ES8506566A1 - Procedimiento para la produccion de derivados de 1-carbonil-1-fenil-2-azolil-etanol - Google Patents

Procedimiento para la produccion de derivados de 1-carbonil-1-fenil-2-azolil-etanol

Info

Publication number
ES8506566A1
ES8506566A1 ES527439A ES527439A ES8506566A1 ES 8506566 A1 ES8506566 A1 ES 8506566A1 ES 527439 A ES527439 A ES 527439A ES 527439 A ES527439 A ES 527439A ES 8506566 A1 ES8506566 A1 ES 8506566A1
Authority
ES
Spain
Prior art keywords
alkyl
unsubstituted
carbonyl
plant growth
phenyl
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
ES527439A
Other languages
English (en)
Other versions
ES527439A0 (es
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Novartis AG
Original Assignee
Ciba Geigy AG
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Ciba Geigy AG filed Critical Ciba Geigy AG
Publication of ES527439A0 publication Critical patent/ES527439A0/es
Publication of ES8506566A1 publication Critical patent/ES8506566A1/es
Expired legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
    • C07D405/10—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a carbon chain containing aromatic rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/12—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/48—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with two nitrogen atoms as the only ring hetero atoms
    • A01N43/50—1,3-Diazoles; Hydrogenated 1,3-diazoles
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/64—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with three nitrogen atoms as the only ring hetero atoms
    • A01N43/647—Triazoles; Hydrogenated triazoles
    • A01N43/653—1,2,4-Triazoles; Hydrogenated 1,2,4-triazoles
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/10—Antimycotics
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C45/00—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds
    • C07C45/61—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by reactions not involving the formation of >C = O groups
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C45/00—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds
    • C07C45/61—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by reactions not involving the formation of >C = O groups
    • C07C45/67—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by reactions not involving the formation of >C = O groups by isomerisation; by change of size of the carbon skeleton
    • C07C45/68—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by reactions not involving the formation of >C = O groups by isomerisation; by change of size of the carbon skeleton by increase in the number of carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C45/00—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds
    • C07C45/61—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by reactions not involving the formation of >C = O groups
    • C07C45/67—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by reactions not involving the formation of >C = O groups by isomerisation; by change of size of the carbon skeleton
    • C07C45/68—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by reactions not involving the formation of >C = O groups by isomerisation; by change of size of the carbon skeleton by increase in the number of carbon atoms
    • C07C45/70—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by reactions not involving the formation of >C = O groups by isomerisation; by change of size of the carbon skeleton by increase in the number of carbon atoms by reaction with functional groups containing oxygen only in singly bound form
    • C07C45/71—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by reactions not involving the formation of >C = O groups by isomerisation; by change of size of the carbon skeleton by increase in the number of carbon atoms by reaction with functional groups containing oxygen only in singly bound form being hydroxy groups
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
    • C07D233/54—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
    • C07D233/56—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with only hydrogen atoms or radicals containing only hydrogen and carbon atoms, attached to ring carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D249/00—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms
    • C07D249/02—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms not condensed with other rings
    • C07D249/08—1,2,4-Triazoles; Hydrogenated 1,2,4-triazoles
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D303/00—Compounds containing three-membered rings having one oxygen atom as the only ring hetero atom
    • C07D303/02—Compounds containing oxirane rings
    • C07D303/12—Compounds containing oxirane rings with hydrocarbon radicals, substituted by singly or doubly bound oxygen atoms
    • C07D303/32—Compounds containing oxirane rings with hydrocarbon radicals, substituted by singly or doubly bound oxygen atoms by aldehydo- or ketonic radicals
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D407/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having oxygen atoms as the only ring hetero atoms, not provided for by group C07D405/00
    • C07D407/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having oxygen atoms as the only ring hetero atoms, not provided for by group C07D405/00 containing two hetero rings
    • C07D407/06—Heterocyclic compounds containing two or more hetero rings, at least one ring having oxygen atoms as the only ring hetero atoms, not provided for by group C07D405/00 containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Health & Medical Sciences (AREA)
  • Dentistry (AREA)
  • Agronomy & Crop Science (AREA)
  • Wood Science & Technology (AREA)
  • Engineering & Computer Science (AREA)
  • Zoology (AREA)
  • Plant Pathology (AREA)
  • Environmental Sciences (AREA)
  • Pest Control & Pesticides (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Medicinal Chemistry (AREA)
  • General Chemical & Material Sciences (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Epoxy Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Polymerization Catalysts (AREA)

Abstract

PROCEDIMIENTO PARA LA PRODUCCION DE DERIVADOS DE 1-CARBONIL-1-FENIL-2-AZOLIL-ETANOL.COMPRENDE, A) HACER REACCIONAR A UN COMPUESTO DE FORMULA (II), CON PARAFORMALDEHIDO, CON UNA BASE FUERTE NO NUCLEOFILA COMO HIDRURO ALCALINO Y CON ADICION DE TRIAZOL DE FORMULA (III), EN PRESENCIA DE DISOLVENTES ANHIDROS Y A UNA TEMPERATURA ENTRE 0 Y 140JC, PARA OBTENER UN COMPUESTO DE FORMULA (IV) Y B) HACER REACCIONAR A (IV) CON UN COMPUESTO DE FORMULA (V), EN UN DISOLVENTE INERTE Y EN PRESENCIA DE UNA BASE ALCALINA, PARA OBTENER UN COMPUESTO DE FORMULA (I), SUS SALES DE ADICION DE ACIDOS Y SALES DE AZOLIO CUATERNARIAS. SIENDO; R1, R2 Y R3 INDEPENDIENTES, H, HAL, ALQUILO DE C 1 A 4 Y OTROS; R4, H, ALQUILO DE C 1 A 10 Y OTROS; R5 ALQUILO DE C A 12, ALQUILO DE C 2 A 4 Y OTROS; HAL HALOGENO Y X -CH F O -N F.
ES527439A 1982-11-23 1983-11-22 Procedimiento para la produccion de derivados de 1-carbonil-1-fenil-2-azolil-etanol Expired ES8506566A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
CH682282 1982-11-23

Publications (2)

Publication Number Publication Date
ES527439A0 ES527439A0 (es) 1985-08-01
ES8506566A1 true ES8506566A1 (es) 1985-08-01

Family

ID=4315565

Family Applications (2)

Application Number Title Priority Date Filing Date
ES527438A Expired ES8504133A1 (es) 1982-11-23 1983-11-22 Procedimiento para la produccion de derivados de 1-carbonil-1-fenoxifenil-2-azolil-etanol
ES527439A Expired ES8506566A1 (es) 1982-11-23 1983-11-22 Procedimiento para la produccion de derivados de 1-carbonil-1-fenil-2-azolil-etanol

Family Applications Before (1)

Application Number Title Priority Date Filing Date
ES527438A Expired ES8504133A1 (es) 1982-11-23 1983-11-22 Procedimiento para la produccion de derivados de 1-carbonil-1-fenoxifenil-2-azolil-etanol

Country Status (19)

Country Link
EP (2) EP0117378A1 (es)
JP (2) JPS59106467A (es)
KR (1) KR840006648A (es)
AT (1) ATE37180T1 (es)
AU (3) AU2158283A (es)
BR (1) BR8306422A (es)
CA (2) CA1215374A (es)
DE (1) DE3377986D1 (es)
DK (1) DK534083A (es)
ES (2) ES8504133A1 (es)
GB (2) GB2130584B (es)
GR (1) GR79723B (es)
IL (2) IL70288A (es)
PH (1) PH19709A (es)
PL (1) PL141026B1 (es)
PT (1) PT77700B (es)
SU (1) SU1331427A3 (es)
TR (1) TR21666A (es)
ZA (2) ZA838696B (es)

Families Citing this family (26)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4517194A (en) * 1982-06-25 1985-05-14 Ciba-Geigy Corporation Azolylmandelic acid derivatives and use thereof for controlling microorganisms
DE3381012D1 (de) * 1983-01-10 1990-02-01 Ciba Geigy Ag Fluorazolyl-propanol-derivate als mikrobizide und wuchsregulierende mittel.
GB8301678D0 (en) * 1983-01-21 1983-02-23 Ici Plc Heterocyclic compounds
JPS59155365A (ja) * 1983-02-23 1984-09-04 Shionogi & Co Ltd ２−ヒドロキシプロピオフエノン誘導体
EP0117578A3 (en) * 1983-02-23 1985-01-30 Shionogi & Co., Ltd. Azole-substituted alcohol derivatives
US4584307A (en) * 1983-08-10 1986-04-22 Pfizer Inc. Antifungal 2-aryl-2-hydroxy perfluoro-1-(1H-1,2,4-triazol-1-yl) alkanones and alkanols
DE3407005A1 (de) * 1983-09-26 1985-04-04 Bayer Ag, 5090 Leverkusen Hydroxyethylazolyl-oxim-derivate
US4849007A (en) * 1985-12-02 1989-07-18 Ciba-Geigy Corporation Herbicidal epoxides
DE3921163A1 (de) * 1989-06-28 1991-01-10 Bayer Ag Hydroxy-keto-azole
US6297239B1 (en) 1997-10-08 2001-10-02 Merck & Co., Inc. Inhibitors of prenyl-protein transferase
KR100811402B1 (ko) * 2005-06-03 2008-03-07 박명호 신발끈 고정고리 와 신발끈 결속방법
CN105008336A (zh) 2012-11-27 2015-10-28 巴斯夫欧洲公司 取代2-[苯氧基苯基]-1-[1,2,4]三唑-1-基乙醇化合物及其作为杀真菌剂的用途
CN104955813A (zh) 2012-11-27 2015-09-30 巴斯夫欧洲公司 取代的[1,2,4]三唑化合物
EP2735563A1 (en) * 2012-11-27 2014-05-28 Basf Se Meta substituted 2-[phenoxy-phenyl]-1-[1,2,4]triazol-1-yl-ethanol compounds and their use as fungicides
WO2014082879A1 (en) 2012-11-27 2014-06-05 Basf Se Substituted [1,2,4]triazole compounds
US20160029630A1 (en) * 2012-11-27 2016-02-04 Basf Se Substituted 2-[phenoxy-phenyl]-1-[1,2,4]triazol-1-yl-ethanol compounds and their use as fungicides
WO2014082872A1 (en) * 2012-11-27 2014-06-05 Basf Se Substituted [1,2,4]triazole compounds
BR112015014753B8 (pt) 2012-12-20 2020-03-03 Basf Agro Bv composições, uso de uma composição, método para o combate de fungos fitopatogênicos e uso dos componentes
CN105008332A (zh) * 2013-01-08 2015-10-28 巴斯夫欧洲公司 作为杀真菌剂的取代的咪唑和(1,2,4)三唑类化合物
CN104968651A (zh) 2013-01-09 2015-10-07 巴斯夫农业公司 制备取代环氧乙烷类和三唑类的方法
PL3019013T3 (pl) 2013-07-08 2021-10-25 BASF Agro B.V. Kompozycje zawierające związek triazolowy i biopestycyd
EP3269245B1 (en) 2014-06-25 2023-08-16 BASF Agro B.V. Pesticidal compositions
UA120628C2 (uk) 2014-11-07 2020-01-10 Басф Се Пестицидні суміші
US11241012B2 (en) 2016-03-16 2022-02-08 Basf Se Use of tetrazolinones for combating resistant phytopathogenic fungi on soybean
EP3429357A1 (en) 2016-03-16 2019-01-23 Basf Se Use of tetrazolinones for combating resistant phytopathogenic fungi on cereals
WO2017157920A1 (en) 2016-03-16 2017-09-21 Basf Se Use of tetrazolinones for combating resistant phytopathogenic fungi on fruits

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE2348663A1 (de) * 1973-09-27 1975-04-03 Bayer Ag Verfahren zur herstellung von neuen 1-aethyl-azolylderivaten
CH647513A5 (de) * 1979-11-13 1985-01-31 Sandoz Ag Triazol-derivate, deren herstellung und verwendung.
GB2104065B (en) * 1981-06-04 1985-11-06 Ciba Geigy Ag Heterocyclyl-substituted mandelic acid compounds and mandelonitriles and their use for combating microorganisms
DE3275088D1 (en) * 1981-08-19 1987-02-19 Ici Plc Triazole derivatives, processes for preparing them, compositions containing them and processes for combating fungi and regulating plant growth

Also Published As

Publication number Publication date
GB2168053A (en) 1986-06-11
ES527439A0 (es) 1985-08-01
EP0117378A1 (de) 1984-09-05
JPS59106468A (ja) 1984-06-20
PH19709A (en) 1986-06-16
DE3377986D1 (en) 1988-10-20
GB8530463D0 (en) 1986-01-22
SU1331427A3 (ru) 1987-08-15
ZA838695B (en) 1984-07-25
IL70288A0 (en) 1984-02-29
EP0114567B1 (de) 1988-09-14
PL244693A1 (en) 1985-10-08
EP0114567A2 (de) 1984-08-01
GB2130584A (en) 1984-06-06
GB8330970D0 (en) 1983-12-29
ZA838696B (en) 1984-07-25
JPS59106467A (ja) 1984-06-20
CA1210404A (en) 1986-08-26
AU1069288A (en) 1988-05-05
ATE37180T1 (de) 1988-09-15
BR8306422A (pt) 1984-06-26
AU570653B2 (en) 1988-03-24
KR840006648A (ko) 1984-12-01
IL70284A (en) 1987-02-27
DK534083D0 (da) 1983-11-22
AU2158183A (en) 1984-05-31
PT77700A (en) 1983-12-01
ES527438A0 (es) 1985-04-16
CA1215374A (en) 1986-12-16
TR21666A (tr) 1985-01-21
GB2168053B (en) 1986-11-26
IL70284A0 (en) 1984-02-29
ES8504133A1 (es) 1985-04-16
EP0114567A3 (en) 1984-09-12
DK534083A (da) 1984-05-24
AU584000B2 (en) 1989-05-11
IL70288A (en) 1989-03-31
GB2130584B (en) 1986-11-26
AU2158283A (en) 1984-05-31
GR79723B (es) 1984-10-31
PT77700B (en) 1986-05-12
PL141026B1 (en) 1987-06-30

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Legal Events

Date Code Title Description
MM4A Patent lapsed

Effective date: 19960506