ES554503A0 - Procedimiento para preparar derivados de 2-amino-tiazol - Google Patents
Procedimiento para preparar derivados de 2-amino-tiazolInfo
- Publication number
- ES554503A0 ES554503A0 ES554503A ES554503A ES554503A0 ES 554503 A0 ES554503 A0 ES 554503A0 ES 554503 A ES554503 A ES 554503A ES 554503 A ES554503 A ES 554503A ES 554503 A0 ES554503 A0 ES 554503A0
- Authority
- ES
- Spain
- Prior art keywords
- amino
- alkyl
- group
- hydrogen atom
- preparing
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
- C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
- C07D417/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P27/00—Drugs for disorders of the senses
- A61P27/02—Ophthalmic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P27/00—Drugs for disorders of the senses
- A61P27/02—Ophthalmic agents
- A61P27/14—Decongestants or antiallergics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/08—Antiallergic agents
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
- C07D277/02—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
- C07D277/20—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D277/32—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D277/38—Nitrogen atoms
- C07D277/42—Amino or imino radicals substituted by hydrocarbon or substituted hydrocarbon radicals
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
- C07D277/02—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
- C07D277/20—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D277/32—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D277/56—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Public Health (AREA)
- Pharmacology & Pharmacy (AREA)
- Animal Behavior & Ethology (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Ophthalmology & Optometry (AREA)
- Rheumatology (AREA)
- Immunology (AREA)
- Pain & Pain Management (AREA)
- Pulmonology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Thiazole And Isothizaole Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Micro-Organisms Or Cultivation Processes Thereof (AREA)
- Agricultural Chemicals And Associated Chemicals (AREA)
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
FR8506568A FR2581063B1 (fr) | 1985-04-30 | 1985-04-30 | Amino-2 thiazoles n-substitues, leur procede de preparation et leur application en therapeutique |
Publications (2)
Publication Number | Publication Date |
---|---|
ES8900045A1 ES8900045A1 (es) | 1988-11-16 |
ES554503A0 true ES554503A0 (es) | 1988-11-16 |
Family
ID=9318828
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
ES554503A Expired ES8900045A1 (es) | 1985-04-30 | 1986-04-29 | Procedimiento para preparar derivados de 2-amino-tiazol |
Country Status (11)
Country | Link |
---|---|
US (1) | US4785008A (es) |
EP (1) | EP0202157B1 (es) |
JP (1) | JPH0629270B2 (es) |
AT (1) | ATE45734T1 (es) |
CA (1) | CA1289144C (es) |
DE (1) | DE3665176D1 (es) |
DK (1) | DK168523B1 (es) |
ES (1) | ES8900045A1 (es) |
FR (1) | FR2581063B1 (es) |
IE (1) | IE59141B1 (es) |
PT (1) | PT82480B (es) |
Families Citing this family (19)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
EP0254259A3 (en) * | 1986-07-21 | 1989-11-23 | Otsuka Pharmaceutical Factory, Inc. | P-aminophenol derivatives |
JPS6339868A (ja) * | 1986-08-04 | 1988-02-20 | Otsuka Pharmaceut Factory Inc | ジ低級アルキルフエノ−ル誘導体 |
FR2612187B1 (fr) * | 1987-03-12 | 1989-07-21 | Sanofi Sa | Derives du thiazole actifs sur le systeme cholinergique, leur procede de preparation et compositions pharmaceutiques en contenant |
AU628485B2 (en) * | 1989-02-23 | 1992-09-17 | Otsuka Pharmaceutical Factory, Inc. | P-aminophenol derivative and production and application thereof |
JPH03111178U (es) * | 1990-02-27 | 1991-11-14 | ||
US6225305B1 (en) | 1993-10-04 | 2001-05-01 | Glaxo Wellcome Inc. | Substituted urea and isothiorea derivatives as no synthase inhibitors |
AU7705694A (en) * | 1993-10-04 | 1995-05-01 | Glaxo Wellcome House | Substituted urea and isothiourea derivatives as no synthase inhibitors |
US6297276B1 (en) | 1993-10-04 | 2001-10-02 | Glaxosmithkline | Substituted urea and isothiourea derivatives as no synthase inhibitors |
US6090846A (en) * | 1994-06-01 | 2000-07-18 | Glaxo Wellcome Inc. | Substituted urea and isothiourea derivatives as no synthase inhibitors |
GB9418912D0 (en) * | 1994-09-20 | 1994-11-09 | Fisons Corp | Pharmaceutically active compounds |
US6100282A (en) | 1998-01-02 | 2000-08-08 | Hoffman-La Roche Inc. | Thiazole derivatives |
ATE365158T1 (de) | 1999-04-28 | 2007-07-15 | Inst Med Molecular Design Inc | Pyrimidincarbonsäurederivate |
BR0013899A (pt) * | 1999-09-10 | 2003-07-08 | Merck & Co Inc | Composto, composição farmacêutica, processos de tratamento ou prevenção de câncer, de uma doença em que a angiogênese esteja implicada, da vascularização retinal, da retinopatia diabética, da degeneração macular relacionada a idade, de doenças inflamatórias, de uma doença ou condições dependentes da tirosina quinase, de patologias associadas com ossos, e, processos para produzir uma composição farmacêutica, e de reduzir ou prevenir dano tecidual em seguida a um evento isquêmico cerebral |
WO2007002461A1 (en) * | 2005-06-23 | 2007-01-04 | Dr. Reddy's Laboratories Ltd. | 3,4-substituted thiazoles as ampk activators |
US8080668B2 (en) * | 2005-07-04 | 2011-12-20 | Dr. Reddy's Laboratories Limited | Thiazoles derivatives as AMPK activator |
CN101977504B (zh) | 2008-03-19 | 2014-11-26 | 拜尔农科股份公司 | 杀真菌剂肟基-四唑衍生物 |
US10696638B2 (en) | 2017-12-26 | 2020-06-30 | Industrial Technology Research Institute | Compounds for inhibiting AGC kinase and pharmaceutical compositions comprising the same |
US11091473B2 (en) | 2018-05-29 | 2021-08-17 | Acadia Pharmaceuticals Inc. | Compounds for pain treatment, compositions comprising same, and methods of using same |
MX2021013524A (es) | 2019-05-10 | 2021-12-10 | Cersci Therapeutics Inc | Metodos de fabricacion y polimorfos de un agente antihiperalgesico de tiazolina. |
Family Cites Families (8)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
BE603739A (es) * | 1960-05-13 | |||
US3299087A (en) * | 1961-04-24 | 1967-01-17 | Geigy Chem Corp | Nu, nu'-bis-(thiazolyl)-phenylenediamines |
US3467666A (en) * | 1966-11-07 | 1969-09-16 | Geigy Chem Corp | 2-substituted aminothiazoles |
BE795907A (fr) * | 1972-02-25 | 1973-06-18 | Luso Farmaco Inst | 2-amino-4-arylthiazoles 5-substitues et leur preparation |
JPS5742629B2 (es) * | 1973-10-29 | 1982-09-09 | ||
JPS565747B2 (es) * | 1973-10-24 | 1981-02-06 | ||
JPS5833870B2 (ja) * | 1976-01-12 | 1983-07-22 | 塩野義製薬株式会社 | チアゾリン誘導体 |
DK150068C (da) * | 1978-06-02 | 1987-06-29 | Pfizer | Analogifremgangsmaade til fremstilling af aminothiazoler |
-
1985
- 1985-04-30 FR FR8506568A patent/FR2581063B1/fr not_active Expired
-
1986
- 1986-04-24 US US06/855,411 patent/US4785008A/en not_active Expired - Fee Related
- 1986-04-28 IE IE111986A patent/IE59141B1/en not_active IP Right Cessation
- 1986-04-29 PT PT82480A patent/PT82480B/pt not_active IP Right Cessation
- 1986-04-29 CA CA000507824A patent/CA1289144C/en not_active Expired - Lifetime
- 1986-04-29 ES ES554503A patent/ES8900045A1/es not_active Expired
- 1986-04-30 DK DK197786A patent/DK168523B1/da not_active IP Right Cessation
- 1986-04-30 AT AT86400959T patent/ATE45734T1/de not_active IP Right Cessation
- 1986-04-30 DE DE8686400959T patent/DE3665176D1/de not_active Expired
- 1986-04-30 EP EP86400959A patent/EP0202157B1/fr not_active Expired
- 1986-04-30 JP JP61100781A patent/JPH0629270B2/ja not_active Expired - Lifetime
Also Published As
Publication number | Publication date |
---|---|
EP0202157A1 (fr) | 1986-11-20 |
JPH0629270B2 (ja) | 1994-04-20 |
ATE45734T1 (de) | 1989-09-15 |
IE59141B1 (en) | 1994-01-12 |
FR2581063B1 (fr) | 1987-07-17 |
DK197786A (da) | 1986-10-31 |
ES8900045A1 (es) | 1988-11-16 |
IE861119L (en) | 1986-10-30 |
US4785008A (en) | 1988-11-15 |
CA1289144C (en) | 1991-09-17 |
DK197786D0 (da) | 1986-04-30 |
PT82480B (pt) | 1988-03-03 |
DE3665176D1 (en) | 1989-09-28 |
PT82480A (en) | 1986-05-01 |
JPS6277375A (ja) | 1987-04-09 |
FR2581063A1 (fr) | 1986-10-31 |
DK168523B1 (da) | 1994-04-11 |
EP0202157B1 (fr) | 1989-08-23 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
FD1A | Patent lapsed |
Effective date: 20001102 |