ES8706623A1 - Procedimiento de preparar compuestos amidicos farmacologicamente activos - Google Patents

Procedimiento de preparar compuestos amidicos farmacologicamente activos

Info

Publication number
ES8706623A1
ES8706623A1 ES554301A ES554301A ES8706623A1 ES 8706623 A1 ES8706623 A1 ES 8706623A1 ES 554301 A ES554301 A ES 554301A ES 554301 A ES554301 A ES 554301A ES 8706623 A1 ES8706623 A1 ES 8706623A1
Authority
ES
Spain
Prior art keywords
same
preparing
pharmaceutical compositions
compositions containing
ethyl
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
ES554301A
Other languages
English (en)
Other versions
ES554301A0 (es
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Taiho Pharmaceutical Co Ltd
Original Assignee
Taiho Pharmaceutical Co Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Taiho Pharmaceutical Co Ltd filed Critical Taiho Pharmaceutical Co Ltd
Publication of ES8706623A1 publication Critical patent/ES8706623A1/es
Publication of ES554301A0 publication Critical patent/ES554301A0/es
Expired legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C235/00—Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by oxygen atoms
    • C07C235/42—Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by oxygen atoms having carbon atoms of carboxamide groups bound to carbon atoms of six-membered aromatic rings and singly-bound oxygen atoms bound to the same carbon skeleton
    • C07C235/44—Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by oxygen atoms having carbon atoms of carboxamide groups bound to carbon atoms of six-membered aromatic rings and singly-bound oxygen atoms bound to the same carbon skeleton with carbon atoms of carboxamide groups and singly-bound oxygen atoms bound to carbon atoms of the same non-condensed six-membered aromatic ring
    • C07C235/56—Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by oxygen atoms having carbon atoms of carboxamide groups bound to carbon atoms of six-membered aromatic rings and singly-bound oxygen atoms bound to the same carbon skeleton with carbon atoms of carboxamide groups and singly-bound oxygen atoms bound to carbon atoms of the same non-condensed six-membered aromatic ring having the nitrogen atom of at least one of the carboxamide groups bound to a carbon atom of a six-membered aromatic ring
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/16—Amides, e.g. hydroxamic acids
    • A61K31/165—Amides, e.g. hydroxamic acids having aromatic rings, e.g. colchicine, atenolol, progabide
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/08—Antiallergic agents
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C233/00—Carboxylic acid amides
    • C07C233/01—Carboxylic acid amides having carbon atoms of carboxamide groups bound to hydrogen atoms or to acyclic carbon atoms
    • C07C233/16—Carboxylic acid amides having carbon atoms of carboxamide groups bound to hydrogen atoms or to acyclic carbon atoms having the nitrogen atom of at least one of the carboxamide groups bound to a carbon atom of a hydrocarbon radical substituted by singly-bound oxygen atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C317/00—Sulfones; Sulfoxides
    • C07C317/44—Sulfones; Sulfoxides having sulfone or sulfoxide groups and carboxyl groups bound to the same carbon skeleton
    • C07C317/48—Sulfones; Sulfoxides having sulfone or sulfoxide groups and carboxyl groups bound to the same carbon skeleton the carbon skeleton being further substituted by singly-bound nitrogen atoms, not being part of nitro or nitroso groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Epidemiology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Pulmonology (AREA)
  • Immunology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

METODO DE PREPARAR COMPUESTOS AMIDICOS. CONSISTE EN HACER REACCIONAR UN COMPUESTO HALURO DE FORMULA (II), DONDE X ES UN ATOMO DE HALOGENO, CON UN COMPUESTO TIOL DE FORMULA R3SH, DONDE R3 ES 2-ACETILAMINO-2-CARBOXIETILENO O 2-(4-AMINO-4-CARBOXIBUTIRILAMINO)-2-(CARBOXIMETILCARBAMOIL)ETILO, PARA OBTENER COMPUESTOS AMIDICOS DE FORMULA (I) DONDE R''''1 ES 2-(2-ACETILAMINO-2-CARBOXIETILTIO)ETILO O [2-(4-AMINO-4-CARBOXIBUTIRILAMINO)-2-(CARBOXIMETILCARBAMOIL)ETILTIO]ETI LO; Y R2 ES HIDROGENO O ALQUILO INFERIOR. TIENEN APLICACIONES FARMACEUTICAS POR SUS PROPIEDADES ANTIALERGICAS. *FORMULA*
ES554301A 1984-09-12 1986-04-24 Procedimiento de preparar compuestos amidicos farmacologicamente activos Expired ES8706623A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
JP59191988A JPS6168455A (ja) 1984-09-12 1984-09-12 アミド化合物

Publications (2)

Publication Number Publication Date
ES8706623A1 true ES8706623A1 (es) 1987-07-01
ES554301A0 ES554301A0 (es) 1987-07-01

Family

ID=16283753

Family Applications (2)

Application Number Title Priority Date Filing Date
ES546846A Expired ES8700653A1 (es) 1984-09-12 1985-09-10 Procedimiento de preparar compuestos amidicos farmacologica-mente activos
ES554301A Expired ES8706623A1 (es) 1984-09-12 1986-04-24 Procedimiento de preparar compuestos amidicos farmacologicamente activos

Family Applications Before (1)

Application Number Title Priority Date Filing Date
ES546846A Expired ES8700653A1 (es) 1984-09-12 1985-09-10 Procedimiento de preparar compuestos amidicos farmacologica-mente activos

Country Status (8)

Country Link
US (1) US4670583A (es)
EP (1) EP0178073B1 (es)
JP (1) JPS6168455A (es)
KR (1) KR910003007B1 (es)
AU (1) AU553738B2 (es)
CA (1) CA1256897A (es)
DE (1) DE3562370D1 (es)
ES (2) ES8700653A1 (es)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2017032384A1 (en) 2015-08-25 2017-03-02 Conrig Pharma Aps Compound and use in the treatment of cough
EP3393463B1 (en) 2015-12-23 2021-01-20 Conrig Pharma ApS Suplatast tosilate for treating cough associated with interstitial lung disease
KR20200045496A (ko) 2017-08-29 2020-05-04 콘리그 파마 에이피에스 수플라타스트 토실레이트를 포함하는 조성물
WO2024168001A1 (en) * 2023-02-07 2024-08-15 Corteva Agriscience Llc Processes related to formation of n-(4-chloro-2-(pyridin-3-yl)thiazol-5-yl)- n-ethyl-3-(methylsulfonyl)propanamide

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR1601M (fr) * 1961-10-18 1962-12-10 Ile De France Nouveaux médicaments analgésiques.
MA19111A1 (fr) * 1979-10-26 1981-12-31 Ciba Geigy Ag Derives de l'homoserine,procede pour leur preparation et leur utilisation en tant que microbicides
US4556737A (en) * 1983-03-11 1985-12-03 Taiho Pharmaceutical Company Limited Sulfonium compounds, processes for preparing the compounds and pharmacological composiitons containing the same
FI832377A0 (fi) * 1983-06-29 1983-06-29 Star Oy Ab Nytt foerfarande foer framstaellning av (r)-, (s)-eller (r,s)-1-(4'-alkylamido-2'-acetyl) fenoxi-3-alkylamino-2-propanoler

Also Published As

Publication number Publication date
KR860002451A (ko) 1986-04-26
ES546846A0 (es) 1986-11-16
AU4714885A (en) 1986-03-20
JPS6168455A (ja) 1986-04-08
EP0178073A1 (en) 1986-04-16
ES554301A0 (es) 1987-07-01
EP0178073B1 (en) 1988-04-27
AU553738B2 (en) 1986-07-24
CA1256897A (en) 1989-07-04
KR910003007B1 (ko) 1991-05-15
JPH0350748B2 (es) 1991-08-02
ES8700653A1 (es) 1986-11-16
DE3562370D1 (en) 1988-06-01
US4670583A (en) 1987-06-02

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Legal Events

Date Code Title Description
FD1A Patent lapsed

Effective date: 20000201