ES2693520T3 - Quinazolinas sustituidas con sulfoximina para composiciones farmacéuticas - Google Patents
Quinazolinas sustituidas con sulfoximina para composiciones farmacéuticas Download PDFInfo
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- ES2693520T3 ES2693520T3 ES14808895.8T ES14808895T ES2693520T3 ES 2693520 T3 ES2693520 T3 ES 2693520T3 ES 14808895 T ES14808895 T ES 14808895T ES 2693520 T3 ES2693520 T3 ES 2693520T3
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- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
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- C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
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Landscapes
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- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
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Applications Claiming Priority (3)
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| EP13195720 | 2013-12-04 | ||
| EP13195720 | 2013-12-04 | ||
| PCT/EP2014/075890 WO2015082324A1 (en) | 2013-12-04 | 2014-11-28 | Sulfoximine substituted quinazolines for pharmaceutical compositions |
Publications (1)
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| ES2693520T3 true ES2693520T3 (es) | 2018-12-12 |
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| ES14808895.8T Active ES2693520T3 (es) | 2013-12-04 | 2014-11-28 | Quinazolinas sustituidas con sulfoximina para composiciones farmacéuticas |
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| EP (1) | EP3077383B1 (https=) |
| JP (1) | JP6457523B2 (https=) |
| AU (1) | AU2014359456B2 (https=) |
| CA (1) | CA2929742C (https=) |
| ES (1) | ES2693520T3 (https=) |
| WO (1) | WO2015082324A1 (https=) |
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| EP3140300B1 (en) * | 2014-05-07 | 2019-08-14 | Evotec International GmbH | Sulfoximine substituted quinazolines for pharmaceutical compositions |
| UY38540A (es) * | 2019-01-14 | 2020-08-31 | Pi Industries Ltd | Compuestos de fenilamidina 3-sustituida, preparación y uso |
| CN112812136B (zh) * | 2019-11-15 | 2022-04-12 | 武汉光谷亚太医药研究院有限公司 | 新型2,3-二氢化茚衍生化合物、制备方法和应用 |
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| US5750471A (en) | 1994-06-08 | 1998-05-12 | E. I. Du Pont De Nemours And Company | Cyclic sulfonamide herbicides |
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| BR0308162A (pt) | 2002-03-01 | 2004-12-07 | Pfizer | Derivados de indolil-uréia de tienopiridinas úteis como agentes antiangiogênicos e métodos para o seu uso |
| GB0315587D0 (en) | 2003-07-03 | 2003-08-13 | Univ Dundee | Anti-inflammatory assay and compounds |
| KR101151932B1 (ko) | 2004-04-08 | 2012-06-01 | 다우 아그로사이언시즈 엘엘씨 | 살충성 ｎ-치환된 설폭시민 |
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| CA2646429A1 (en) | 2006-03-09 | 2007-09-13 | Pharmacopeia, Inc. | 8-heteroarylpurine mnk2 inhibitors for treating metabolic disorders |
| CA2651898A1 (en) * | 2006-04-07 | 2007-10-18 | Develogen Aktiengesellschaft | Thienopyrimidines having mnk1/mnk2 inhibiting activity for pharmaceutical compositions |
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| DE102007024470A1 (de) | 2007-05-24 | 2008-11-27 | Bayer Schering Pharma Aktiengesellschaft | Neue Sulfoximin-substituierte Chinolin- bzw. Chinazolinderivate als Kinase-Inhibitoren |
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| EP2500340A1 (en) | 2008-01-25 | 2012-09-19 | Syngenta Participations AG. | 2-Cyanophenyl Sulfonamide Derivatives Useful as Pesticides |
| US20120232073A1 (en) | 2009-11-23 | 2012-09-13 | Santhosh Francis Neelamkavil | Fused bicyclic pyrimidine derivatives and methods of use thereof |
| EP2539343B1 (en) | 2010-02-26 | 2015-12-30 | Evotec International GmbH | Thienopyrimidines containing a substituted alkyl group for pharmaceutical compositions |
| UY33241A (es) * | 2010-02-26 | 2011-09-30 | Boehringer Ingelheim Int | ?Tienopirimidinas que contienen heterocicloalquilo para composiciones farmacéuticas?. |
| AR088082A1 (es) | 2011-10-13 | 2014-05-07 | Lilly Co Eli | Moduladores selectivos del receptor androgeno |
| WO2014072244A1 (en) * | 2012-11-09 | 2014-05-15 | Boehringer Ingelheim International Gmbh | Sulfoximine substituted quinazolines for pharmaceutical compositions |
| DK3013805T3 (en) * | 2013-06-28 | 2018-04-23 | Evotec Int Gmbh | Sulfoximine-substituted quinazolines and their use as MNK1 and / or MNK2 kinase inhibitors |
-
2014
- 2014-11-28 CA CA2929742A patent/CA2929742C/en active Active
- 2014-11-28 WO PCT/EP2014/075890 patent/WO2015082324A1/en not_active Ceased
- 2014-11-28 ES ES14808895.8T patent/ES2693520T3/es active Active
- 2014-11-28 JP JP2016536528A patent/JP6457523B2/ja not_active Expired - Fee Related
- 2014-11-28 AU AU2014359456A patent/AU2014359456B2/en not_active Ceased
- 2014-11-28 US US15/101,620 patent/US10093660B2/en active Active
- 2014-11-28 EP EP14808895.8A patent/EP3077383B1/en active Active
Also Published As
| Publication number | Publication date |
|---|---|
| AU2014359456B2 (en) | 2019-01-24 |
| US10093660B2 (en) | 2018-10-09 |
| CA2929742C (en) | 2022-09-20 |
| EP3077383A1 (en) | 2016-10-12 |
| AU2014359456A1 (en) | 2016-06-09 |
| EP3077383B1 (en) | 2018-08-22 |
| JP2016539148A (ja) | 2016-12-15 |
| WO2015082324A1 (en) | 2015-06-11 |
| CA2929742A1 (en) | 2015-06-11 |
| JP6457523B2 (ja) | 2019-01-23 |
| US20170174668A1 (en) | 2017-06-22 |
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