ES245281A1 - Procedimiento para la obtencion de nuevas suifonamidas - Google Patents
Procedimiento para la obtencion de nuevas suifonamidasInfo
- Publication number
- ES245281A1 ES245281A1 ES0245281A ES245281A ES245281A1 ES 245281 A1 ES245281 A1 ES 245281A1 ES 0245281 A ES0245281 A ES 0245281A ES 245281 A ES245281 A ES 245281A ES 245281 A1 ES245281 A1 ES 245281A1
- Authority
- ES
- Spain
- Prior art keywords
- sulphanilamido
- group
- hydrogen
- pyrazolo
- pyrimidine
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired
Links
- -1 sulphanilamido Chemical group 0.000 abstract 7
- 229910052739 hydrogen Inorganic materials 0.000 abstract 6
- 239000001257 hydrogen Substances 0.000 abstract 6
- 125000004169 (C1-C6) alkyl group Chemical group 0.000 abstract 4
- 239000004215 Carbon black (E152) Substances 0.000 abstract 4
- 125000003277 amino group Chemical group 0.000 abstract 4
- 229930195733 hydrocarbon Natural products 0.000 abstract 4
- 150000003839 salts Chemical class 0.000 abstract 4
- JHODSSCKWDXARA-UHFFFAOYSA-N 4-amino-N-(1H-pyrazolo[4,3-d]pyrimidin-3-yl)benzenesulfonamide Chemical class S(=O)(C1=CC=C(C=C1)N)(=O)NC1=NNC=2C=NC=NC21 JHODSSCKWDXARA-UHFFFAOYSA-N 0.000 abstract 3
- UFHFLCQGNIYNRP-UHFFFAOYSA-N Hydrogen Chemical compound [H][H] UFHFLCQGNIYNRP-UHFFFAOYSA-N 0.000 abstract 2
- 239000002253 acid Substances 0.000 abstract 2
- 125000001931 aliphatic group Chemical group 0.000 abstract 2
- 229910052783 alkali metal Inorganic materials 0.000 abstract 2
- 150000001340 alkali metals Chemical class 0.000 abstract 2
- 229910052784 alkaline earth metal Inorganic materials 0.000 abstract 2
- 150000001342 alkaline earth metals Chemical class 0.000 abstract 2
- 150000001875 compounds Chemical class 0.000 abstract 2
- 150000002431 hydrogen Chemical class 0.000 abstract 2
- 125000004435 hydrogen atom Chemical group [H]* 0.000 abstract 2
- 125000002950 monocyclic group Chemical group 0.000 abstract 2
- 238000002360 preparation method Methods 0.000 abstract 2
- KHBQMWCZKVMBLN-UHFFFAOYSA-N Benzenesulfonamide Chemical class NS(=O)(=O)C1=CC=CC=C1 KHBQMWCZKVMBLN-UHFFFAOYSA-N 0.000 abstract 1
- 125000004442 acylamino group Chemical group 0.000 abstract 1
- OGEBRHQLRGFBNV-RZDIXWSQSA-N chembl2036808 Chemical compound C12=NC(NCCCC)=NC=C2C(C=2C=CC(F)=CC=2)=NN1C[C@H]1CC[C@H](N)CC1 OGEBRHQLRGFBNV-RZDIXWSQSA-N 0.000 abstract 1
- 239000000470 constituent Substances 0.000 abstract 1
- 239000006071 cream Substances 0.000 abstract 1
- 239000008298 dragée Substances 0.000 abstract 1
- 239000003937 drug carrier Substances 0.000 abstract 1
- 239000000839 emulsion Substances 0.000 abstract 1
- 150000002430 hydrocarbons Chemical class 0.000 abstract 1
- 230000007062 hydrolysis Effects 0.000 abstract 1
- 238000006460 hydrolysis reaction Methods 0.000 abstract 1
- 125000001449 isopropyl group Chemical group [H]C([H])([H])C([H])(*)C([H])([H])[H] 0.000 abstract 1
- 239000002674 ointment Substances 0.000 abstract 1
- 238000007911 parenteral administration Methods 0.000 abstract 1
- 239000000825 pharmaceutical preparation Substances 0.000 abstract 1
- CCGKZVRTYSYOAR-UHFFFAOYSA-N pyrazolo[4,3-d]pyrimidin-2-amine Chemical class NN1N=C2C=NC=NC2=C1 CCGKZVRTYSYOAR-UHFFFAOYSA-N 0.000 abstract 1
- 239000000243 solution Substances 0.000 abstract 1
- 150000003456 sulfonamides Chemical class 0.000 abstract 1
- 239000000725 suspension Substances 0.000 abstract 1
- 239000003826 tablet Substances 0.000 abstract 1
- 238000011200 topical administration Methods 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| CH5314957A CH367510A (de) | 1957-11-27 | 1957-11-27 | Verfahren zur Herstellung neuer Sulfonamide |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ES245281A1 true ES245281A1 (es) | 1959-06-01 |
Family
ID=4518466
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ES0245281A Expired ES245281A1 (es) | 1957-11-27 | 1958-11-13 | Procedimiento para la obtencion de nuevas suifonamidas |
Country Status (7)
| Country | Link |
|---|---|
| US (1) | US3036070A (es) |
| CH (1) | CH367510A (es) |
| DE (1) | DE1092922B (es) |
| ES (1) | ES245281A1 (es) |
| FR (1) | FR1217070A (es) |
| GB (1) | GB889146A (es) |
| NL (1) | NL233475A (es) |
Families Citing this family (11)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US3134933A (en) * | 1962-08-13 | 1964-05-26 | Varian Associates | Adjustable gap magnet |
| GB9114760D0 (en) * | 1991-07-09 | 1991-08-28 | Pfizer Ltd | Therapeutic agents |
| TW444018B (en) | 1992-12-17 | 2001-07-01 | Pfizer | Pyrazolopyrimidines |
| ES2386420T3 (es) * | 1997-11-12 | 2012-08-20 | Bayer Pharma Aktiengesellschaft | Imidazotriazinonas sustituidas con fenilo en la posición 2 como inhibidores de fosfodiesterasas |
| ES2278927T3 (es) * | 2001-05-09 | 2007-08-16 | Bayer Healthcare Ag | Nuevo uso de imidazotriazinonas de 2-(2-etoxi-5-(4-metil-piperazin-1-sulfonil)-fenil)-5-metil-7-propil-3h-imidazo(5,1-f)(1,2,4)triazin-4-ona. |
| DE10232113A1 (de) | 2002-07-16 | 2004-01-29 | Bayer Ag | Vardenafil Hydrochlorid Trihydrat enthaltende Arzneimittel |
| DE102005009240A1 (de) * | 2005-03-01 | 2006-09-07 | Bayer Healthcare Ag | Arzneiformen mit verbesserten pharmakokinetischen Eigenschaften |
| DE102005009241A1 (de) * | 2005-03-01 | 2006-09-07 | Bayer Healthcare Ag | Arzneiformen mit kontrollierter Bioverfügbarkeit |
| US20090186896A1 (en) * | 2005-09-29 | 2009-07-23 | Bayer Healthcare Ag | PDE Inhibitors and Combinations Thereof for the Treatment of Urological Disorders |
| CN101711153A (zh) * | 2007-06-13 | 2010-05-19 | 拜耳先灵制药股份公司 | 用于治疗听觉损伤的pde抑制剂 |
| AU2010232727A1 (en) | 2009-03-31 | 2011-10-20 | Arqule, Inc. | Substituted heterocyclic compounds |
Family Cites Families (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| FR876296A (fr) * | 1939-05-23 | 1942-11-02 | Deutsche Hydrierwerke Ag | Perfectionnements apportés aux procédés de fabrication de dérivés de sulfonamides |
| FR880590A (fr) * | 1941-05-14 | 1943-03-30 | Deutsche Hydrierwerke Ag | Perfectionnements apportés aux procédés de fabrication de dérivés de sulfonamides |
| FR882813A (fr) * | 1941-05-14 | 1943-06-16 | Deutsche Hydrierwerke Ag | Perfectionnements apportés aux procédés de fabrication de dérivés de sulfonamides |
| DE834995C (de) * | 1941-06-26 | 1952-03-27 | Boehringer & Soehne Gmbh | Verfahren zur Herstellung bactericid wirkender Purine |
| FR880591A (fr) * | 1941-06-28 | 1943-03-30 | Deutsche Hydrierwerke Ag | Perfectionnements apportés aux procédés de fabrication de dérivés de sulfamidescycliques |
| DE889300C (de) * | 1951-11-03 | 1953-09-10 | Erich Rabald Dr | Verfahren zur Herstellung von Sulfonamiden der aza-Purinreihe |
-
1957
- 1957-11-27 CH CH5314957A patent/CH367510A/de unknown
-
1958
- 1958-11-07 DE DEC17804A patent/DE1092922B/de active Pending
- 1958-11-13 ES ES0245281A patent/ES245281A1/es not_active Expired
- 1958-11-20 FR FR779583A patent/FR1217070A/fr not_active Expired
- 1958-11-21 US US775375A patent/US3036070A/en not_active Expired - Lifetime
- 1958-11-21 NL NL233475D patent/NL233475A/xx unknown
- 1958-11-24 GB GB37828/58A patent/GB889146A/en not_active Expired
Also Published As
| Publication number | Publication date |
|---|---|
| US3036070A (en) | 1962-05-22 |
| GB889146A (en) | 1962-02-07 |
| FR1217070A (fr) | 1960-05-02 |
| CH367510A (de) | 1963-02-28 |
| DE1092922B (de) | 1960-11-17 |
| NL233475A (es) | 1964-01-15 |
Similar Documents
| Publication | Publication Date | Title |
|---|---|---|
| ES245281A1 (es) | Procedimiento para la obtencion de nuevas suifonamidas | |
| GB913710A (en) | 2,4-diaminopyrido(2,3-d) pyrimidines and the manufacture thereof | |
| GB1271466A (en) | Thiocarbamic acid derivatives | |
| ES289813A1 (es) | Un procedimiento para preparar derivados benzodiazepinicos | |
| GB1016071A (en) | New guanidine derivatives and process for preparing the same | |
| GB1364294A (en) | 2-styrylquinazoline compounds | |
| GB1494560A (en) | 4-aryl-5-aminoalkyl-4-thiazolin-2-ones and their preparation | |
| GB1272337A (en) | New basic carbamates and preparation thereof | |
| GB1250353A (es) | ||
| GB1173809A (en) | N-Substituted Nor-Morphines | |
| GB1198690A (en) | Improvements in or relating to New Biguanides | |
| ES266848A1 (es) | Un procedimeinto para la producciën de esteres del acido 4-halo-3-sulfamoilbenzoico | |
| GB1421089A (en) | Arginine pyroglutamate and a procedure for its preparation | |
| ES273933A1 (es) | Procedimiento para la producciën de sales de pirimidina | |
| GB1154494A (en) | Novel N-Cycloalkyl-Azabicyclooctanes and Nonanes and Novel Intermediates and process for preparation | |
| ES433357A1 (es) | Un metodo para preparar una formulacion farmaceutica que comprende trimetoprim, sulfacetamida y polimixina. | |
| GB1280887A (en) | New isothiocyano-diphenylamines their production and compositions containing same | |
| GB1113802A (en) | Improvements in or relating to substituted quinolines and the manufacture thereof | |
| GB1056823A (en) | New benzenesulphonyl-ureas and process for their manufacture | |
| GB1284582A (en) | Substituted piperazinopyrimidinones | |
| GB1141266A (en) | Novel n-[substituted-3-pyrrolidinyl]-phthalimides and process for the preparation thereof | |
| GB1364318A (en) | Laurotetanine derivatives | |
| GB1320951A (en) | Adamantyl and adamantylalkyl lactams | |
| GB1200199A (en) | New carbamates of pyridine-methanol derivatives and their production | |
| GB929054A (en) | Improvements in and relating to heterocyclic compounds and the manufacture thereof |