ES8608516A1 - Procedimiento para la preparacion de acidos 4-isoxazolil- tiazol-2-oxamicos y sus derivados - Google Patents
Procedimiento para la preparacion de acidos 4-isoxazolil- tiazol-2-oxamicos y sus derivadosInfo
- Publication number
- ES8608516A1 ES8608516A1 ES546420A ES546420A ES8608516A1 ES 8608516 A1 ES8608516 A1 ES 8608516A1 ES 546420 A ES546420 A ES 546420A ES 546420 A ES546420 A ES 546420A ES 8608516 A1 ES8608516 A1 ES 8608516A1
- Authority
- ES
- Spain
- Prior art keywords
- isoxazolyl
- thiazole
- acid derivatives
- oxamic acid
- compounds
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D261/00—Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings
- C07D261/02—Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings not condensed with other rings
- C07D261/06—Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings not condensed with other rings having two or more double bonds between ring members or between ring members and non-ring members
- C07D261/10—Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings not condensed with other rings having two or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D261/00—Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings
- C07D261/02—Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings not condensed with other rings
- C07D261/06—Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings not condensed with other rings having two or more double bonds between ring members or between ring members and non-ring members
- C07D261/08—Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings not condensed with other rings having two or more double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D261/00—Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings
- C07D261/02—Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings not condensed with other rings
- C07D261/06—Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings not condensed with other rings having two or more double bonds between ring members or between ring members and non-ring members
- C07D261/10—Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings not condensed with other rings having two or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D261/12—Oxygen atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D261/00—Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings
- C07D261/02—Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings not condensed with other rings
- C07D261/06—Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings not condensed with other rings having two or more double bonds between ring members or between ring members and non-ring members
- C07D261/10—Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings not condensed with other rings having two or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D261/18—Carbon atoms having three bonds to hetero atoms, with at the most one bond to halogen
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
- C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
- C07D417/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings directly linked by a ring-member-to-ring-member bond
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Agricultural Chemicals And Associated Chemicals (AREA)
- Thiazole And Isothizaole Compounds (AREA)
Abstract
PROCEDIMIENTO PARA PREPARAR ACIDOS 4-(ISOXAZOLIL)TIAZOL-2-OXAMICOS. CONSISTE EN HACER REACCIONAR A UN C.D.F. (II) CON UN C.D.F. (III), EN PRESENCIA DE UN DISOLVENTE INERTE Y DE UN ACEPTOR DE ACIDO Y ENTRE 50 Y 100JC, PARA OBTENER UN C.D.F. (I) Y SUS SALES FARMACEUTICAMENTE ACEPTABLES CON BASES ORGANICAS O INORGANICAS. SIENDO: R Y R1, H, HAL,HIDROXILO, UN GRUPO DE CARBONILO DE C 1 A 3 Y OTROS; R2, UN GRUPO CICLOALQUILO DE C 3 A 6 O UN GRUPO ALQUILO DE C 1 A 4; R3, H O UN GRUPO ALQUILO DE C 1 A 3; Z, UN GRUPO D.F. (IV) O (V); Y C.D.F., COMPUESTO DE FORMULA. SE UTILIZAN COMO AGENTES ANTIALERGICOS.
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
IT22150/84A IT1183061B (it) | 1984-07-31 | 1984-07-31 | Composti dotati di attivita'antiallergica |
Publications (2)
Publication Number | Publication Date |
---|---|
ES8608516A1 true ES8608516A1 (es) | 1986-07-16 |
ES546420A0 ES546420A0 (es) | 1986-07-16 |
Family
ID=11192238
Family Applications (4)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
ES546420A Expired ES8608516A1 (es) | 1984-07-31 | 1985-07-30 | Procedimiento para la preparacion de acidos 4-isoxazolil- tiazol-2-oxamicos y sus derivados |
ES546419A Expired ES8703459A1 (es) | 1984-07-31 | 1985-07-30 | Procedimiento para la preparacion de derivados de acido 4- (isoxazolil)-tiazol-2-oxamico |
ES552514A Expired ES8705434A1 (es) | 1984-07-31 | 1986-02-28 | Procedimiento para la preparacion de derivados de acido 4-(isoxazolil)-tiazol-2-oxamico |
ES552513A Expired ES8800217A1 (es) | 1984-07-31 | 1986-02-28 | Procedimiento para la preparacion de acidos 4-(isoxazolil)-tiazol-2-oxamicos y sus derivados |
Family Applications After (3)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
ES546419A Expired ES8703459A1 (es) | 1984-07-31 | 1985-07-30 | Procedimiento para la preparacion de derivados de acido 4- (isoxazolil)-tiazol-2-oxamico |
ES552514A Expired ES8705434A1 (es) | 1984-07-31 | 1986-02-28 | Procedimiento para la preparacion de derivados de acido 4-(isoxazolil)-tiazol-2-oxamico |
ES552513A Expired ES8800217A1 (es) | 1984-07-31 | 1986-02-28 | Procedimiento para la preparacion de acidos 4-(isoxazolil)-tiazol-2-oxamicos y sus derivados |
Country Status (13)
Country | Link |
---|---|
US (2) | US4766137A (es) |
EP (2) | EP0190298B1 (es) |
JP (2) | JPS61502959A (es) |
AU (2) | AU583847B2 (es) |
CA (2) | CA1243318A (es) |
DE (2) | DE3574874D1 (es) |
DK (2) | DK164364C (es) |
ES (4) | ES8608516A1 (es) |
FI (2) | FI83650C (es) |
IL (1) | IL75981A (es) |
IT (1) | IT1183061B (es) |
WO (2) | WO1986000899A1 (es) |
ZA (1) | ZA855743B (es) |
Families Citing this family (9)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
IT1183061B (it) * | 1984-07-31 | 1987-10-05 | Zambon Spa | Composti dotati di attivita'antiallergica |
IT1204960B (it) * | 1987-03-25 | 1989-03-10 | Zambon Farmaceutici Spa | Composti dotati di attivita' antiallergica |
US4946963A (en) * | 1987-11-13 | 1990-08-07 | The University Of North Carolina At Chapel Hill | Compounds for the control of hyperlipidemia using N-substituted isoxazolidine-3,5-diones |
DE3844227A1 (de) * | 1988-12-29 | 1990-07-05 | Basf Ag | 3(2h)-pyridazinonderivate, verfahren zu ihrer herstellung und ihre verwendung zur bekaempfung von schaedlingen |
DE19638667C2 (de) | 1996-09-20 | 2001-05-17 | Osram Opto Semiconductors Gmbh | Mischfarbiges Licht abstrahlendes Halbleiterbauelement mit Lumineszenzkonversionselement |
DE19625622A1 (de) * | 1996-06-26 | 1998-01-02 | Siemens Ag | Lichtabstrahlendes Halbleiterbauelement mit Lumineszenzkonversionselement |
EP1441396B1 (de) | 1996-06-26 | 2011-06-01 | OSRAM Opto Semiconductors GmbH | Licht abstrahlendes Halbleiterbauelement mit Lumineszenzkonversionselement |
EA013249B1 (ru) * | 2003-12-26 | 2010-04-30 | Киова Хакко Кирин Ко., Лтд. | Производные тиазола |
WO2007099828A1 (ja) | 2006-02-23 | 2007-09-07 | Shionogi & Co., Ltd. | 環式基で置換された含窒素複素環誘導体 |
Family Cites Families (4)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
FR2429210A1 (fr) * | 1978-06-19 | 1980-01-18 | Fabre Sa Pierre | Derives de phenyl-4 thiazolyl-2 oxamates utiles dans le traitement de l'asthme |
DE3027527A1 (de) * | 1980-07-19 | 1982-02-18 | Basf Ag, 6700 Ludwigshafen | Neue oxamidsaeure-derivate, verfahren zu ihrer herstellung und diese enthaltende therapeutische mittel |
FR2494272A1 (fr) * | 1980-11-19 | 1982-05-21 | Fabre Sa Pierre | Derives de l'acide thiazolyl-2 oxamique substitues en position 4 par un radical thienyle ou furyle, leur preparation et leur utilisation comme medicaments |
IT1183061B (it) * | 1984-07-31 | 1987-10-05 | Zambon Spa | Composti dotati di attivita'antiallergica |
-
1984
- 1984-07-31 IT IT22150/84A patent/IT1183061B/it active
-
1985
- 1985-07-30 DE DE8585903835T patent/DE3574874D1/de not_active Expired - Fee Related
- 1985-07-30 EP EP85904099A patent/EP0190298B1/en not_active Expired
- 1985-07-30 ES ES546420A patent/ES8608516A1/es not_active Expired
- 1985-07-30 DE DE8585904099T patent/DE3573781D1/de not_active Expired
- 1985-07-30 WO PCT/EP1985/000380 patent/WO1986000899A1/en active IP Right Grant
- 1985-07-30 US US06/845,694 patent/US4766137A/en not_active Expired - Lifetime
- 1985-07-30 AU AU46717/85A patent/AU583847B2/en not_active Ceased
- 1985-07-30 AU AU47248/85A patent/AU584118B2/en not_active Ceased
- 1985-07-30 EP EP85903835A patent/EP0191045B1/en not_active Expired
- 1985-07-30 WO PCT/EP1985/000381 patent/WO1986000900A1/en active IP Right Grant
- 1985-07-30 US US06/849,458 patent/US4766138A/en not_active Expired - Fee Related
- 1985-07-30 JP JP60503407A patent/JPS61502959A/ja active Granted
- 1985-07-30 ES ES546419A patent/ES8703459A1/es not_active Expired
- 1985-07-30 JP JP60503735A patent/JPS61502896A/ja active Granted
- 1985-07-30 ZA ZA855743A patent/ZA855743B/xx unknown
- 1985-07-31 CA CA000487852A patent/CA1243318A/en not_active Expired
- 1985-07-31 IL IL75981A patent/IL75981A/xx not_active IP Right Cessation
- 1985-07-31 CA CA000487853A patent/CA1246583A/en not_active Expired
-
1986
- 1986-02-28 ES ES552514A patent/ES8705434A1/es not_active Expired
- 1986-02-28 ES ES552513A patent/ES8800217A1/es not_active Expired
- 1986-03-26 DK DK141986A patent/DK164364C/da not_active IP Right Cessation
- 1986-03-26 DK DK142086A patent/DK142086A/da unknown
- 1986-03-26 FI FI861330A patent/FI83650C/fi not_active IP Right Cessation
- 1986-03-26 FI FI861329A patent/FI85473C/fi not_active IP Right Cessation
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