ES329444A1 - Procedure for the preparation of new substituted basic replacement aril-alkil. (Machine-translation by Google Translate, not legally binding) - Google Patents

Procedure for the preparation of new substituted basic replacement aril-alkil. (Machine-translation by Google Translate, not legally binding)

Info

Publication number
ES329444A1
ES329444A1 ES0329444A ES329444A ES329444A1 ES 329444 A1 ES329444 A1 ES 329444A1 ES 0329444 A ES0329444 A ES 0329444A ES 329444 A ES329444 A ES 329444A ES 329444 A1 ES329444 A1 ES 329444A1
Authority
ES
Spain
Prior art keywords
general formula
translation
formula
carbon atoms
preparation
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
ES0329444A
Other languages
Spanish (es)
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Novartis AG
Original Assignee
JR Geigy AG
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from CH1044465A external-priority patent/CH458347A/en
Application filed by JR Geigy AG filed Critical JR Geigy AG
Publication of ES329444A1 publication Critical patent/ES329444A1/en
Expired legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D491/00—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00
    • C07D491/02—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains two hetero rings
    • C07D491/10—Spiro-condensed systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D207/00—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D207/02—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D207/04—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
    • C07D207/10—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D207/12—Oxygen or sulfur atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D211/00—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
    • C07D211/04—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D211/06—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
    • C07D211/36—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D211/40—Oxygen atoms
    • C07D211/44—Oxygen atoms attached in position 4
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D211/00—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
    • C07D211/04—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D211/68—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having one double bond between ring members or between a ring member and a non-ring member
    • C07D211/72—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having one double bond between ring members or between a ring member and a non-ring member with hetero atoms or with carbon atoms having three bonds to hetero atoms, with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D211/74—Oxygen atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D495/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
    • C07D495/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
    • C07D495/10—Spiro-condensed systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D497/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having oxygen and sulfur atoms as the only ring hetero atoms
    • C07D497/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having oxygen and sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
    • C07D497/10—Spiro-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Compositions Of Macromolecular Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)

Abstract

Process for the preparation of new substituted basic aryl alkyl ketones of the general formula I, ** (See formula) ** in which X and Y mean, independently of each other, oxygen or sulfur, R1 means a bivalent hydrocarbon radical with 2-11 carbon atoms, which combines X and Y on 2-4 carbon atoms, and does not carry unsaturated bonds in the two terminal carbon atoms, R2, R3 and R4 mean, independently of each other, hydrogen, lower alkyl or alkoxy radicals or chlorine atoms, and R2 and R3 together signify, beside hydrogen as R4, also the methylenedioxy radical, and R5 means hydrogen, the methyl or ethyl radical, and its addition salts with inorganic and organic acids, characterized in that a compound of the general formula II, ** (See formula) ** wherein R2, R3, R4 and R5 have the same significance indicated in formula I, a mineral acid salt of a compound of the general formula III, ** (See formula) ** where R1, X and Y have the same significance given above, and formaldehyde are reacted together, and the obtained compound of the general formula I, if desired, is transformed into a salt with an inorganic or organic acid. (Machine-translation by Google Translate, not legally binding)
ES0329444A 1965-07-26 1966-07-23 Procedure for the preparation of new substituted basic replacement aril-alkil. (Machine-translation by Google Translate, not legally binding) Expired ES329444A1 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
CH1044465A CH458347A (en) 1965-07-26 1965-07-26 Process for the preparation of new, basic substituted aryl-alkyl-ketones
CH867066 1966-06-15

Publications (1)

Publication Number Publication Date
ES329444A1 true ES329444A1 (en) 1967-05-16

Family

ID=25703605

Family Applications (3)

Application Number Title Priority Date Filing Date
ES0329444A Expired ES329444A1 (en) 1965-07-26 1966-07-23 Procedure for the preparation of new substituted basic replacement aril-alkil. (Machine-translation by Google Translate, not legally binding)
ES0329446A Expired ES329446A1 (en) 1965-07-26 1966-07-23 Procedure for the preparation of new substituted basic replacement aril-alkil. (Machine-translation by Google Translate, not legally binding)
ES0329445A Expired ES329445A1 (en) 1965-07-26 1966-07-23 Procedure for the preparation of new substituted basic replacement aril-alkil. (Machine-translation by Google Translate, not legally binding)

Family Applications After (2)

Application Number Title Priority Date Filing Date
ES0329446A Expired ES329446A1 (en) 1965-07-26 1966-07-23 Procedure for the preparation of new substituted basic replacement aril-alkil. (Machine-translation by Google Translate, not legally binding)
ES0329445A Expired ES329445A1 (en) 1965-07-26 1966-07-23 Procedure for the preparation of new substituted basic replacement aril-alkil. (Machine-translation by Google Translate, not legally binding)

Country Status (5)

Country Link
BE (1) BE684556A (en)
ES (3) ES329444A1 (en)
GB (1) GB1112096A (en)
IL (1) IL26208A (en)
SE (1) SE306742B (en)

Also Published As

Publication number Publication date
SE306742B (en) 1968-12-09
ES329445A1 (en) 1967-11-16
GB1112096A (en) 1968-05-01
IL26208A (en) 1970-08-19
ES329446A1 (en) 1967-05-16
BE684556A (en) 1967-01-25

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