ES8301997A1 - Procedimiento para la preparacion de nuevas penicilinas. - Google Patents

Procedimiento para la preparacion de nuevas penicilinas.

Info

Publication number
ES8301997A1
ES8301997A1 ES506960A ES506960A ES8301997A1 ES 8301997 A1 ES8301997 A1 ES 8301997A1 ES 506960 A ES506960 A ES 506960A ES 506960 A ES506960 A ES 506960A ES 8301997 A1 ES8301997 A1 ES 8301997A1
Authority
ES
Spain
Prior art keywords
group
salts
penicillins
formula
preparation
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
ES506960A
Other languages
English (en)
Other versions
ES506960A0 (es
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Boehringer Ingelheim Pharma GmbH and Co KG
Original Assignee
Dr Karl Thomae GmbH
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Dr Karl Thomae GmbH filed Critical Dr Karl Thomae GmbH
Publication of ES506960A0 publication Critical patent/ES506960A0/es
Publication of ES8301997A1 publication Critical patent/ES8301997A1/es
Expired legal-status Critical Current

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D239/00Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/46Two or more oxygen, sulphur or nitrogen atoms
    • C07D239/48Two nitrogen atoms
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D499/00Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines Containing Antibodies Or Antigens For Use As Internal Diagnostic Agents (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)

Abstract

PROCEDIMIENTO PARA LA OBTENCION DE PENICILINA Y DE SUS SALES CON BASES, DE FORMULA (I) EN LA QUE Q ES UN RADICAL DE FORMULA (II) O (III), SIENDO R Y A VARIOS TIPOS DE RADICALES. CONSISTE EN LA REACCION DE UN COMPUESTO DE FORMULA (IV), CON UN DERIVADO DE PIRIMIDINA DE FORMULA (V) O UN DERIVADO REACTIVO DEL MISMO, EN LAS QUE B ES EL GRUPO <024>NCO; Y A Y R TIENEN EL MISMO SIGNIFICADO QUE EN LA FORMULA (I). LA REACCION SE LLEVA A CABO EN UN DISOLVENTE INERTE, A UN PH ENTRE 2,0 Y 9,0, A UNA TEMPERATURA ENTRE -20<025>C Y 50<025>C. ESTOS COMPUESTOS TIENEN APLICACIONES FARMACOLOGICAS POR SU ACTIVIDAD COMO ANTIBIOTICOS.
ES506960A 1980-11-11 1981-11-10 Procedimiento para la preparacion de nuevas penicilinas. Expired ES8301997A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE19803042440 DE3042440A1 (de) 1980-11-11 1980-11-11 Neue penicilline, ihre salze, verfahren zu ihrer herstellung und diese verbindungen enthaltende arzneimittel

Publications (2)

Publication Number Publication Date
ES506960A0 ES506960A0 (es) 1983-01-01
ES8301997A1 true ES8301997A1 (es) 1983-01-01

Family

ID=6116454

Family Applications (2)

Application Number Title Priority Date Filing Date
ES506960A Expired ES8301997A1 (es) 1980-11-11 1981-11-10 Procedimiento para la preparacion de nuevas penicilinas.
ES513341A Granted ES513341A0 (es) 1980-11-11 1982-06-22 "procedimiento para la preparacion de nuevas penicilinas".

Family Applications After (1)

Application Number Title Priority Date Filing Date
ES513341A Granted ES513341A0 (es) 1980-11-11 1982-06-22 "procedimiento para la preparacion de nuevas penicilinas".

Country Status (15)

Country Link
EP (1) EP0051773A1 (es)
JP (1) JPS57109793A (es)
AU (1) AU7735481A (es)
DD (1) DD201904A5 (es)
DE (1) DE3042440A1 (es)
DK (1) DK494981A (es)
ES (2) ES8301997A1 (es)
FI (1) FI813530L (es)
GB (1) GB2086904A (es)
GR (1) GR76931B (es)
IL (1) IL64245A0 (es)
NO (1) NO813806L (es)
PL (1) PL233755A1 (es)
PT (1) PT73970B (es)
ZA (1) ZA817745B (es)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN111518147A (zh) * 2020-04-29 2020-08-11 华东理工大学 苯甲酰苯胺类化合物及在制备铜绿假单胞菌抑制剂的增敏剂中的应用

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE2828261A1 (de) * 1978-06-28 1980-01-10 Thomae Gmbh Dr K Neue penicilline, ihre salze, verfahren zu ihrer herstellung und diese verbindungen enthaltende arzneimittel
DE2910190A1 (de) * 1979-03-15 1980-10-02 Thomae Gmbh Dr K Neue penicilline, ihre salze, verfahren zu ihrer herstellung und diese verbindungen enthaltende arzneimittel
DE2928344A1 (de) * 1979-07-13 1981-02-05 Thomae Gmbh Dr K Neue lactame, verfahren zu ihrer herstellung und diese verbindungen enthaltende arzneimittel

Also Published As

Publication number Publication date
AU7735481A (en) 1982-05-20
NO813806L (no) 1982-05-12
JPS57109793A (en) 1982-07-08
PL233755A1 (en) 1983-01-17
PT73970B (de) 1983-11-23
ZA817745B (en) 1983-07-27
GB2086904A (en) 1982-05-19
DE3042440A1 (de) 1982-06-24
GR76931B (es) 1984-09-04
ES506960A0 (es) 1983-01-01
FI813530L (fi) 1982-05-12
IL64245A0 (en) 1982-02-28
DD201904A5 (de) 1983-08-17
DK494981A (da) 1982-05-12
EP0051773A1 (de) 1982-05-19
PT73970A (de) 1981-12-01
ES8304993A1 (es) 1983-03-16
ES513341A0 (es) 1983-03-16

Similar Documents

Publication Publication Date Title
PH22166A (en) Propenylamines, method of use, pharmaceutical composition containing them
ES8304072A1 (es) &#34;procedimiento de preparacion de derivados de 1-fenil-1-hidroxi-etilamina&#34;.
ES480850A1 (es) Procedimiento para preparar hidantoinas.
IL60975A (en) Substituted oxiranecarboxylic acids,processes for their preparation and pharmaceutical compositions containing them
ES8304076A1 (es) &#34;procedimiento de preparacion de compuestos del tipo arilbencensulfonamida&#34;.
ES476682A1 (es) Un procedimiento para la preparacion de nuevos dericados de 1-aza-biciclo (2,2,2)octano, utiles como psicotrupos.
ES8206480A1 (es) Procedimiento para la preparacion de 2-halo piridinas
ES8301997A1 (es) Procedimiento para la preparacion de nuevas penicilinas.
DE3267188D1 (en) Hydroxybenzylamino-aryl compounds, process for preparing and pharmaceutical compositions containing the same
ES8302694A1 (es) &#34;un procedimiento para la preparacion de un derivado de imidazolina&#34;.
ES8305359A1 (es) Un procedimiento para la preparacion de benzamitas sustituidas.
JPS54106477A (en) Moranoline derivative
HUT39741A (en) Process for preparing pyridine derivatives and pharmaceutical compositions containing such compounds as active ingredients
ES8201962A1 (es) Un procedimiento para la preparacion de un compuesto de biu-ret 1,1,3,5-sustituido
ES482460A1 (es) Procedimiento para la obtencion de esteres de acido 2-ciclo-propil-pirimidin (4)il-tionofosfonico.
ES8307233A1 (es) Procedimiento para preparar derivados del acido 1,4-tiazan-3-carboxilico.
ES8301919A1 (es) Procedimiento para preparar derivados de indano
WO1989005787A3 (en) Processes and compounds useful for resolving 1-methyl-3-phenylpropylamine
ATE21693T1 (de) Substituierte pyrimid-2-one, ihre salze, verfahren zu ihrer herstellung und pharmazeutische zusammensetzungen, die diese enthalten.
ES478338A1 (es) Procedimiento para la obtencion de derivados de disulfimida.
NZ220589A (en) Morpholine alkyl aryl sulphonates and microbicidal agrochemical compositions thereof with certain triazoles
ES476712A1 (es) Procedimiento para la preparacion de derivados sustituidos de acido 1,4-ciclohexadieno carboxilico.
ES8206534A1 (es) Un procedimiento para la preparacion de derivados acilicos de cefalosporina
ES8305367A1 (es) &#34;procedimiento para la preparacion de nuevas penicilinas&#34;.
JPS5759856A (en) Benzene derivative