ES2579628T3 - Iminoazúcares y métodos de tratamiento de enfermedades virales - Google Patents
Iminoazúcares y métodos de tratamiento de enfermedades virales Download PDFInfo
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- ES2579628T3 ES2579628T3 ES10744432.5T ES10744432T ES2579628T3 ES 2579628 T3 ES2579628 T3 ES 2579628T3 ES 10744432 T ES10744432 T ES 10744432T ES 2579628 T3 ES2579628 T3 ES 2579628T3
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- 229940095064 tartrate Drugs 0.000 description 1
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Classifications
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
- A61K31/445—Non condensed piperidines, e.g. piperocaine
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/70—Carbohydrates; Sugars; Derivatives thereof
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/66—Phosphorus compounds
- A61K31/665—Phosphorus compounds having oxygen as a ring hetero atom, e.g. fosfomycin
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/12—Antivirals
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/12—Antivirals
- A61P31/14—Antivirals for RNA viruses
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/12—Antivirals
- A61P31/20—Antivirals for DNA viruses
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D211/00—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
- C07D211/04—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D211/06—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
- C07D211/36—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D211/40—Oxygen atoms
- C07D211/44—Oxygen atoms attached in position 4
- C07D211/46—Oxygen atoms attached in position 4 having a hydrogen atom as the second substituent in position 4
-
- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
- Y02A—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE
- Y02A50/00—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE in human health protection, e.g. against extreme weather
- Y02A50/30—Against vector-borne diseases, e.g. mosquito-borne, fly-borne, tick-borne or waterborne diseases whose impact is exacerbated by climate change
Landscapes
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Veterinary Medicine (AREA)
- Pharmacology & Pharmacy (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Medicinal Chemistry (AREA)
- Epidemiology (AREA)
- Organic Chemistry (AREA)
- Virology (AREA)
- Molecular Biology (AREA)
- Communicable Diseases (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Oncology (AREA)
- Engineering & Computer Science (AREA)
- Biotechnology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Saccharide Compounds (AREA)
Applications Claiming Priority (5)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US20236709P | 2009-02-23 | 2009-02-23 | |
| US202367P | 2009-02-23 | ||
| US27225509P | 2009-09-04 | 2009-09-04 | |
| US272255P | 2009-09-04 | ||
| PCT/US2010/024920 WO2010096764A1 (en) | 2009-02-23 | 2010-02-22 | Iminosugars and methods of treating viral diseases |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ES2579628T3 true ES2579628T3 (es) | 2016-08-12 |
Family
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Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ES10744432.5T Active ES2579628T3 (es) | 2009-02-23 | 2010-02-22 | Iminoazúcares y métodos de tratamiento de enfermedades virales |
Country Status (8)
| Country | Link |
|---|---|
| US (4) | US8450345B2 (enExample) |
| EP (1) | EP2398321B1 (enExample) |
| JP (3) | JP5600329B2 (enExample) |
| KR (2) | KR20120042716A (enExample) |
| CN (2) | CN106420740A (enExample) |
| CA (1) | CA2753195C (enExample) |
| ES (1) | ES2579628T3 (enExample) |
| WO (1) | WO2010096764A1 (enExample) |
Families Citing this family (8)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CA2875975A1 (en) | 2012-06-06 | 2013-12-12 | Unither Virology, Llc | Novel iminosugars and their applications |
| WO2014143999A1 (en) * | 2013-03-15 | 2014-09-18 | Unither Virology, Llc | Antibacterial compounds |
| CA2924026C (en) * | 2013-09-16 | 2021-12-28 | Emergent Virology Llc | Deoxynojirimycin derivatives and methods of their using |
| CA2966893C (en) | 2014-11-05 | 2023-10-24 | Emergent Virology Llc | Iminosugars |
| US20190282558A1 (en) * | 2016-05-16 | 2019-09-19 | Emergent Virology Llc | Methods of Treating Zika Virus Infection |
| KR101942757B1 (ko) | 2017-08-23 | 2019-01-28 | 주식회사 유앤아이미트 | 마이크로웨이브를 이용한 n-노닐데옥시노지리마이신의 제조방법 |
| CN113425720A (zh) * | 2020-04-03 | 2021-09-24 | 深圳前海诺贝尔奖科学家技术转移转化有限公司 | 亚胺糖化合物在制备抗SARS-CoV-2病毒的药物中的用途 |
| CN119841765B (zh) * | 2025-01-09 | 2025-10-10 | 中南大学 | Dnj衍生物、药物组合物及其应用 |
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| DE2834122A1 (de) | 1978-08-03 | 1980-02-14 | Bayer Ag | Verfahren zur herstellung von 6-amino-6-desoxy-l-sorbose |
| DE2839309A1 (de) | 1978-09-09 | 1980-03-27 | Bayer Ag | 3,4,5-trihydroxypiperidin-derivate |
| DE2853573A1 (de) | 1978-12-12 | 1980-07-03 | Bayer Ag | Herstellung von n-substituierten derivaten des l-desoxynojirimycins |
| DE3038901A1 (de) | 1980-10-15 | 1982-05-06 | Bayer Ag, 5090 Leverkusen | Verfahren zur herstellung von n-substituierten derivaten des 1-desoxynojirimycins |
| DE3611841A1 (de) | 1986-04-09 | 1987-10-15 | Bayer Ag | Verfahren zur herstellung von 1-desoxynojirimycin und dessen n-derivaten |
| US5043273A (en) | 1989-08-17 | 1991-08-27 | Monsanto Company | Phosphorylated glycosidase inhibitor prodrugs |
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| KR20100127842A (ko) | 2008-03-26 | 2010-12-06 | 유니버시티 오브 옥스퍼드 | 소포체 표적화 리포좀 |
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| WO2010144759A1 (en) | 2009-06-12 | 2010-12-16 | United Therapeutics Corporation | Iminosugars and methods of treating bunyaviral and togaviral diseases |
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| JP5575246B2 (ja) | 2009-09-04 | 2014-08-20 | ユナイテッド セラピューティクス コーポレイション | ポックスウイルス感染の治療方法 |
| EP2473482B1 (en) | 2009-09-04 | 2014-03-05 | United Therapeutics Corporation | Methods of treating orthomyxoviral infections |
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2010
- 2010-02-22 ES ES10744432.5T patent/ES2579628T3/es active Active
- 2010-02-22 CN CN201610416182.XA patent/CN106420740A/zh active Pending
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- 2010-02-22 CN CN201080017591.3A patent/CN102655746B/zh not_active Expired - Fee Related
- 2010-02-22 WO PCT/US2010/024920 patent/WO2010096764A1/en not_active Ceased
- 2010-02-22 CA CA2753195A patent/CA2753195C/en not_active Expired - Fee Related
- 2010-02-22 KR KR1020117021770A patent/KR20120042716A/ko not_active Ceased
- 2010-02-22 JP JP2011551274A patent/JP5600329B2/ja not_active Expired - Fee Related
- 2010-02-22 KR KR1020157006783A patent/KR101755133B1/ko not_active Expired - Fee Related
- 2010-02-22 EP EP10744432.5A patent/EP2398321B1/en not_active Not-in-force
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2013
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Also Published As
| Publication number | Publication date |
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| EP2398321A1 (en) | 2011-12-28 |
| US8450345B2 (en) | 2013-05-28 |
| US20170304333A1 (en) | 2017-10-26 |
| JP5940607B2 (ja) | 2016-06-29 |
| HK1165221A1 (zh) | 2012-10-05 |
| KR101755133B1 (ko) | 2017-07-06 |
| JP2016175937A (ja) | 2016-10-06 |
| US9943532B2 (en) | 2018-04-17 |
| JP5600329B2 (ja) | 2014-10-01 |
| CN106420740A (zh) | 2017-02-22 |
| JP2012518649A (ja) | 2012-08-16 |
| CN102655746A (zh) | 2012-09-05 |
| EP2398321B1 (en) | 2015-11-25 |
| JP2014237706A (ja) | 2014-12-18 |
| US20100222383A1 (en) | 2010-09-02 |
| CA2753195A1 (en) | 2010-08-26 |
| KR20120042716A (ko) | 2012-05-03 |
| KR20150038684A (ko) | 2015-04-08 |
| US20130237567A1 (en) | 2013-09-12 |
| US9579334B2 (en) | 2017-02-28 |
| EP2398321A4 (en) | 2012-01-04 |
| WO2010096764A1 (en) | 2010-08-26 |
| US9044470B2 (en) | 2015-06-02 |
| CA2753195C (en) | 2015-06-02 |
| CN102655746B (zh) | 2016-08-03 |
| US20150224128A1 (en) | 2015-08-13 |
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