16
NO302297B1 (no) 1998-02-16
HU219636B (hu) 2001-06-28
NO942964D0 (no) 1994-08-10
JP3208142B2 (ja) 2001-09-10
HUT68185A (en) 1995-05-29

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