ES368552A1 - Un procedimiento para la preparacion de i - sustituido - 4 - aroilpiperidinas. - Google Patents
Un procedimiento para la preparacion de i - sustituido - 4 - aroilpiperidinas.Info
- Publication number
- ES368552A1 ES368552A1 ES368552A ES368552A ES368552A1 ES 368552 A1 ES368552 A1 ES 368552A1 ES 368552 A ES368552 A ES 368552A ES 368552 A ES368552 A ES 368552A ES 368552 A1 ES368552 A1 ES 368552A1
- Authority
- ES
- Spain
- Prior art keywords
- reacting
- halide
- acetyl
- alkyl
- aroyl
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D317/00—Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms
- C07D317/08—Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms having the hetero atoms in positions 1 and 3
- C07D317/10—Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms having the hetero atoms in positions 1 and 3 not condensed with other rings
- C07D317/14—Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms having the hetero atoms in positions 1 and 3 not condensed with other rings with substituted hydrocarbon radicals attached to ring carbon atoms
- C07D317/18—Radicals substituted by singly bound oxygen or sulfur atoms
- C07D317/20—Free hydroxyl or mercaptan
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D211/00—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
- C07D211/04—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D211/06—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
- C07D211/08—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms
- C07D211/18—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms with substituted hydrocarbon radicals attached to ring carbon atoms
- C07D211/30—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms with substituted hydrocarbon radicals attached to ring carbon atoms with hydrocarbon radicals, substituted by doubly bound oxygen or sulfur atoms or by two oxygen or sulfur atoms singly bound to the same carbon atom
- C07D211/32—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms with substituted hydrocarbon radicals attached to ring carbon atoms with hydrocarbon radicals, substituted by doubly bound oxygen or sulfur atoms or by two oxygen or sulfur atoms singly bound to the same carbon atom by oxygen atoms
-
- G—PHYSICS
- G06—COMPUTING; CALCULATING OR COUNTING
- G06Q—INFORMATION AND COMMUNICATION TECHNOLOGY [ICT] SPECIALLY ADAPTED FOR ADMINISTRATIVE, COMMERCIAL, FINANCIAL, MANAGERIAL OR SUPERVISORY PURPOSES; SYSTEMS OR METHODS SPECIALLY ADAPTED FOR ADMINISTRATIVE, COMMERCIAL, FINANCIAL, MANAGERIAL OR SUPERVISORY PURPOSES, NOT OTHERWISE PROVIDED FOR
- G06Q20/00—Payment architectures, schemes or protocols
- G06Q20/04—Payment circuits
- G06Q20/047—Payment circuits using payment protocols involving electronic receipts
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Business, Economics & Management (AREA)
- Accounting & Taxation (AREA)
- Strategic Management (AREA)
- Physics & Mathematics (AREA)
- General Business, Economics & Management (AREA)
- General Physics & Mathematics (AREA)
- Engineering & Computer Science (AREA)
- Theoretical Computer Science (AREA)
- Hydrogenated Pyridines (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US73842068A | 1968-06-20 | 1968-06-20 |
Publications (1)
Publication Number | Publication Date |
---|---|
ES368552A1 true ES368552A1 (es) | 1971-07-01 |
Family
ID=24967943
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
ES368552A Expired ES368552A1 (es) | 1968-06-20 | 1969-06-19 | Un procedimiento para la preparacion de i - sustituido - 4 - aroilpiperidinas. |
Country Status (20)
Country | Link |
---|---|
US (1) | US3576810A (xx) |
JP (2) | JPS5022033B1 (xx) |
AT (1) | AT291258B (xx) |
BE (1) | BE734755A (xx) |
BR (1) | BR6909774D0 (xx) |
CA (1) | CA991642A (xx) |
CH (2) | CH555335A (xx) |
DE (1) | DE1930818C3 (xx) |
DK (1) | DK132947C (xx) |
ES (1) | ES368552A1 (xx) |
FI (1) | FI51347C (xx) |
FR (1) | FR2011339A1 (xx) |
GB (1) | GB1268909A (xx) |
IE (1) | IE33848B1 (xx) |
IL (1) | IL32431A (xx) |
MY (1) | MY7300424A (xx) |
NL (1) | NL158488B (xx) |
NO (1) | NO136493C (xx) |
SE (1) | SE377118B (xx) |
TR (1) | TR17521A (xx) |
Families Citing this family (48)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
BE791088A (fr) * | 1971-11-09 | 1973-03-01 | Richardson Merrell Inc | Nouveaux derives d'aryl (piperidyl-4) cetone, utiles notamment comme analgesiques et anticoagulants, et leur procede de preparation |
US4101662A (en) * | 1973-05-03 | 1978-07-18 | A. H. Robins Company, Incorporated | Method for inhibiting emesis and compositions therefor |
SE7409245L (xx) * | 1973-07-19 | 1975-01-20 | Robins Co Inc A H | |
US3922276A (en) * | 1974-12-11 | 1975-11-25 | Robins Co Inc A H | 1-Substituted-4-benzylidenepiperidines |
US3956296A (en) * | 1974-12-11 | 1976-05-11 | A. H. Robins Company, Incorporated | 1-Substituted-4-benzylpiperidines |
US4032642A (en) * | 1974-12-11 | 1977-06-28 | A. H. Robins Company, Incorporated | 1-Substituted-4-benzylpiperidines |
JPS52142126U (xx) * | 1976-04-23 | 1977-10-27 | ||
GB1561023A (en) * | 1977-04-22 | 1980-02-13 | Beecham Group Ltd | 2-methoxy - 5 - chloro aniline derivatives |
JPS54139937U (xx) * | 1978-03-20 | 1979-09-28 | ||
US4216325A (en) * | 1978-07-11 | 1980-08-05 | A. H. Robins Company, Inc. | 4-(p-Fluorobenzoyl)-1-[3-(p-fluorobenzoyl)propyl]piperidine |
US4246268A (en) * | 1979-02-09 | 1981-01-20 | Richardson-Merrell Inc. | Neuroleptic-4-(naphthylmethyl)piperidine derivatives |
JPS5628625U (xx) * | 1979-08-10 | 1981-03-18 | ||
US4283404A (en) * | 1979-09-04 | 1981-08-11 | Richardson-Merrell Inc. | Aroylethenylpiperidinobutyrophenone antipsychotic agents |
US4284636A (en) * | 1979-09-04 | 1981-08-18 | Richardson-Merrell Inc. | Cinnamoylpiperidinobutyrophenone antipsychotic agents |
JPS56129232U (xx) * | 1980-02-29 | 1981-10-01 | ||
DK149133C (da) * | 1980-09-18 | 1986-09-08 | Ucb Sa | Analogifremgangsmaade til fremstilling af 2-(4-(diphenylmethylen)- l-piperidinyl)- eddikesyrer eller farmaceutisk acceptable salte heraf |
JPS5783219A (en) * | 1980-11-12 | 1982-05-25 | Iseki Agricult Mach | Conveying device for threshed straw |
US4408053A (en) * | 1981-11-12 | 1983-10-04 | Hoechst-Roussel Pharmaceuticals Inc. | (4-Piperidyl)-substituted phenyl ketones |
FR2581993B1 (fr) * | 1985-05-14 | 1988-03-18 | Synthelabo | Derives de (benzoyl-4 piperidino)-2 phenyl-1 alcanols, leur preparation et leur application en therapeutique |
US4912117A (en) * | 1985-07-02 | 1990-03-27 | Merrell Dow Pharmaceuticals Inc. | Novel chemical compounds |
US4783471A (en) * | 1985-07-02 | 1988-11-08 | Merrell Dow Pharmaceuticals Inc. | N-aralkyl piperidine methanol derivatives and the uses thereof |
DK623586A (da) * | 1985-12-27 | 1987-06-28 | Eisai Co Ltd | Piperidinderivater eller salte deraf og farmaceutiske kompositioner indeholdende forbindelserne |
KR910006138B1 (ko) * | 1986-09-30 | 1991-08-16 | 에자이 가부시끼가이샤 | 환상아민 유도체 |
US5523307A (en) * | 1987-11-27 | 1996-06-04 | Eisai Co., Ltd. | Cyclic amine and pharmacological composition |
US5196439A (en) * | 1987-11-27 | 1993-03-23 | Eisai Co., Ltd. | Piperidine compounds useful to treat cerebrovascular diseases |
DE3854991T2 (de) * | 1987-11-27 | 1996-07-18 | Eisai Co Ltd | Cyclische Amine und pharmakologische Verbindungen |
US5093341A (en) * | 1987-12-17 | 1992-03-03 | Merrell Dow Pharmaceuticals Inc. | N-aralkyl piperidine derivatives useful as antithrombolytic agents |
US5064838A (en) * | 1988-01-21 | 1991-11-12 | Merrell Dow Pharmaceuticals | 1,4-disubstituted-piperidinyl compounds as pain relievers |
US4921863A (en) * | 1988-02-17 | 1990-05-01 | Eisai Co., Ltd. | Cyclic amine derivatives |
US5198449A (en) * | 1990-04-27 | 1993-03-30 | A. H. Robins Company Incorporated | N-substituted alpha-arylazacycloalkylmethanamines and their use as cardiovascular agents |
US5225412A (en) * | 1991-04-29 | 1993-07-06 | Hoechst-Roussel Pharmaceuticals Incorporated | Benzoisothiazole-and benzisoxazole-3-carboxamides |
US5143923B1 (en) * | 1991-04-29 | 1993-11-02 | Hoechst-Roussel Pharmaceuticals Incorporated | Benzoisothiazole-and benzisoxazole-3-carboxamides |
US5378714A (en) * | 1991-11-27 | 1995-01-03 | Novo Nordisk A/S | Antipsychotic piperidine derivatives |
ES2066721B1 (es) * | 1993-05-18 | 1996-02-16 | Ferrer Int | Nuevos compuestos derivados de la piridina 1,4-disustituida. |
DK60893D0 (da) * | 1993-05-26 | 1993-05-26 | Novo Nordisk As | Piperidinderivater, deres fremstilling og anvendelse |
EP0661266A1 (en) * | 1993-12-27 | 1995-07-05 | Toa Eiyo Ltd. | Substituted cyclic amine compounds as 5HT2 antagonists |
IL112764A0 (en) * | 1994-03-18 | 1995-05-26 | Ferrer Int | New chromene derivatives |
DE4410822A1 (de) * | 1994-03-24 | 1995-09-28 | Schering Ag | Neue Piperidin-Derivate |
US5880128A (en) * | 1996-05-08 | 1999-03-09 | Schering Corporation | Carbonyl piperazinyl and piperidinyl compounds |
CN1571782A (zh) * | 2001-10-17 | 2005-01-26 | 先灵公司 | 作为3型17β-羟基类固醇脱氢酶抑制剂用于治疗雄激素依赖疾病的哌啶乙酰胺类化合物和哌嗪乙酰胺类化合物 |
US6770659B2 (en) * | 2002-08-26 | 2004-08-03 | Sk Corporation | Benzoyl piperidine compounds |
US20080312281A1 (en) * | 2004-12-24 | 2008-12-18 | Matthew Colin Thor Fyfe | G-Protein Coupled Receptor (Gpr116) Agonists and Use Thereof for Treating Obesity and Diabetes |
NZ564759A (en) * | 2005-06-30 | 2011-08-26 | Prosidion Ltd | GPCR agonists |
RS51647B (en) * | 2006-10-18 | 2011-10-31 | Pfizer Products Inc. | BIARIL ETAR UREE UNITS |
ES2373181T3 (es) * | 2007-01-04 | 2012-02-01 | Prosidion Ltd | Agonistas de gpcr de piperidina. |
CL2008000017A1 (es) * | 2007-01-04 | 2008-08-01 | Prosidion Ltd | Compuestos derivados de heterociclos de nitrogeno y oxigeno, agonistas de gpcr; composicion farmaceutica que comprende a dicho compuesto; y uso del compuesto para el tratamiento de la obesidad, diabetes, sindrome metabolico, hiperlipidemia, toleranci |
CL2008000018A1 (es) * | 2007-01-04 | 2008-08-01 | Prosidion Ltd | Compuestos derivados de heterociclos de nitrogeno y oxigeno, agonistas de gpcr; composicion farmaceutica que comprende a dicho compuesto; y uso del compuesto para el tratamiento de la obesidad, diabetes, sindrome metabolico, hiperlipidemia, toleranci |
DE102011118614B9 (de) | 2011-11-16 | 2013-08-22 | Johannes Herrnsdorf | Kopfunterlage, System zum Abstellen von Schnarchen und Verfahren hierzu |
Family Cites Families (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US3029244A (en) * | 1959-08-31 | 1962-04-10 | Research Corp | Aroylpiperidinols and esters thereof |
-
1968
- 1968-06-20 US US738420A patent/US3576810A/en not_active Expired - Lifetime
-
1969
- 1969-06-16 IE IE821/69A patent/IE33848B1/xx unknown
- 1969-06-16 BR BR209774/69A patent/BR6909774D0/pt unknown
- 1969-06-18 SE SE6908681A patent/SE377118B/xx unknown
- 1969-06-18 GB GB30871/69A patent/GB1268909A/en not_active Expired
- 1969-06-18 BE BE734755D patent/BE734755A/xx not_active IP Right Cessation
- 1969-06-18 DE DE1930818A patent/DE1930818C3/de not_active Expired
- 1969-06-19 FI FI691833A patent/FI51347C/fi active
- 1969-06-19 CH CH145673A patent/CH555335A/xx not_active IP Right Cessation
- 1969-06-19 IL IL32431A patent/IL32431A/xx unknown
- 1969-06-19 NL NL6909384.A patent/NL158488B/xx not_active IP Right Cessation
- 1969-06-19 CH CH940769A patent/CH555334A/xx not_active IP Right Cessation
- 1969-06-19 ES ES368552A patent/ES368552A1/es not_active Expired
- 1969-06-19 CA CA054,803A patent/CA991642A/en not_active Expired
- 1969-06-19 NO NO2524/69A patent/NO136493C/no unknown
- 1969-06-19 DK DK330369A patent/DK132947C/da not_active IP Right Cessation
- 1969-06-20 TR TR17521A patent/TR17521A/xx unknown
- 1969-06-20 AT AT587569A patent/AT291258B/de not_active IP Right Cessation
- 1969-06-20 FR FR6920789A patent/FR2011339A1/fr not_active Withdrawn
- 1969-06-20 JP JP44048351A patent/JPS5022033B1/ja active Pending
-
1973
- 1973-12-30 MY MY424/73A patent/MY7300424A/xx unknown
-
1974
- 1974-11-20 JP JP49133473A patent/JPS5112633B1/ja active Pending
Also Published As
Publication number | Publication date |
---|---|
NO136493B (xx) | 1977-06-06 |
BE734755A (xx) | 1969-12-01 |
FR2011339A1 (xx) | 1970-02-27 |
AT291258B (de) | 1971-07-12 |
NO136493C (no) | 1977-09-14 |
SE377118B (xx) | 1975-06-23 |
IL32431A0 (en) | 1969-08-27 |
IL32431A (en) | 1974-05-16 |
BR6909774D0 (pt) | 1973-02-08 |
JPS5112633B1 (xx) | 1976-04-21 |
DE1930818A1 (de) | 1970-01-08 |
TR17521A (tr) | 1975-07-23 |
NL6909384A (xx) | 1969-12-23 |
CH555335A (de) | 1974-10-31 |
IE33848L (en) | 1969-12-20 |
NL158488B (nl) | 1978-11-15 |
DE1930818B2 (de) | 1981-04-09 |
GB1268909A (en) | 1972-03-29 |
MY7300424A (en) | 1973-12-31 |
DK132947B (da) | 1976-03-01 |
FI51347B (xx) | 1976-08-31 |
JPS5022033B1 (xx) | 1975-07-28 |
CH555334A (de) | 1974-10-31 |
IE33848B1 (en) | 1974-11-27 |
CA991642A (en) | 1976-06-22 |
US3576810A (en) | 1971-04-27 |
DK132947C (da) | 1976-08-02 |
FI51347C (fi) | 1976-12-10 |
DE1930818C3 (de) | 1982-05-06 |
Similar Documents
Publication | Publication Date | Title |
---|---|---|
ES368552A1 (es) | Un procedimiento para la preparacion de i - sustituido - 4 - aroilpiperidinas. | |
KR100244626B1 (ko) | 5-ht1a 길항제로서의 피페라진 유도체, 이의 제조방법 및 이를 함유하는 약제학적 조성물 | |
ES8607234A1 (es) | Un procedimiento para la preparacion de derivados de indol. | |
GB992732A (en) | 1-arylalkyl-4-(n-arylalkanamido)piperidines and related compounds and method for their preparation | |
US3852338A (en) | N-substituted phenylalanine derivatives | |
US3712924A (en) | Halo-substituted 2-amino-benzylamineamides and salts thereof | |
US3789073A (en) | Adamantylalkylaminoalkyl benzamides | |
US6818644B1 (en) | Substituted piperazine derivatives, the preparation thereof and their use as medicaments | |
DE3164741D1 (en) | 2-(4-(diphenylmethylene)-1-piperidinyl)-acetic acids and their amides, their preparation and pharmaceutical preparations containing them | |
US3772308A (en) | Cyclopentanecetamides and cyclopentaneacetonitriles | |
ES8609212A1 (es) | Un procedimiento para la preparacion de derivados de etanolamina. | |
EP0356152B1 (en) | Quaternary ammonium salts | |
IL45995A (en) | 4-pyridylthiazole-2-carboxamides and acetamides their preparation and pharmaceutical compositions containing them | |
HUT37131A (en) | Process for producing 5,10-dihydro-11h-dibenzo/b,e//1,4/diazepin-11-one derivatives substitutes at the 5 position and pharmaceutical compositions containing them | |
KR870002053A (ko) | P-아실아미노벤즈아미드의 제조 방법 | |
GB1027963A (en) | Quinoline derivatives | |
US4758585A (en) | Saturated cycloalkyl (B) pyrrol-1 (2H)- acetic acid amides and derivatives thereof | |
US3702327A (en) | N-beta-1-(3-phenylimidazolidin-2-one)ethyl 4,4-ethylene dioxypiperidines | |
GB1490771A (en) | 2-substituted 4,5-diphenylthiazoles and synthesis thereof | |
ES8602762A1 (es) | Metodo de obtener compuestos utiles como agentes inhibidores de la agregacion de plaquetas | |
US3352865A (en) | Alkyl phenylpiperazinylalkylcarbamates | |
EP0018107B1 (en) | Oxazoline and thiazoline derivatives, processes for their preparation and pharmaceutical compositions containing them | |
ES8606258A1 (es) | Procedimiento de preparacion de eteres oximas basicos, y de sus sales de adicion acidas farmaceuticamente aceptables | |
RU2006113947A (ru) | Амидины и их производные и содержащие их фармацевтические композиции | |
EP0219706B1 (en) | N,n-dialkylaminoalkyl-hexahydro-5-oxo-1h-pyrrolizine-3-carboxamides |