ES8403434A1 - Procedimiento para preparar un derivado fluorado de alquileno diamina. - Google Patents

Procedimiento para preparar un derivado fluorado de alquileno diamina.

Info

Publication number
ES8403434A1
ES8403434A1 ES515093A ES515093A ES8403434A1 ES 8403434 A1 ES8403434 A1 ES 8403434A1 ES 515093 A ES515093 A ES 515093A ES 515093 A ES515093 A ES 515093A ES 8403434 A1 ES8403434 A1 ES 8403434A1
Authority
ES
Spain
Prior art keywords
derivatives
diaminoalkene
fluorinated
represents hydrogen
alkyl
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
ES515093A
Other languages
English (en)
Other versions
ES515093A0 (es
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Merrell Toraude et Cie
Original Assignee
Merrell Toraude et Cie
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Merrell Toraude et Cie filed Critical Merrell Toraude et Cie
Publication of ES8403434A1 publication Critical patent/ES8403434A1/es
Publication of ES515093A0 publication Critical patent/ES515093A0/es
Granted legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C209/00—Preparation of compounds containing amino groups bound to a carbon skeleton
    • C07C209/04—Preparation of compounds containing amino groups bound to a carbon skeleton by substitution of functional groups by amino groups
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
    • C07D209/44—Iso-indoles; Hydrogenated iso-indoles
    • C07D209/48—Iso-indoles; Hydrogenated iso-indoles with oxygen atoms in positions 1 and 3, e.g. phthalimide
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/13—Amines
    • A61K31/15—Oximes (>C=N—O—); Hydrazines (>N—N<); Hydrazones (>N—N=) ; Imines (C—N=C)
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C43/00—Ethers; Compounds having groups, groups or groups
    • C07C43/02—Ethers
    • C07C43/03—Ethers having all ether-oxygen atoms bound to acyclic carbon atoms
    • C07C43/14—Unsaturated ethers
    • C07C43/17—Unsaturated ethers containing halogen
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00—Technologies relating to chemical industry
    • Y02P20/50—Improvements relating to the production of bulk chemicals
    • Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Epidemiology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Polymers With Sulfur, Phosphorus Or Metals In The Main Chain (AREA)

Abstract

PROCEDIMIENTOS PARA LA OBTENCION DE DERIVADOS FLUORADOS DE ALQUENILENO DIAMINAS Y SUS SALES FISIOLOGICAMENTE COMPATIBLES, DE FORMULA (I).CONSISTE EN LA REACCION DE AMINACION DE UN DERIVADO AMINO-PROTEGIDO DE UN COMPUESTO DE FORMULA (II), EN LA QUE Y ES UN GRUPO SALIENTE, R9 ES HIDROGENO, CIANO O ALCOXICARBONIL C2-9, Y LOS DEMAS SIMBOLOS TIENEN EL MISMO SIGNIFICADO QUE EN LA FORMULA (I). LA REACCION SE LLEVA A CABO POR CALENTAMIENTO A TEMPERATURAS ENTRE 10JC Y 100JC, EN UN DISOLVENTE INERTE.ESTOS COMPUESTOS TIENEN APLICACIONES PARA EL CONTROL DEL CRECIMIENTO DE TEJIDOSCON TUMOR, DE HIPERTROFIA PROSTATICA BENIGNA Y PARA EL CONTROL DEL CRECIMIENTO DE PROTOZOOS PARASITOS PATOGENOS.
ES515093A 1981-08-19 1982-08-18 Procedimiento para preparar un derivado fluorado de alquileno diamina. Granted ES515093A0 (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GB8125392 1981-08-19
GB8125360 1981-08-19

Publications (2)

Publication Number Publication Date
ES8403434A1 true ES8403434A1 (es) 1984-04-01
ES515093A0 ES515093A0 (es) 1984-04-01

Family

ID=26280522

Family Applications (1)

Application Number Title Priority Date Filing Date
ES515093A Granted ES515093A0 (es) 1981-08-19 1982-08-18 Procedimiento para preparar un derivado fluorado de alquileno diamina.

Country Status (14)

Country Link
EP (1) EP0072762B1 (es)
KR (1) KR890000621B1 (es)
AT (1) ATE15485T1 (es)
AU (1) AU548622B2 (es)
CA (1) CA1204770A (es)
DE (1) DE3266199D1 (es)
DK (1) DK161068C (es)
ES (1) ES515093A0 (es)
GB (1) GB2104072B (es)
GR (1) GR77603B (es)
IE (1) IE54303B1 (es)
IL (1) IL66568A0 (es)
NO (1) NO153173C (es)
NZ (1) NZ201590A (es)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4423073A (en) 1981-08-19 1983-12-27 Merrell Toraude Et Compagnie Fluorinated diaminopentene derivatives
DE3226550A1 (de) * 1982-07-13 1984-01-19 Schering AG, 1000 Berlin und 4709 Bergkamen Neue carbacycline, verfahren zu ihrer herstellung und ihre verwendung als arzneimittel

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4134918A (en) * 1977-09-06 1979-01-16 Merrell Toraude Et Compagnie Alpha-halomethyl derivatives of amines
NZ194347A (en) * 1979-07-26 1982-11-23 Merrell Toraude & Co Fluorinated alkenylamines intermediate alkenyl fluorinated methyl ketimine magnesium halides and preparation of certain amino alkanoic acids
GB2083030B (en) * 1980-08-23 1984-03-07 Merrell Toraude & Co Fluorinated pentene diamine derivatives

Also Published As

Publication number Publication date
AU548622B2 (en) 1985-12-19
GB2104072B (en) 1985-02-06
IE821942L (en) 1983-02-19
DE3266199D1 (de) 1985-10-17
ATE15485T1 (de) 1985-09-15
DK370882A (da) 1983-02-20
AU8724482A (en) 1983-02-24
NZ201590A (en) 1985-05-31
KR840001123A (ko) 1984-03-28
EP0072762A1 (en) 1983-02-23
GR77603B (es) 1984-09-25
CA1204770A (en) 1986-05-20
DK161068B (da) 1991-05-27
NO153173B (no) 1985-10-21
DK161068C (da) 1991-11-04
NO153173C (no) 1986-01-29
IL66568A0 (en) 1982-12-31
IE54303B1 (en) 1989-08-16
NO822810L (no) 1983-02-21
GB2104072A (en) 1983-03-02
EP0072762B1 (en) 1985-09-11
KR890000621B1 (ko) 1989-03-22
ES515093A0 (es) 1984-04-01

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Legal Events

Date Code Title Description
FD1A Patent lapsed

Effective date: 20040601