ES479122A1 - Procedimiento para la obtencion de preparados de accion diu-retica para administracion parenteral. - Google Patents

Procedimiento para la obtencion de preparados de accion diu-retica para administracion parenteral.

Info

Publication number
ES479122A1
ES479122A1 ES479122A ES479122A ES479122A1 ES 479122 A1 ES479122 A1 ES 479122A1 ES 479122 A ES479122 A ES 479122A ES 479122 A ES479122 A ES 479122A ES 479122 A1 ES479122 A1 ES 479122A1
Authority
ES
Spain
Prior art keywords
quick
diuretic compositions
acting
acting diuretic
compositions
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
ES479122A
Other languages
English (en)
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Roehm Pharma GmbH
Original Assignee
Roehm Pharma GmbH
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Roehm Pharma GmbH filed Critical Roehm Pharma GmbH
Publication of ES479122A1 publication Critical patent/ES479122A1/es
Expired legal-status Critical Current

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D295/00Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms
    • C07D295/04Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms
    • C07D295/08Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by singly bound oxygen or sulfur atoms
    • C07D295/096Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by singly bound oxygen or sulfur atoms with the ring nitrogen atoms and the oxygen or sulfur atoms separated by carbocyclic rings or by carbon chains interrupted by carbocyclic rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/63Compounds containing para-N-benzenesulfonyl-N-groups, e.g. sulfanilamide, p-nitrobenzenesulfonyl hydrazide
    • A61K31/635Compounds containing para-N-benzenesulfonyl-N-groups, e.g. sulfanilamide, p-nitrobenzenesulfonyl hydrazide having a heterocyclic ring, e.g. sulfadiazine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00Drugs for disorders of the blood or the extracellular fluid
    • A61P7/10Antioedematous agents; Diuretics
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D475/00Heterocyclic compounds containing pteridine ring systems
    • C07D475/06Heterocyclic compounds containing pteridine ring systems with a nitrogen atom directly attached in position 4
    • C07D475/08Heterocyclic compounds containing pteridine ring systems with a nitrogen atom directly attached in position 4 with a nitrogen atom directly attached in position 2

Abstract

Procedimiento para la obtención de preparados de acción diurética para administración parenteral, caracterizado porque se disuelve ácido 4-cloro-N-furfuril-5-sulfamoilantranílico (furosemida) conjuntamente con por lo menos un compuesto de la fórmula general I: ***1 (Ver fórmula 1) como materias activas en un medio por lo menos parcialmente acuoso adecuado para aplicación intravenosa, comprendiendo el medio acuoso por lo menos 100 veces el peso de las materias activas.
ES479122A 1978-04-10 1979-03-30 Procedimiento para la obtencion de preparados de accion diu-retica para administracion parenteral. Expired ES479122A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE19782815442 DE2815442A1 (de) 1978-04-10 1978-04-10 Rasch wirksame diuretika

Publications (1)

Publication Number Publication Date
ES479122A1 true ES479122A1 (es) 1979-07-01

Family

ID=6036603

Family Applications (1)

Application Number Title Priority Date Filing Date
ES479122A Expired ES479122A1 (es) 1978-04-10 1979-03-30 Procedimiento para la obtencion de preparados de accion diu-retica para administracion parenteral.

Country Status (10)

Country Link
US (1) US4335119A (es)
JP (2) JPS54135795A (es)
AT (1) AT365452B (es)
CH (1) CH638980A5 (es)
DE (1) DE2815442A1 (es)
ES (1) ES479122A1 (es)
FR (1) FR2422403A1 (es)
GB (1) GB2018133B (es)
IT (1) IT1121452B (es)
SE (1) SE7903200L (es)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2486082A2 (fr) * 1977-01-03 1982-01-08 Roehm Pharma Gmbh Composes de la pteridine et leur application en tant que matieres therapeutiquement actives dans des preparations pharmaceutiques
US4481095A (en) * 1982-02-03 1984-11-06 Inoue-Japax Research Incorporated Apparatus for supplying a working fluid and a wire electrode to a work portion of a wire-cut electrical discharge machine
DE3305935C2 (de) * 1983-02-21 1985-05-30 Medice Chem.-Pharm. Fabrik Pütter GmbH & Co KG, 5860 Iserlohn Kaliumneutrales Saluretikum mit antihypertensiver Wirkung
DE3448490C2 (de) * 1984-04-05 1995-04-27 Roehm Pharma Gmbh Verwendung von Pteridinderivaten zur Behandlung von Herzarrhythmien
US5944021A (en) * 1995-06-07 1999-08-31 Rodriguez; Victorio C. Therapeutic use of a carbonic anhydrase enzyme inhibitor for the treatment of brain edema
US7671029B2 (en) 1999-08-06 2010-03-02 Immupharma Sa Compositions and methods for enhanced pharmacological activity of compositions comprising peptide drug substances

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE2614738C2 (de) * 1976-04-06 1985-01-31 Röhm Pharma GmbH, 6100 Darmstadt Diuretisch wirkende Arzneimittel
US4252809A (en) * 1977-01-03 1981-02-24 Rohm Pharma Gmbh Substituted pteridine compounds and pharmaceutical compositions containing the same
DE2700073A1 (de) * 1977-01-03 1978-07-13 Roehm Pharma Gmbh Pteridinverbindungen mit pharmazeutischer wirksamkeit

Also Published As

Publication number Publication date
US4335119A (en) 1982-06-15
FR2422403A1 (fr) 1979-11-09
ATA216079A (de) 1981-06-15
JPH04210983A (ja) 1992-08-03
SE7903200L (sv) 1979-10-11
IT1121452B (it) 1986-04-02
DE2815442A1 (de) 1979-10-18
JPS54135795A (en) 1979-10-22
GB2018133B (en) 1982-08-18
AT365452B (de) 1982-01-25
JPH0338249B2 (es) 1991-06-10
DE2815442C2 (es) 1989-05-11
GB2018133A (en) 1979-10-17
IT7967612A0 (it) 1979-03-23
CH638980A5 (de) 1983-10-31
FR2422403B1 (es) 1983-01-28

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