ES2867799T3 - Compuestos para tratar afecciones pruríticas - Google Patents
Compuestos para tratar afecciones pruríticas Download PDFInfo
- Publication number
- ES2867799T3 ES2867799T3 ES16784019T ES16784019T ES2867799T3 ES 2867799 T3 ES2867799 T3 ES 2867799T3 ES 16784019 T ES16784019 T ES 16784019T ES 16784019 T ES16784019 T ES 16784019T ES 2867799 T3 ES2867799 T3 ES 2867799T3
- Authority
- ES
- Spain
- Prior art keywords
- compound
- composition
- alkyl
- nalbuphine
- acid
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
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Classifications
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D489/00—Heterocyclic compounds containing 4aH-8, 9 c- Iminoethano-phenanthro [4, 5-b, c, d] furan ring systems, e.g. derivatives of [4, 5-epoxy]-morphinan of the formula:
- C07D489/06—Heterocyclic compounds containing 4aH-8, 9 c- Iminoethano-phenanthro [4, 5-b, c, d] furan ring systems, e.g. derivatives of [4, 5-epoxy]-morphinan of the formula: with a hetero atom directly attached in position 14
- C07D489/08—Oxygen atom
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
- A61P17/04—Antipruritics
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Dermatology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicinal Preparation (AREA)
- Steroid Compounds (AREA)
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| PCT/US2016/029024 WO2016172613A1 (en) | 2015-04-23 | 2016-04-22 | Compounds for treating pruritic conditions |
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| US4477456A (en) | 1981-07-02 | 1984-10-16 | E. I. Du Pont De Nemours And Company | Octahydro-4A,7-ethano- and -etheno-benzofuro[3,2-e]isoquinoline derivatives having analgesic, narcotic antagonist and anorexigenic properties |
| US7195882B2 (en) * | 2003-06-03 | 2007-03-27 | Roche Diagnostics Operations, Inc. | Monoclonal antibodies specific for buprenorphine and metabolites thereof |
| CA2682125C (en) * | 2007-03-29 | 2015-06-16 | Progenics Pharmaceuticals, Inc. | Peripheral opioid receptor antagonists and uses thereof |
| EP2935278B1 (en) * | 2012-12-19 | 2017-03-15 | Novartis AG | Tricyclic compounds for inhibiting the cftr channel |
-
2016
- 2016-04-22 CA CA2981625A patent/CA2981625C/en active Active
- 2016-04-22 EP EP16784019.8A patent/EP3286198B1/en active Active
- 2016-04-22 WO PCT/US2016/029024 patent/WO2016172613A1/en not_active Ceased
- 2016-04-22 PL PL16784019T patent/PL3286198T3/pl unknown
- 2016-04-22 ES ES16784019T patent/ES2867799T3/es active Active
- 2016-04-22 SI SI201631169T patent/SI3286198T1/sl unknown
- 2016-04-22 DK DK16784019.8T patent/DK3286198T3/da active
- 2016-04-22 LT LTEP16784019.8T patent/LT3286198T/lt unknown
- 2016-04-22 HU HUE16784019A patent/HUE054399T2/hu unknown
- 2016-04-22 PT PT167840198T patent/PT3286198T/pt unknown
- 2016-04-22 AU AU2016252892A patent/AU2016252892B2/en active Active
- 2016-04-22 JP JP2017555210A patent/JP6744327B2/ja active Active
- 2016-04-22 HR HRP20210606TT patent/HRP20210606T1/hr unknown
- 2016-04-22 US US15/136,742 patent/US9624233B2/en active Active
-
2021
- 2021-05-18 CY CY20211100427T patent/CY1124163T1/el unknown
Also Published As
| Publication number | Publication date |
|---|---|
| EP3286198A4 (en) | 2018-09-26 |
| AU2016252892A1 (en) | 2017-10-26 |
| CA2981625A1 (en) | 2016-10-27 |
| EP3286198A1 (en) | 2018-02-28 |
| CA2981625C (en) | 2023-05-23 |
| CY1124163T1 (el) | 2022-05-27 |
| PL3286198T3 (pl) | 2021-09-06 |
| EP3286198B1 (en) | 2021-02-24 |
| HUE054399T2 (hu) | 2021-09-28 |
| HRP20210606T1 (hr) | 2021-05-28 |
| DK3286198T3 (da) | 2021-05-03 |
| SI3286198T1 (sl) | 2021-08-31 |
| AU2016252892B2 (en) | 2019-05-02 |
| US20160311832A1 (en) | 2016-10-27 |
| PT3286198T (pt) | 2021-04-26 |
| LT3286198T (lt) | 2021-07-12 |
| JP2018513174A (ja) | 2018-05-24 |
| US9624233B2 (en) | 2017-04-18 |
| JP6744327B2 (ja) | 2020-08-19 |
| WO2016172613A1 (en) | 2016-10-27 |
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