ES8604232A1 - Un procedimiento para la preparacion de derivados de penicilina - Google Patents

Un procedimiento para la preparacion de derivados de penicilina

Info

Publication number
ES8604232A1
ES8604232A1 ES528490A ES528490A ES8604232A1 ES 8604232 A1 ES8604232 A1 ES 8604232A1 ES 528490 A ES528490 A ES 528490A ES 528490 A ES528490 A ES 528490A ES 8604232 A1 ES8604232 A1 ES 8604232A1
Authority
ES
Spain
Prior art keywords
hydrogen
general formula
beta
hydrocarbon group
lactam antibiotics
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
ES528490A
Other languages
English (en)
Other versions
ES528490A0 (es
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Beecham Group PLC
Original Assignee
Beecham Group PLC
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Beecham Group PLC filed Critical Beecham Group PLC
Publication of ES528490A0 publication Critical patent/ES528490A0/es
Publication of ES8604232A1 publication Critical patent/ES8604232A1/es
Expired legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D241/00—Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings
    • C07D241/02—Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings not condensed with other rings
    • C07D241/06—Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings not condensed with other rings having one or two double bonds between ring members or between ring members and non-ring members
    • C07D241/08—Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings not condensed with other rings having one or two double bonds between ring members or between ring members and non-ring members with oxygen atoms directly attached to ring carbon atoms
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D499/00—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • H—ELECTRICITY
    • H10—SEMICONDUCTOR DEVICES; ELECTRIC SOLID-STATE DEVICES NOT OTHERWISE PROVIDED FOR
    • H10P—GENERIC PROCESSES OR APPARATUS FOR THE MANUFACTURE OR TREATMENT OF DEVICES COVERED BY CLASS H10
    • H10P76/00—Manufacture or treatment of masks on semiconductor bodies, e.g. by lithography or photolithography
    • H10P76/20—Manufacture or treatment of masks on semiconductor bodies, e.g. by lithography or photolithography of masks comprising organic materials
    • H10P76/204—Manufacture or treatment of masks on semiconductor bodies, e.g. by lithography or photolithography of masks comprising organic materials of organic photoresist masks
    • H10P76/2041—Photolithographic processes
    • H10P76/2043—Photolithographic processes using an anti-reflective coating

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Oncology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Communicable Diseases (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

PROCEDIMIENTO PARA LA PREPARACION DE DERIVADOS DE LA PENICILINA, DE FORMULA GENERAL (I) O UNA SAL O UN ESTER HIDROLIZABLE IN VIVO DEL MISMO FARMACEUTICAMENTE ACEPTABLE, EN LA QUE R ES HIDROGENO O ALQUILO; R1 ES HIDROGENO O UN GRUPO HIDROCARBONADO; Y R2 ES HIDROGENO O UN GRUPO HIDROCARBONADO OPCIONALMENTE SUSTITUIDO. CONSISTE EN HACER REACCIONAR UN COMPUESTO DE FORMULA GENERAL (II) CON UN DERIVADO N-ACILANTE DE UN ACIDO DE FORMULA GENERAL (III). DE APLICACION EN EL TRATAMIENTO DE INFECCIONES EN ANIMALES, ESPECIALMENTE MAMIFEROS, INCLUYENDO EL HOMBRE.
ES528490A 1982-04-29 1983-12-28 Un procedimiento para la preparacion de derivados de penicilina Expired ES8604232A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB8212525 1982-04-29

Publications (2)

Publication Number Publication Date
ES528490A0 ES528490A0 (es) 1985-06-16
ES8604232A1 true ES8604232A1 (es) 1985-06-16

Family

ID=10530083

Family Applications (2)

Application Number Title Priority Date Filing Date
ES521933A Expired ES8406076A1 (es) 1982-04-29 1983-04-28 Un procedimiento para la fabricacion de un compuesto.
ES528490A Expired ES8604232A1 (es) 1982-04-29 1983-12-28 Un procedimiento para la preparacion de derivados de penicilina

Family Applications Before (1)

Application Number Title Priority Date Filing Date
ES521933A Expired ES8406076A1 (es) 1982-04-29 1983-04-28 Un procedimiento para la fabricacion de un compuesto.

Country Status (7)

Country Link
US (1) US4540688A (es)
EP (1) EP0093564B1 (es)
JP (1) JPS58203996A (es)
AU (1) AU1398183A (es)
DE (1) DE3372208D1 (es)
ES (2) ES8406076A1 (es)
ZA (1) ZA832964B (es)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE3479731D1 (en) * 1983-07-07 1989-10-19 Beecham Group Plc Substituted phenylglycine derivatives of beta-lactam antibiotics
WO2006002474A1 (en) * 2004-07-02 2006-01-12 The Walter And Eliza Hall Institute Of Medical Research Alpha-helical mimetics

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3487074A (en) * 1966-01-14 1969-12-30 Bristol Myers Co Derivatives of 6-amino-3-penamylcarboxylic acid and 7-amino-2,2-dimethyl-cephalosporanic acid
US4229348A (en) * 1978-05-26 1980-10-21 Chugai Seiyaku Kabushiki Kaisha Penicillanic acid derivatives
DE2828261A1 (de) * 1978-06-28 1980-01-10 Thomae Gmbh Dr K Neue penicilline, ihre salze, verfahren zu ihrer herstellung und diese verbindungen enthaltende arzneimittel
US4189482A (en) * 1978-10-12 1980-02-19 E. R. Squibb & Sons, Inc. Penicillins having an imino substituted piperazindioncarbonylamino acyl sidechain
US4206116A (en) * 1978-10-16 1980-06-03 Bristol-Myers Company Novel penicillins
ZA813610B (en) * 1980-06-06 1982-06-30 Beecham Group Plc Penicillin derivatives,processes for their preparation and compositions containing them
ZA813996B (en) * 1980-06-26 1982-06-30 Beecham Group Plc Penicillin derivatives

Also Published As

Publication number Publication date
AU1398183A (en) 1983-11-03
ES528490A0 (es) 1985-06-16
EP0093564B1 (en) 1987-06-24
ES521933A0 (es) 1984-07-01
JPS58203996A (ja) 1983-11-28
DE3372208D1 (en) 1987-07-30
US4540688A (en) 1985-09-10
ES8406076A1 (es) 1984-07-01
EP0093564A1 (en) 1983-11-09
ZA832964B (en) 1984-03-28

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