ES8104215A1 - Un procedimiento para la preparacion de sulfamidas. - Google Patents

Un procedimiento para la preparacion de sulfamidas.

Info

Publication number
ES8104215A1
ES8104215A1 ES491531A ES491531A ES8104215A1 ES 8104215 A1 ES8104215 A1 ES 8104215A1 ES 491531 A ES491531 A ES 491531A ES 491531 A ES491531 A ES 491531A ES 8104215 A1 ES8104215 A1 ES 8104215A1
Authority
ES
Spain
Prior art keywords
preparation
medicines
substituted
sulphonamide derivatives
methyl
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
ES491531A
Other languages
English (en)
Other versions
ES491531A0 (es
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
WUELFING JOHANN A KG
Original Assignee
WUELFING JOHANN A KG
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by WUELFING JOHANN A KG filed Critical WUELFING JOHANN A KG
Publication of ES8104215A1 publication Critical patent/ES8104215A1/es
Publication of ES491531A0 publication Critical patent/ES491531A0/es
Granted legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D295/00—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms
    • C07D295/04—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms
    • C07D295/12—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by singly or doubly bound nitrogen atoms
    • C07D295/125—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by singly or doubly bound nitrogen atoms with the ring nitrogen atoms and the substituent nitrogen atoms attached to the same carbon chain, which is not interrupted by carbocyclic rings
    • C07D295/13—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by singly or doubly bound nitrogen atoms with the ring nitrogen atoms and the substituent nitrogen atoms attached to the same carbon chain, which is not interrupted by carbocyclic rings to an acyclic saturated chain
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/06—Antiarrhythmics

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Cardiology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Hydrogenated Pyridines (AREA)
  • Pyrrole Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)

Abstract

PROCEDIMIENTO PARA LA PREPARACION DE SULFONAMIDAS, DE FORMULA (I), O UNA SAL DEL MISMO, DONDE NR2 REPRESENTA UN GRUPO PIPERIDILO, PIRROLIDILO O N-METIL PIPERAZILO; R ELEVADO A 1 ES UN GRUPO 1-NAFTILO QUE PUEDE ESTAR SUSTITUIDO POR DISTINTOS TIPOS DE RADICALES. SE OBTIENEN HACIENDO REACCIONAR UN COMPUESTO DE FORMULA (II) Y UN COMPUESTO DE FORMULA (III) O UN EQUIVALENTE QUIMICO DEL MISMO. ESTOS COMPUESTOS SE APLICAN COMO INHIBIDORES DE LA AGREGACION DE PLAQUETAS, R2N-(CH2)N-NH-SO2R ELEVADO A 1 (I) R2N-(CH2)N-NH2 (II) CL-SO2-R ELEVADO A 1 (III)
ES491531A 1979-05-16 1980-05-14 Un procedimiento para la preparacion de sulfamidas. Granted ES491531A0 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB7917035 1979-05-16

Publications (2)

Publication Number Publication Date
ES8104215A1 true ES8104215A1 (es) 1981-04-01
ES491531A0 ES491531A0 (es) 1981-04-01

Family

ID=10505195

Family Applications (1)

Application Number Title Priority Date Filing Date
ES491531A Granted ES491531A0 (es) 1979-05-16 1980-05-14 Un procedimiento para la preparacion de sulfamidas.

Country Status (12)

Country Link
US (2) US4436908A (es)
EP (1) EP0021580B1 (es)
JP (1) JPS56161371A (es)
AU (1) AU531826B2 (es)
CA (1) CA1166256A (es)
DE (1) DE3065868D1 (es)
DK (1) DK156643C (es)
ES (1) ES491531A0 (es)
IE (1) IE49799B1 (es)
IL (1) IL60087A0 (es)
NZ (1) NZ193654A (es)
ZA (1) ZA802911B (es)

Families Citing this family (14)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE3276313D1 (en) * 1981-09-24 1987-06-19 Beecham Wuelfing Gmbh & Co Kg Sulphonamides
JP2000504677A (ja) * 1996-02-09 2000-04-18 スミスクライン・ビーチャム・パブリック・リミテッド・カンパニー ５ｈｔ７レセプター・アンタゴニスト用のスルホンアミド誘導体
GB9612884D0 (en) * 1996-06-20 1996-08-21 Smithkline Beecham Plc Novel compounds
DZ2376A1 (fr) 1996-12-19 2002-12-28 Smithkline Beecham Plc Dérivés de sulfonamides nouveaux procédé pour leurpréparation et compositions pharmaceutiques les c ontenant.
GB9803536D0 (en) * 1998-02-19 1998-04-15 Black James Foundation Histamine H,receptor ligands
US7928121B2 (en) 2002-02-19 2011-04-19 Laboratorios Del Dr. Esteve, S.A. 5-HT7 receptor antagonists
EP1676844A1 (en) 2004-12-28 2006-07-05 Laboratorios Del Dr. Esteve, S.A. 5-HT7 receptor antagonists
EP1676840A1 (en) 2004-12-28 2006-07-05 Laboratorios Del Dr. Esteve, S.A. 5-HT7 Receptor antagonists
US7553965B2 (en) 2002-11-07 2009-06-30 Laboratories Del Dr. Esteve, S.A. 5-HT7 receptor antagonists
ES2257168B1 (es) 2004-08-18 2007-06-01 Laboratorios Del Dr Esteve, S.A. Ligandos del receptor 5-ht7.
US7211585B2 (en) 2004-08-18 2007-05-01 Laboratorios Del Dr. Esteve, S.A. 5-HT7 receptor antagonists
US7211584B2 (en) 2004-08-18 2007-05-01 Laboratorios Del Dr. Esteve, S.A. 5-HT7 receptor ligands
EP1630158A1 (en) 2004-08-18 2006-03-01 Laboratorios Del Dr. Esteve, S.A. 5-HT7 receptor antagonists
RU2565404C1 (ru) * 2014-12-02 2015-10-20 Общество с ограниченной ответственностью "Научно-исследовательский центр "Парк активных молекул" Средство, проявляющее антиаритмическую активность

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB1052977A (es) 1963-09-14
US4001229A (en) 1974-04-04 1977-01-04 Mead Johnson & Company Alkanesulfonamido triphenylethylenes
US3929803A (en) 1974-05-28 1975-12-30 Pfizer Aryl carboxylic acids
FR2313918A1 (fr) * 1975-06-09 1977-01-07 Choay Sa Methoxy-2 benzenesulfonamides n-substitues, procede pour les preparer et medicaments les contenant
JPS5829784B2 (ja) * 1975-08-22 1983-06-24 萬有製薬株式会社 オメガ − （ アリ−ルスルホンアミド ）− アルキルアミンノ セイホウ
DE2718405A1 (de) 1977-04-26 1978-11-02 Boehringer Sohn Ingelheim Neue n- eckige klammer auf 1-(3-benzoylpropyl)-4-piperidyl eckige klammer zu -sulfonsaeureamide und verfahren zu deren herstellung
JPS5533439A (en) 1978-08-31 1980-03-08 Konishiroku Photo Ind Co Ltd 2-sulfamoyl-5-sulfamido-1-naphthol

Also Published As

Publication number Publication date
US4372955A (en) 1983-02-08
DK156643C (da) 1990-02-05
ZA802911B (en) 1981-05-27
AU531826B2 (en) 1983-09-08
IL60087A0 (en) 1980-07-31
CA1166256A (en) 1984-04-24
EP0021580A1 (en) 1981-01-07
DE3065868D1 (en) 1984-01-19
NZ193654A (en) 1984-08-24
JPS56161371A (en) 1981-12-11
EP0021580B1 (en) 1983-12-14
AU5850180A (en) 1980-11-20
DK156643B (da) 1989-09-18
IE801001L (en) 1980-11-16
IE49799B1 (en) 1985-12-25
DK215980A (da) 1980-11-17
ES491531A0 (es) 1981-04-01
US4436908A (en) 1984-03-13

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