ES548238A0 - Procedimiento para preparar analogos de adenosinas n6 susti-tuidas - Google Patents

Procedimiento para preparar analogos de adenosinas n6 susti-tuidas

Info

Publication number
ES548238A0
ES548238A0 ES548238A ES548238A ES548238A0 ES 548238 A0 ES548238 A0 ES 548238A0 ES 548238 A ES548238 A ES 548238A ES 548238 A ES548238 A ES 548238A ES 548238 A0 ES548238 A0 ES 548238A0
Authority
ES
Spain
Prior art keywords
tuidas
susti
adenosins
procedure
preparing analogs
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
ES548238A
Other languages
English (en)
Other versions
ES8701774A1 (es
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Warner Lambert Co LLC
Original Assignee
Warner Lambert Co LLC
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Warner Lambert Co LLC filed Critical Warner Lambert Co LLC
Publication of ES548238A0 publication Critical patent/ES548238A0/es
Publication of ES8701774A1 publication Critical patent/ES8701774A1/es
Expired legal-status Critical Current

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07HSUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H19/00Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof
    • C07H19/02Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof sharing nitrogen
    • C07H19/04Heterocyclic radicals containing only nitrogen atoms as ring hetero atom
    • C07H19/16Purine radicals

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Health & Medical Sciences (AREA)
  • Biochemistry (AREA)
  • Biotechnology (AREA)
  • General Health & Medical Sciences (AREA)
  • Genetics & Genomics (AREA)
  • Molecular Biology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)
ES548238A 1984-10-26 1985-10-25 Procedimiento para preparar analogos de adenosinas n6 susti-tuidas Expired ES8701774A1 (es)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
US66523284A 1984-10-26 1984-10-26
US66523384A 1984-10-26 1984-10-26
US66521784A 1984-10-26 1984-10-26
US77231585A 1985-09-06 1985-09-06

Publications (2)

Publication Number Publication Date
ES548238A0 true ES548238A0 (es) 1986-12-01
ES8701774A1 ES8701774A1 (es) 1986-12-01

Family

ID=27505316

Family Applications (1)

Application Number Title Priority Date Filing Date
ES548238A Expired ES8701774A1 (es) 1984-10-26 1985-10-25 Procedimiento para preparar analogos de adenosinas n6 susti-tuidas

Country Status (13)

Country Link
EP (1) EP0181129B1 (es)
KR (1) KR910002226B1 (es)
CN (1) CN1013448B (es)
AU (1) AU575438B2 (es)
CA (1) CA1260931A (es)
DE (1) DE3568582D1 (es)
DK (1) DK488485A (es)
ES (1) ES8701774A1 (es)
FI (1) FI81587C (es)
GR (1) GR852583B (es)
NO (1) NO165495C (es)
NZ (1) NZ213971A (es)
PT (1) PT81373B (es)

Families Citing this family (22)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0206497B1 (en) * 1985-05-15 1994-07-20 The Wellcome Foundation Limited Therapeutic nucleosides and their preparation
WO1988003147A1 (en) * 1986-10-31 1988-05-05 Warner-Lambert Company Selected n6-substituted adenosines having selective a2 binding activity
GB2226027B (en) * 1988-12-13 1992-05-20 Sandoz Ltd Adenosine derivatives,their production and use
JPH0725785B2 (ja) * 1989-01-11 1995-03-22 日本臓器製薬株式会社 アデノシン誘導体及び該化合物を有効成分として含有する医薬組成物
ZA902280B (en) * 1989-03-29 1990-12-28 Merrell Dow Pharma Selective adenosine receptor agents
EP0550631B1 (en) * 1990-09-25 1997-01-02 Rhone-Poulenc Rorer International (Holdings) Inc. Compounds having antihypertensive and anti-ischemic properties
US5561134A (en) * 1990-09-25 1996-10-01 Rhone-Poulenc Rorer Pharmaceuticals Inc. Compounds having antihypertensive, cardioprotective, anti-ischemic and antilipolytic properties
US5705491A (en) * 1992-10-27 1998-01-06 Nippon Zoki Pharmaceutical Co., Ltd. Adenosine deaminase inhibitor
US5589467A (en) * 1993-09-17 1996-12-31 Novo Nordisk A/S 2,5',N6-trisubstituted adenosine derivatives
CN1168138A (zh) * 1995-11-14 1997-12-17 法玛西雅厄普约翰公司 芳基和杂芳基嘌呤化合物
TW528755B (en) 1996-12-24 2003-04-21 Glaxo Group Ltd 2-(purin-9-yl)-tetrahydrofuran-3,4-diol derivatives
YU44900A (sh) 1998-01-31 2003-01-31 Glaxo Group Limited Derivati 2-(purin-9-il)tetrahidrofuran-3,4-diola
HUP0103025A3 (en) 1998-06-23 2002-04-29 Glaxo Group Ltd A2a agonist 2-(purin-9-yl)tetrahydrofuran-3,4-diol derivatives, medicaments containing the same, process for producing them and the useful intermediates
JP3619017B2 (ja) 1998-06-24 2005-02-09 日本臓器製薬株式会社 新規アラビノシルアデニン誘導体
US6946449B2 (en) 2001-07-13 2005-09-20 Cv Therapeutics, Inc. Partial and full agonists of A1 adenosine receptors
US7713946B2 (en) 2002-07-11 2010-05-11 Cv Therapeutics, Inc. Partial and full agonists A1 adenosine receptors
US7157440B2 (en) 2001-07-13 2007-01-02 Cv Therapeutics, Inc. Partial and full agonists of A1 adenosine receptors
US7265111B2 (en) 2002-06-27 2007-09-04 Sanofi-Aventis Deutschland Gmbh Adenosine analogues and their use as pharmaceutical agents
EP1375508A1 (en) * 2002-06-27 2004-01-02 Aventis Pharma Deutschland GmbH N6-substituted adenosine analogues and their use as pharmaceutical agents
EP1590359A2 (en) 2003-02-03 2005-11-02 CV Therapeutics Inc. PARTIAL AND FULL AGONISTS OF A sb 1 /sb ADENOSINE RECEPTORS
AR049384A1 (es) 2004-05-24 2006-07-26 Glaxo Group Ltd Derivados de purina
GB0514809D0 (en) 2005-07-19 2005-08-24 Glaxo Group Ltd Compounds

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE1545645A1 (de) * 1965-12-06 1969-08-21 Boehringer Mannheim Gmbh Verfahren zur Herstellung von disubstituierten Adenosin-Derivaten
DE1670077C3 (de) * 1966-05-07 1975-04-24 Boehringer Mannheim Gmbh, 6800 Mannheim Adenosin-Derivate und Verfahren zu ihrer Herstellung
SE361760B (es) * 1972-04-05 1973-11-12 Haldex Ab
DE2230160A1 (de) * 1972-06-21 1974-01-31 Merck Patent Gmbh Adenosinderivat
US4373097A (en) * 1981-04-27 1983-02-08 Bioresearch S.R.L. Process for preparing adenosine derivatives of anti-inflammatory and analgesic activity
DE3576344D1 (de) * 1984-04-18 1990-04-12 Whitby Research Inc Cardio-vasodilatatore n-6-substituierte adenosine.
US5310731A (en) * 1984-06-28 1994-05-10 Whitby Research, Inc. N-6 substituted-5'-(N-substitutedcarboxamido)adenosines as cardiac vasodilators and antihypertensive agents
CA1255297A (en) * 1984-10-26 1989-06-06 Bharat Trivedi N.sup.6-benzopyrano and benzothiopyrano adenosines

Also Published As

Publication number Publication date
PT81373A (en) 1985-11-01
FI854153A0 (fi) 1985-10-23
PT81373B (pt) 1987-11-11
NZ213971A (en) 1988-03-30
DE3568582D1 (en) 1989-04-13
NO165495C (no) 1991-02-20
GR852583B (es) 1986-02-26
FI81587C (fi) 1990-11-12
NO165495B (no) 1990-11-12
EP0181129A3 (en) 1987-05-13
FI81587B (fi) 1990-07-31
ES8701774A1 (es) 1986-12-01
KR910002226B1 (ko) 1991-04-08
CA1260931A (en) 1989-09-26
KR860003256A (ko) 1986-05-21
DK488485A (da) 1986-04-27
DK488485D0 (da) 1985-10-24
FI854153L (fi) 1986-04-27
EP0181129B1 (en) 1989-03-08
NO854278L (no) 1986-04-28
CN85108658A (zh) 1986-07-16
AU4888885A (en) 1986-05-08
CN1013448B (zh) 1991-08-07
EP0181129A2 (en) 1986-05-14
AU575438B2 (en) 1988-07-28

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Legal Events

Date Code Title Description
FD1A Patent lapsed

Effective date: 19960603