ES8706107A1 - Procedimiento para preparar esteres de acido n-acil-2,3-deshidroaminocarboxilico - Google Patents
Procedimiento para preparar esteres de acido n-acil-2,3-deshidroaminocarboxilicoInfo
- Publication number
- ES8706107A1 ES8706107A1 ES552839A ES552839A ES8706107A1 ES 8706107 A1 ES8706107 A1 ES 8706107A1 ES 552839 A ES552839 A ES 552839A ES 552839 A ES552839 A ES 552839A ES 8706107 A1 ES8706107 A1 ES 8706107A1
- Authority
- ES
- Spain
- Prior art keywords
- radical
- group
- polysubstituted
- halogen
- unsubstituted
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
- C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
- C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D213/78—Carbon atoms having three bonds to hetero atoms, with at the most one bond to halogen, e.g. ester or nitrile radicals
- C07D213/81—Amides; Imides
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D307/00—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom
- C07D307/02—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings
- C07D307/34—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D307/56—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D307/68—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D333/00—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
- C07D333/02—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings
- C07D333/04—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom
- C07D333/06—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to the ring carbon atoms
- C07D333/24—Radicals substituted by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D333/00—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
- C07D333/02—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings
- C07D333/04—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom
- C07D333/26—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D333/28—Halogen atoms
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Health & Medical Sciences (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Oncology (AREA)
- Pharmacology & Pharmacy (AREA)
- Communicable Diseases (AREA)
- Animal Behavior & Ethology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Cephalosporin Compounds (AREA)
- Medicines Containing Antibodies Or Antigens For Use As Internal Diagnostic Agents (AREA)
- Heterocyclic Compounds Containing Sulfur Atoms (AREA)
- Furan Compounds (AREA)
- Pyridine Compounds (AREA)
Abstract
PROCEDIMIENTO PARA LA OBTENCION DE ESTERES DE FORMULA (I). COMPRENDE LA REACCION DE UN ESTER DE ACIDO 2-AZIDOCARBOXILICO, DE FORMULA (II), CON UN HALOGENURO DE ACIDO, DE FORMULA R4COHAL, PARA OBTENER UN COMPUESTO DE FORMULA (I), EN LAS QUE HAL REPRESENTA CLORO O BROMO, R2 ES HIDROGENO O METILO Y R1, R3 Y R4 PUEDEN SER VARIOS TIPOS DE RADICALES. LA REACCION SE EFECTUA EN PRESENCIA DE UN PERRENATO, A UNA TEMPERATURA COMPRENDIDA ENTRE 0JC Y 150JC. ESTOS COMPUESTOS TIENEN APLICACIONES FARMACOLOGICAS COMO ANTIBIOTICOS.
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
DE19853508564 DE3508564A1 (de) | 1985-03-11 | 1985-03-11 | Verfahren zur herstellung von n-acyl-2, 3-dehydroaminocarbonsaeureestern |
Publications (2)
Publication Number | Publication Date |
---|---|
ES8706107A1 true ES8706107A1 (es) | 1987-06-01 |
ES552839A0 ES552839A0 (es) | 1987-06-01 |
Family
ID=6264801
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
ES552839A Expired ES8706107A1 (es) | 1985-03-11 | 1986-03-10 | Procedimiento para preparar esteres de acido n-acil-2,3-deshidroaminocarboxilico |
Country Status (6)
Country | Link |
---|---|
EP (1) | EP0195201B1 (es) |
JP (1) | JPS61212546A (es) |
AT (1) | ATE53008T1 (es) |
CA (1) | CA1277988C (es) |
DE (2) | DE3508564A1 (es) |
ES (1) | ES8706107A1 (es) |
Families Citing this family (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US5559268A (en) * | 1994-11-17 | 1996-09-24 | E. I. Du Pont De Nemours And Company | Process for the efficient preparation of N-substituted dehydroamino acid esters |
Family Cites Families (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
NZ190994A (en) * | 1978-07-24 | 1981-10-19 | Merck & Co Inc | Z-2-acylamino-3-monosubstituted propenoates |
DE3140227C1 (de) * | 1981-10-09 | 1982-12-16 | Degussa Ag, 6000 Frankfurt | Verfahren zur Herstellung von N-Acetyl-2,3-dehydro-aminocarbonsaeureestern |
-
1985
- 1985-03-11 DE DE19853508564 patent/DE3508564A1/de active Granted
-
1986
- 1986-01-27 AT AT86101048T patent/ATE53008T1/de not_active IP Right Cessation
- 1986-01-27 DE DE8686101048T patent/DE3671431D1/de not_active Expired - Lifetime
- 1986-01-27 EP EP86101048A patent/EP0195201B1/de not_active Expired - Lifetime
- 1986-03-10 ES ES552839A patent/ES8706107A1/es not_active Expired
- 1986-03-10 CA CA000503677A patent/CA1277988C/en not_active Expired - Lifetime
- 1986-03-11 JP JP61051616A patent/JPS61212546A/ja active Pending
Also Published As
Publication number | Publication date |
---|---|
EP0195201A3 (en) | 1988-01-13 |
CA1277988C (en) | 1990-12-18 |
DE3508564C2 (es) | 1988-02-18 |
ATE53008T1 (de) | 1990-06-15 |
DE3508564A1 (de) | 1986-09-11 |
JPS61212546A (ja) | 1986-09-20 |
EP0195201B1 (de) | 1990-05-23 |
DE3671431D1 (de) | 1990-06-28 |
ES552839A0 (es) | 1987-06-01 |
EP0195201A2 (de) | 1986-09-24 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
MM4A | Patent lapsed |
Effective date: 19960401 |