ES420175A1 - Procedimiento para preparar derivados de tetrahidropinol (1,2-a) pirazinas. - Google Patents
Procedimiento para preparar derivados de tetrahidropinol (1,2-a) pirazinas.Info
- Publication number
- ES420175A1 ES420175A1 ES420175A ES420175A ES420175A1 ES 420175 A1 ES420175 A1 ES 420175A1 ES 420175 A ES420175 A ES 420175A ES 420175 A ES420175 A ES 420175A ES 420175 A1 ES420175 A1 ES 420175A1
- Authority
- ES
- Spain
- Prior art keywords
- radical
- mono
- angle
- alkylamino
- tetrahydropyrrolo
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired
Links
- RWRDLPDLKQPQOW-UHFFFAOYSA-N Pyrrolidine Chemical compound C1CCNC1 RWRDLPDLKQPQOW-UHFFFAOYSA-N 0.000 abstract 3
- 125000003545 alkoxy group Chemical group 0.000 abstract 3
- -1 alkyl radical Chemical class 0.000 abstract 3
- YNAVUWVOSKDBBP-UHFFFAOYSA-N Morpholine Chemical compound C1COCCN1 YNAVUWVOSKDBBP-UHFFFAOYSA-N 0.000 abstract 2
- NQRYJNQNLNOLGT-UHFFFAOYSA-N Piperidine Chemical compound C1CCNCC1 NQRYJNQNLNOLGT-UHFFFAOYSA-N 0.000 abstract 2
- 125000003282 alkyl amino group Chemical group 0.000 abstract 2
- 229910052739 hydrogen Inorganic materials 0.000 abstract 2
- 239000001257 hydrogen Substances 0.000 abstract 2
- 125000004435 hydrogen atom Chemical group [H]* 0.000 abstract 2
- 150000003254 radicals Chemical class 0.000 abstract 2
- SLRMQYXOBQWXCR-UHFFFAOYSA-N 2154-56-5 Chemical compound [CH2]C1=CC=CC=C1 SLRMQYXOBQWXCR-UHFFFAOYSA-N 0.000 abstract 1
- 101100295738 Gallus gallus COR3 gene Proteins 0.000 abstract 1
- 125000004423 acyloxy group Chemical group 0.000 abstract 1
- 125000000217 alkyl group Chemical group 0.000 abstract 1
- 150000001875 compounds Chemical class 0.000 abstract 1
- 125000002887 hydroxy group Chemical group [H]O* 0.000 abstract 1
- 125000001997 phenyl group Chemical group [H]C1=C([H])C([H])=C(*)C([H])=C1[H] 0.000 abstract 1
- 125000004193 piperazinyl group Chemical group 0.000 abstract 1
- 125000002924 primary amino group Chemical group [H]N([H])* 0.000 abstract 1
- 239000003204 tranquilizing agent Substances 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D207/00—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom
- C07D207/02—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D207/04—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
- C07D207/10—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D207/16—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| IT3127672 | 1972-11-03 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ES420175A1 true ES420175A1 (es) | 1976-07-16 |
Family
ID=11233382
Family Applications (2)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ES420175A Expired ES420175A1 (es) | 1972-11-03 | 1973-10-31 | Procedimiento para preparar derivados de tetrahidropinol (1,2-a) pirazinas. |
| ES421819A Expired ES421819A1 (es) | 1972-11-03 | 1973-12-27 | Procedimiento para preparar derivados de tetrahidropirrol (1,2-a) pirazina. |
Family Applications After (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ES421819A Expired ES421819A1 (es) | 1972-11-03 | 1973-12-27 | Procedimiento para preparar derivados de tetrahidropirrol (1,2-a) pirazina. |
Country Status (18)
Families Citing this family (12)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4697016A (en) * | 1984-10-26 | 1987-09-29 | Ciba-Geigy Corporation | Intermediates for the preparation of a carboxylic acid |
| US4595766A (en) * | 1984-10-26 | 1986-06-17 | Ciba-Geigy Corporation | Process for the preparation of an indoline carboxylic acid |
| JPH0745501B2 (ja) * | 1986-11-27 | 1995-05-17 | 日本臓器製薬株式会社 | 新規環状ジペプチド化合物 |
| DE3830096A1 (de) * | 1988-09-03 | 1990-03-15 | Hoechst Ag | Piperazindione mit psychotroper wirkung |
| WO1993023404A1 (en) * | 1992-05-19 | 1993-11-25 | Immunopharmaceutics, Inc. | Compounds that modulate endothelin activity |
| US6057314A (en) * | 1995-12-21 | 2000-05-02 | Biochem Pharma Inc. | Low molecular weight bicyclic thrombin inhibitors |
| US5958905A (en) | 1996-03-26 | 1999-09-28 | Texas Biotechnology Corporation | Phosphoramidates, phosphinic amides and related compounds and the use thereof to modulate the activity of endothelin |
| US6124291A (en) * | 1996-06-18 | 2000-09-26 | Warner-Lambert Company | Pyrrolo[1,2-a]pyrazine-1,4-dione serine protease inhibitors |
| MXPA02006134A (es) | 1999-12-21 | 2002-12-13 | Guilford Pharm Inc | Compuestos derivados de hidantoina, composiciones farmaceuticas y metodos de uso de los mismos. |
| US6815214B2 (en) | 2000-12-29 | 2004-11-09 | Celltech R & D, Inc. | Pharmaceutical uses and synthesis of diketopiperazines |
| JP6465803B2 (ja) * | 2012-10-22 | 2019-02-06 | シティ・オブ・ホープＣｉｔｙ ｏｆ Ｈｏｐｅ | Ｅｔｐ誘導体 |
| WO2018053345A1 (en) | 2016-09-15 | 2018-03-22 | City Of Hope | Dithio etp derivatives |
Family Cites Families (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US3176017A (en) * | 1963-02-26 | 1965-03-30 | American Home Prod | Aroylalkyl derivatives of diazabicyclo-nonanes and-decanes |
| US3503980A (en) * | 1965-10-04 | 1970-03-31 | Ciba Geigy Corp | Tetrahydroazacycloalkano(1,2-a) pyridazines |
| DE1695554C3 (de) * | 1966-02-12 | 1974-02-21 | Nautschno-Issledowatelskij Institut Farmakologii I Chimioterapii, Moskau | Verfahren zur Herstellung kondensierter Piperazinonderivate |
| US3563992A (en) * | 1967-10-31 | 1971-02-16 | Abbott Lab | 1,4-diaza-bicyclo(4,3,0)nonane-2,5,9-triones |
-
1973
- 1973-01-01 AR AR250020A patent/AR206504A1/es active
- 1973-09-28 ZA ZA737653*A patent/ZA737653B/xx unknown
- 1973-10-01 GB GB4580773A patent/GB1409185A/en not_active Expired
- 1973-10-16 AU AU61417/73A patent/AU475776B2/en not_active Expired
- 1973-10-19 US US408243A patent/US3920660A/en not_active Expired - Lifetime
- 1973-10-25 IL IL43485A patent/IL43485A0/xx unknown
- 1973-10-25 NL NL7314665A patent/NL7314665A/xx unknown
- 1973-10-29 DE DE19732354056 patent/DE2354056A1/de active Pending
- 1973-10-30 LU LU68719A patent/LU68719A1/xx unknown
- 1973-10-30 FR FR7338685A patent/FR2205323B1/fr not_active Expired
- 1973-10-30 RO RO7300076461A patent/RO63259A/ro unknown
- 1973-10-31 ES ES420175A patent/ES420175A1/es not_active Expired
- 1973-10-31 BE BE137334A patent/BE806827A/xx unknown
- 1973-11-01 DD DD174415A patent/DD107930A5/xx unknown
- 1973-11-02 HU HULE726A patent/HU166438B/hu unknown
- 1973-11-02 JP JP48123936A patent/JPS4976896A/ja active Pending
- 1973-11-02 SU SU1965998A patent/SU513627A3/ru active
- 1973-11-02 AT AT925273A patent/AT336622B/de not_active IP Right Cessation
- 1973-11-09 IL IL43606A patent/IL43606A0/xx unknown
- 1973-12-27 ES ES421819A patent/ES421819A1/es not_active Expired
Also Published As
| Publication number | Publication date |
|---|---|
| DE2354056A1 (de) | 1974-05-16 |
| ATA925273A (de) | 1976-09-15 |
| ZA737653B (en) | 1974-08-28 |
| IL43485A0 (en) | 1974-01-14 |
| US3920660A (en) | 1975-11-18 |
| JPS4976896A (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html) | 1974-07-24 |
| AT336622B (de) | 1977-05-10 |
| DD107930A5 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html) | 1974-08-20 |
| AR206504A1 (es) | 1976-07-30 |
| SU513627A3 (ru) | 1976-05-05 |
| HU166438B (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html) | 1975-03-28 |
| AU475776B2 (en) | 1976-09-02 |
| NL7314665A (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html) | 1974-05-07 |
| AU6141773A (en) | 1975-04-17 |
| FR2205323A1 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html) | 1974-05-31 |
| GB1409185A (en) | 1975-10-08 |
| RO63259A (fr) | 1978-08-15 |
| IL43606A0 (en) | 1974-03-14 |
| FR2205323B1 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html) | 1976-12-03 |
| LU68719A1 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html) | 1974-01-08 |
| BE806827A (fr) | 1974-02-15 |
| ES421819A1 (es) | 1976-06-16 |
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