ES504316A0 - Procedimiento para la obtencion de derivados del acido 2-(3'-hidroxipirid-2'-il)-2-tiazolin-4-carboxilico - Google Patents

Procedimiento para la obtencion de derivados del acido 2-(3'-hidroxipirid-2'-il)-2-tiazolin-4-carboxilico

Info

Publication number
ES504316A0
ES504316A0 ES504316A ES504316A ES504316A0 ES 504316 A0 ES504316 A0 ES 504316A0 ES 504316 A ES504316 A ES 504316A ES 504316 A ES504316 A ES 504316A ES 504316 A0 ES504316 A0 ES 504316A0
Authority
ES
Spain
Prior art keywords
tiazolin
hidroxipirid
carboxilico
procedure
obtaining
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
ES504316A
Other languages
English (en)
Spanish (es)
Other versions
ES8301476A1 (es
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Novartis AG
Original Assignee
Ciba Geigy AG
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Ciba Geigy AG filed Critical Ciba Geigy AG
Publication of ES8301476A1 publication Critical patent/ES8301476A1/es
Publication of ES504316A0 publication Critical patent/ES504316A0/es
Granted legal-status Critical Current

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D213/00Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
    • C07D213/02Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/60Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D213/78Carbon atoms having three bonds to hetero atoms, with at the most one bond to halogen, e.g. ester or nitrile radicals
    • C07D213/79Acids; Esters
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D417/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/04Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07FACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F7/00Compounds containing elements of Groups 4 or 14 of the Periodic Table
    • C07F7/02Silicon compounds
    • C07F7/08Compounds having one or more C—Si linkages
    • C07F7/0803Compounds with Si-C or Si-Si linkages
    • C07F7/081Compounds with Si-C or Si-Si linkages comprising at least one atom selected from the elements N, O, halogen, S, Se or Te
    • C07F7/0812Compounds with Si-C or Si-Si linkages comprising at least one atom selected from the elements N, O, halogen, S, Se or Te comprising a heterocyclic ring
    • CCHEMISTRY; METALLURGY
    • C12BIOCHEMISTRY; BEER; SPIRITS; WINE; VINEGAR; MICROBIOLOGY; ENZYMOLOGY; MUTATION OR GENETIC ENGINEERING
    • C12NMICROORGANISMS OR ENZYMES; COMPOSITIONS THEREOF; PROPAGATING, PRESERVING, OR MAINTAINING MICROORGANISMS; MUTATION OR GENETIC ENGINEERING; CULTURE MEDIA
    • C12N1/00Microorganisms, e.g. protozoa; Compositions thereof; Processes of propagating, maintaining or preserving microorganisms or compositions thereof; Processes of preparing or isolating a composition containing a microorganism; Culture media therefor
    • C12N1/20Bacteria; Culture media therefor
    • C12N1/205Bacterial isolates
    • CCHEMISTRY; METALLURGY
    • C12BIOCHEMISTRY; BEER; SPIRITS; WINE; VINEGAR; MICROBIOLOGY; ENZYMOLOGY; MUTATION OR GENETIC ENGINEERING
    • C12PFERMENTATION OR ENZYME-USING PROCESSES TO SYNTHESISE A DESIRED CHEMICAL COMPOUND OR COMPOSITION OR TO SEPARATE OPTICAL ISOMERS FROM A RACEMIC MIXTURE
    • C12P17/00Preparation of heterocyclic carbon compounds with only O, N, S, Se or Te as ring hetero atoms
    • C12P17/16Preparation of heterocyclic carbon compounds with only O, N, S, Se or Te as ring hetero atoms containing two or more hetero rings
    • C12P17/167Heterorings having sulfur atoms as ring heteroatoms, e.g. vitamin B1, thiamine nucleus and open chain analogs
    • CCHEMISTRY; METALLURGY
    • C12BIOCHEMISTRY; BEER; SPIRITS; WINE; VINEGAR; MICROBIOLOGY; ENZYMOLOGY; MUTATION OR GENETIC ENGINEERING
    • C12RINDEXING SCHEME ASSOCIATED WITH SUBCLASSES C12C - C12Q, RELATING TO MICROORGANISMS
    • C12R2001/00Microorganisms ; Processes using microorganisms
    • C12R2001/01Bacteria or Actinomycetales ; using bacteria or Actinomycetales
    • C12R2001/465Streptomyces
    • C12R2001/48Streptomyces antibioticus ; Actinomyces antibioticus

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Zoology (AREA)
  • Wood Science & Technology (AREA)
  • Genetics & Genomics (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Biotechnology (AREA)
  • General Health & Medical Sciences (AREA)
  • Biochemistry (AREA)
  • General Engineering & Computer Science (AREA)
  • Microbiology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Virology (AREA)
  • Biomedical Technology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
ES504316A 1980-07-28 1981-07-27 Procedimiento para la obtencion de derivados del acido 2-(3'-hidroxipirid-2'-il)-2-tiazolin-4-carboxilico Granted ES504316A0 (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
CH575580 1980-07-28
CH592580 1980-08-05

Publications (2)

Publication Number Publication Date
ES8301476A1 ES8301476A1 (es) 1982-12-01
ES504316A0 true ES504316A0 (es) 1982-12-01

Family

ID=25698328

Family Applications (4)

Application Number Title Priority Date Filing Date
ES504316A Granted ES504316A0 (es) 1980-07-28 1981-07-27 Procedimiento para la obtencion de derivados del acido 2-(3'-hidroxipirid-2'-il)-2-tiazolin-4-carboxilico
ES514588A Expired ES8308878A1 (es) 1980-07-28 1982-07-30 Procedimiento para la obtencion de derivados del acido 2-(3'-hidroxi-pirid-2'-il)-2-tiazolin-4-carboxilico.
ES514586A Granted ES514586A0 (es) 1980-07-28 1982-07-30 Procedimiento para la obtencion de derivados del acido 2-(3'-hidroxi-pirid-2'-il)-2-tiazolin-4-carboxilico.
ES514587A Granted ES514587A0 (es) 1980-07-28 1982-07-30 Procedimiento para la obtencion de derivados del acido 2-(3'-hidroxi-pirid-2'-il)-2-tiazolin-4-carboxilico.

Family Applications After (3)

Application Number Title Priority Date Filing Date
ES514588A Expired ES8308878A1 (es) 1980-07-28 1982-07-30 Procedimiento para la obtencion de derivados del acido 2-(3'-hidroxi-pirid-2'-il)-2-tiazolin-4-carboxilico.
ES514586A Granted ES514586A0 (es) 1980-07-28 1982-07-30 Procedimiento para la obtencion de derivados del acido 2-(3'-hidroxi-pirid-2'-il)-2-tiazolin-4-carboxilico.
ES514587A Granted ES514587A0 (es) 1980-07-28 1982-07-30 Procedimiento para la obtencion de derivados del acido 2-(3'-hidroxi-pirid-2'-il)-2-tiazolin-4-carboxilico.

Country Status (13)

Country Link
US (1) US4406905A (OSRAM)
EP (1) EP0045281B1 (OSRAM)
AU (1) AU548331B2 (OSRAM)
CA (1) CA1172188A (OSRAM)
DE (1) DE3170401D1 (OSRAM)
DK (1) DK160304C (OSRAM)
ES (4) ES504316A0 (OSRAM)
GB (1) GB2085873B (OSRAM)
GR (1) GR74313B (OSRAM)
IE (1) IE51430B1 (OSRAM)
IL (1) IL63428A (OSRAM)
NZ (1) NZ197840A (OSRAM)
PT (1) PT73439B (OSRAM)

Families Citing this family (26)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
HU200177B (en) * 1985-06-18 1990-04-28 Biogal Gyogyszergyar Process for producing thiazolidinecarboxylic acids and pharmaceutical compositions comprising such compounds
JPS63225373A (ja) * 1986-07-24 1988-09-20 Sumitomo Pharmaceut Co Ltd 新規チアゾリジン−4−オン誘導体およびその酸付加塩
CN1030415A (zh) * 1987-02-20 1989-01-18 山之内制药株式会社 饱和的杂环碳酰胺衍生物和它的制备方法
US4992455A (en) * 1987-05-22 1991-02-12 Sumitomo Pharmaceuticals Company, Limited Thiazolidin-4-one derivatives useful for treating diseases caused by platelet activating factor
ATE98631T1 (de) * 1988-01-20 1994-01-15 Ciba Geigy Ag Verfahren zur herstellung von komplexverbindungen.
US5021435A (en) * 1988-01-22 1991-06-04 Sumitomo Pharmaceuticals Company, Limited Certain pyridyl-thiazolidin-4-one having anti-ulcer activity
US5840739A (en) * 1992-11-16 1998-11-24 University Of Florida Research Foundation, Inc. Thiazoline acid derivatives
WO1994011367A1 (en) * 1992-11-16 1994-05-26 University Of Florida Research Foundation Inc. 2-(pyrid-2'-yl)-2-thiazoline-4(s)-carboxylic acid derivatives
DE69525439T2 (de) * 1994-08-05 2002-08-08 SHIONOGI & CO., LTD. Antibiotikum und verfahren zu dessen herstellung
US6083966A (en) * 1998-08-31 2000-07-04 University Of Florida Thiazoline acid derivatives
CN1585639A (zh) * 1998-09-21 2005-02-23 佛罗里达大学研究基金会 抗疟疾制剂
AU139723S (en) * 1999-02-09 2000-02-07 Colgate Palmolive Co Container
AT500490A1 (de) * 2001-10-16 2006-01-15 Dsm Fine Chem Austria Gmbh Verfahren zur herstellung von substituierten thiazolinen und deren zwischenprodukte
US6794515B2 (en) * 2002-05-15 2004-09-21 Genzyme Corporation Synthesis of 2-alkylcysteine via substituted thiazoline amide
EP1548013A4 (en) * 2002-10-01 2006-07-12 Kaneka Corp PROCESS FOR PRODUCTION OF OPTICALLY ACTIVE ALPHA-SUBSTITUTED CYSTEINE OR SALT THEREOF, INTERMEDIATE THEREFOR AND PROCESS FOR PRODUCTION THEREOF
WO2005034949A1 (en) * 2003-09-09 2005-04-21 University Of Florida Desferrithiocin derivatives and their use as iron chelators
PL1866296T3 (pl) 2005-04-04 2017-05-31 University Of Florida Research Foundation, Inc. Polieterowe analogi desferritiocyny
CA2680592C (en) * 2007-03-15 2016-07-05 University Of Florida Research Foundation, Inc. Desferrithiocin polyether analogues and uses thereof in treating pathological conditions
KR102111176B1 (ko) 2011-12-16 2020-05-15 유니버시티 오브 플로리다 리서치 파운데이션, 인코포레이티드 4'-데스페리티오신 유사체의 용도
USD736089S1 (en) 2012-06-14 2015-08-11 S.C. Johnson & Son, Inc. Bottle
USD722879S1 (en) 2012-06-14 2015-02-24 S.C. Johnson & Son, Inc. Bottle
USD736637S1 (en) 2012-06-14 2015-08-18 S.C. Johnson & Son, Inc. Bottle
EP3071201A4 (en) 2013-11-22 2017-04-26 University of Florida Research Foundation, Inc. Desferrithiocin analogs and uses thereof
CN106660957B (zh) 2014-07-08 2019-11-29 美国陶氏益农公司 4-烷氧基-3-羟基吡啶甲酸的制备方法
CA2954268C (en) 2014-07-08 2022-11-22 Dow Agrosciences Llc Process for the preparation of 3-hydroxypicolinic acids
KR20170140306A (ko) 2015-04-27 2017-12-20 유니버시티 오브 플로리다 리서치 파운데이션, 인코포레이티드 대사적으로 프로그램화된 금속 킬레이트화제 및 그의 용도

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3592905A (en) * 1969-10-30 1971-07-13 Merck & Co Inc Therapeutic methods
CA962269A (en) * 1971-05-05 1975-02-04 Robert E. Grahame (Jr.) Thiazoles, and their use as insecticides
US3852293A (en) * 1972-06-21 1974-12-03 Uniroyal Inc 4-phenyl-2-(3-pyridyl)-thiazole carboxamides
US3842172A (en) * 1972-10-06 1974-10-15 Uniroyal Inc Pharmaceutical compositions containing a 4-substituted-2-(3-pyridyl)thiazole and methods of using same
FR2356423A1 (fr) * 1976-07-01 1978-01-27 Oeriu Simion Derives de l'acide thiazolidinecarboxylique, leur preparation et leur application comme medicaments

Also Published As

Publication number Publication date
IE51430B1 (en) 1986-12-24
DK335781A (da) 1982-01-29
US4406905A (en) 1983-09-27
ES8308877A1 (es) 1983-10-01
AU7343981A (en) 1982-02-04
PT73439A (de) 1981-08-01
EP0045281A1 (de) 1982-02-03
CA1172188A (en) 1984-08-07
IL63428A (en) 1984-12-31
IL63428A0 (en) 1981-10-30
EP0045281B1 (de) 1985-05-08
DE3170401D1 (en) 1985-06-13
IE811697L (en) 1982-01-28
NZ197840A (en) 1985-08-30
ES8301476A1 (es) 1982-12-01
ES8400425A1 (es) 1983-11-01
ES514588A0 (es) 1983-10-01
ES8308878A1 (es) 1983-10-01
DK160304B (da) 1991-02-25
ES514587A0 (es) 1983-10-01
DK160304C (da) 1991-07-29
AU548331B2 (en) 1985-12-05
GB2085873B (en) 1984-03-21
ES514586A0 (es) 1983-11-01
PT73439B (de) 1983-06-20
GB2085873A (en) 1982-05-06
GR74313B (OSRAM) 1984-06-22

Similar Documents

Publication Publication Date Title
ES504316A0 (es) Procedimiento para la obtencion de derivados del acido 2-(3'-hidroxipirid-2'-il)-2-tiazolin-4-carboxilico
ES525435A0 (es) Procedimiento para la produccion de n-piridinsulfonil-n'-pirimidinil- y -triacinilureas
ES524495A0 (es) Procedimiento para la preparacion de derivados del acido metilendifosfonico
MX162188A (es) Procedimiento para la produccion de las n-arilsulfonil-n'-pirimidinil-ureas
ES515426A0 (es) Procedimiento para la obtencion de compuestos del acido 7 b-aminotiadiazolilacetilamino-3-amoniometil-3-cefem-4-carboxilico.
AR225363A1 (es) Procedimiento para la preparacion de acido alfa-hidroxi-gamma-metilmercaptobutirico
MX7101E (es) Procedimiento para la preparacion de derivados de acido quinolin-carboxilico
AR230056A1 (es) Procedimiento para la preparacion de derivados del acido 3-ridilmetilo 3-piridilmetilo 3-inidazolilmetil indolil-acrilico
ES516594A0 (es) Procedimiento para la obtencion de esteres del acido 7 -2-(2amino-4-tiazolil)-2-(sin)-metoxiimionoacetamido)-3-cefem-4-carboxilico.
ES494538A0 (es) Procedimiento para la obtencion de compuestos de acido 7 b- aminotiadiazolilacetilamino-3-cefem-4 carboxilico
MX153817A (es) Procedimiento para la preparacion de acido 4,4'-dinitro-estilben-2,2-disulfonico
ES508811A0 (es) "prodedimiento para la preparacion de derivados de fenoxi-aminipropanol"
ES514791A0 (es) "procedimiento para la preparacion de nuevos derivados de acido fenoxi-fenil-aminico".
ES508346A0 (es) Un procedimiento para la preparacion de derivados del acido 2 beta-clorometil-2 alfa-metilpenam-3 alfa-carboxilico.
ES502952A0 (es) Procedimiento para la obtencion de amidas de acido 1,4-dihi-dropiridin-4-carboxilico
ES545068A0 (es) Procedimiento para la fabricacion de derivados del acido aminotiazolilpropandicarboxilico
AR227793A1 (es) Procedimiento para la produccion de derivados de 1,4-dioxido de 2-alpha-de derivados de 1,4-dioxido de 2-(alpha-hidrazino-alpha-hidroximetil)-quinoxalina
ES515170A0 (es) "procedimiento para la preparacion de esteres del acido alcoxivincaminico".
ES502848A0 (es) Procedimiento para la preparacion de derivados de acido in- dolacetico
ES514136A0 (es) "procedimiento para la fabricacion de derivados de la nitrosourea".
ES495554A0 (es) Un procedimiento para la preparacion de acido 6-(2-(2'- metilfenoxicarbonil)-2-tien-3'-ilacetamido)penicilanico
ES527129A0 (es) Procedimiento para la obtencion de derivados de acido maloico sustituidos
ES496624A0 (es) Procedimiento para la preparacion de nuevas n-3-trifluorome-tilfenil-n'-benzoilureas substituidas
ES535195A0 (es) Procedimiento para la obtencion de compuestos del acido 7b -acilamido-3-cefem-4-carboxilico
ES510704A0 (es) "procedimiento de obtencion de nuevos derivados del acido 2-hidro-xibenzoico".

Legal Events

Date Code Title Description
PC1A Transfer granted