ES2427724T3 - Composiciones farmacéuticas, que contienen mezclas de polímeros y de sustancias activas difícilmente solubles en agua - Google Patents
Composiciones farmacéuticas, que contienen mezclas de polímeros y de sustancias activas difícilmente solubles en agua Download PDFInfo
- Publication number
- ES2427724T3 ES2427724T3 ES07703962T ES07703962T ES2427724T3 ES 2427724 T3 ES2427724 T3 ES 2427724T3 ES 07703962 T ES07703962 T ES 07703962T ES 07703962 T ES07703962 T ES 07703962T ES 2427724 T3 ES2427724 T3 ES 2427724T3
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- 125000000391 vinyl group Chemical group [H]C([*])=C([H])[H] 0.000 description 1
- 229920002554 vinyl polymer Polymers 0.000 description 1
- 239000002544 virustatic Substances 0.000 description 1
- 230000001790 virustatic effect Effects 0.000 description 1
- 239000002023 wood Substances 0.000 description 1
Classifications
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- A61K9/2022—Organic macromolecular compounds
- A61K9/2027—Organic macromolecular compounds obtained by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyvinyl pyrrolidone, poly(meth)acrylates
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- A61K9/16—Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
- A61K9/1605—Excipients; Inactive ingredients
- A61K9/1629—Organic macromolecular compounds
- A61K9/1635—Organic macromolecular compounds obtained by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyvinyl pyrrolidone, poly(meth)acrylates
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- A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
- A61K9/16—Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
- A61K9/1605—Excipients; Inactive ingredients
- A61K9/1629—Organic macromolecular compounds
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- A61K9/20—Pills, tablets, discs, rods
- A61K9/2072—Pills, tablets, discs, rods characterised by shape, structure or size; Tablets with holes, special break lines or identification marks; Partially coated tablets; Disintegrating flat shaped forms
- A61K9/2077—Tablets comprising drug-containing microparticles in a substantial amount of supporting matrix; Multiparticulate tablets
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- A—HUMAN NECESSITIES
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- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
- A61K9/50—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals
- A61K9/5084—Mixtures of one or more drugs in different galenical forms, at least one of which being granules, microcapsules or (coated) microparticles according to A61K9/16 or A61K9/50, e.g. for obtaining a specific release pattern or for combining different drugs
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
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- A61P25/06—Antimigraine agents
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- A—HUMAN NECESSITIES
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
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- A—HUMAN NECESSITIES
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- A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
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- A61P3/00—Drugs for disorders of the metabolism
- A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
- A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/12—Antivirals
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P5/00—Drugs for disorders of the endocrine system
- A61P5/24—Drugs for disorders of the endocrine system of the sex hormones
- A61P5/28—Antiandrogens
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P5/00—Drugs for disorders of the endocrine system
- A61P5/24—Drugs for disorders of the endocrine system of the sex hormones
- A61P5/30—Oestrogens
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P7/00—Drugs for disorders of the blood or the extracellular fluid
- A61P7/12—Antidiuretics, e.g. drugs for diabetes insipidus
Landscapes
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Pharmacology & Pharmacy (AREA)
- Medicinal Chemistry (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Organic Chemistry (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Epidemiology (AREA)
- Diabetes (AREA)
- Pain & Pain Management (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Biomedical Technology (AREA)
- Endocrinology (AREA)
- Psychiatry (AREA)
- Communicable Diseases (AREA)
- Oncology (AREA)
- Ophthalmology & Optometry (AREA)
- Hematology (AREA)
- Virology (AREA)
- Emergency Medicine (AREA)
- Obesity (AREA)
- Rheumatology (AREA)
- Orthopedic Medicine & Surgery (AREA)
- Physical Education & Sports Medicine (AREA)
- Medicinal Preparation (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| DE102006005485 | 2006-02-03 | ||
| DE102006005485 | 2006-02-03 | ||
| PCT/EP2007/050465 WO2007090721A1 (de) | 2006-02-03 | 2007-01-17 | Pharmazeutische zusammensetzungen, enthaltend mischungen aus polymeren und in wasser schlecht löslichen wirkstoffen |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ES2427724T3 true ES2427724T3 (es) | 2013-10-31 |
Family
ID=38229086
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
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| ES07703962T Active ES2427724T3 (es) | 2006-02-03 | 2007-01-17 | Composiciones farmacéuticas, que contienen mezclas de polímeros y de sustancias activas difícilmente solubles en agua |
Country Status (13)
| Country | Link |
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| US (1) | US20090011007A1 (https=) |
| EP (1) | EP1978936B1 (https=) |
| JP (1) | JP2009525300A (https=) |
| KR (1) | KR101387249B1 (https=) |
| CN (1) | CN101370480A (https=) |
| BR (1) | BRPI0707465B8 (https=) |
| CA (1) | CA2641351C (https=) |
| ES (1) | ES2427724T3 (https=) |
| IL (1) | IL191604A (https=) |
| PL (1) | PL1978936T3 (https=) |
| SI (1) | SI1978936T1 (https=) |
| TW (1) | TWI394584B (https=) |
| WO (1) | WO2007090721A1 (https=) |
Families Citing this family (30)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US20100297248A1 (en) * | 2004-09-01 | 2010-11-25 | Board Of Regents, The University Of Texas System | Encapsulated particles for amorphous stability enhancement |
| US20100297251A1 (en) * | 2004-09-01 | 2010-11-25 | Board Of Regents, The University Of Texas System | Encapsulated particles for enteric release |
| US20060045822A1 (en) * | 2004-09-01 | 2006-03-02 | Board Of Regents, The University Of Texas System | Plasma polymerization for encapsulating particles |
| CN101272769B (zh) * | 2005-07-28 | 2013-04-24 | Isp投资有限公司 | 生物利用度提高的苯醌类化合物 |
| GB0607105D0 (en) * | 2006-04-10 | 2006-05-17 | Leuven K U Res & Dev | Enhancing solubility and dissolution rate of poorly soluble drugs |
| PE20080422A1 (es) * | 2006-08-10 | 2008-04-28 | Cipla Ltd | Composicion solida antirretroviral de administracion oral |
| PL382311A1 (pl) * | 2007-04-27 | 2008-11-10 | Zakłady Farmaceutyczne POLPHARMA Spółka Akcyjna | Kompozycja farmaceutyczna o polepszonej stabilności zawierająca inhibitor acetylocholinoesterazy lub farmaceutycznie dopuszczalną jego sól oraz sposób jej wytwarzania |
| US8088451B2 (en) | 2008-03-13 | 2012-01-03 | Board Of Regents, The University Of Texas System | Covalently functionalized particles for synthesis of new composite materials |
| CN103260609B (zh) * | 2010-12-23 | 2017-08-11 | 雅培股份有限两合公司 | 基于固体分散体的固体延缓制剂 |
| EP2550863A1 (de) * | 2011-07-27 | 2013-01-30 | Bayer Intellectual Property GmbH | Aktivstoffhaltige Partikel auf Polyacrylat-Basis |
| US20150011525A1 (en) * | 2011-09-13 | 2015-01-08 | Isp Investments Inc. | Solid dispersion of poorly soluble compounds comprising crospovidone and at least one water-soluble polymer |
| ES2652266T3 (es) * | 2012-04-02 | 2018-02-01 | Pharma Seeds Create, Llc | Composición sólida de dosificación oral de ibuprofeno que comprende un copolímero de ácido metacrílico |
| KR101659983B1 (ko) * | 2012-12-31 | 2016-09-26 | 주식회사 삼양바이오팜 | 용융 압출된 방출 제어용 약학 조성물, 및 이를 포함하는 경구용 제제 |
| JP6052319B2 (ja) * | 2015-03-25 | 2016-12-27 | Ｎｔｔエレクトロニクス株式会社 | 動画像符号化装置 |
| GB201604484D0 (en) | 2016-03-16 | 2016-04-27 | Antibiotx Aps And Københavns Uni University Of Copenhagen | Topical antibacterial compositions |
| US10532632B2 (en) | 2016-06-30 | 2020-01-14 | Emerson Climate Technologies, Inc. | Startup control systems and methods for high ambient conditions |
| US10315495B2 (en) | 2016-06-30 | 2019-06-11 | Emerson Climate Technologies, Inc. | System and method of controlling compressor, evaporator fan, and condenser fan speeds during a battery mode of a refrigeration system for a container of a vehicle |
| US10414241B2 (en) | 2016-06-30 | 2019-09-17 | Emerson Climate Technologies, Inc. | Systems and methods for capacity modulation through eutectic plates |
| US10828963B2 (en) | 2016-06-30 | 2020-11-10 | Emerson Climate Technologies, Inc. | System and method of mode-based compressor speed control for refrigerated vehicle compartment |
| US10569620B2 (en) | 2016-06-30 | 2020-02-25 | Emerson Climate Technologies, Inc. | Startup control systems and methods to reduce flooded startup conditions |
| US10562377B2 (en) | 2016-06-30 | 2020-02-18 | Emerson Climate Technologies, Inc. | Battery life prediction and monitoring |
| US10300766B2 (en) * | 2016-06-30 | 2019-05-28 | Emerson Climate Technologies, Inc. | System and method of controlling passage of refrigerant through eutectic plates and an evaporator of a refrigeration system for a container of a vehicle |
| US10328771B2 (en) | 2016-06-30 | 2019-06-25 | Emerson Climated Technologies, Inc. | System and method of controlling an oil return cycle for a refrigerated container of a vehicle |
| KR20260007295A (ko) | 2018-05-24 | 2026-01-13 | 셀라니즈 이브이에이 퍼포먼스 폴리머스 엘엘씨 | 거대 분자 약물 화합물의 지속적인 방출을 위한 이식가능 장치 |
| US11690806B2 (en) | 2018-05-24 | 2023-07-04 | Celanese Eva Performance Polymers Llc | Implantable device for sustained release of a macromolecular drug compound |
| US11689849B2 (en) | 2018-05-24 | 2023-06-27 | Nureva, Inc. | Method, apparatus and computer-readable media to manage semi-constant (persistent) sound sources in microphone pickup/focus zones |
| CN110755396B (zh) * | 2019-12-06 | 2022-04-08 | 北京悦康科创医药科技股份有限公司 | 一种布洛芬缓释小丸及其制备方法 |
| CN116744917A (zh) | 2020-09-04 | 2023-09-12 | 礼蓝美国公司 | 适口调配物 |
| BR112023022439A2 (pt) | 2021-04-26 | 2023-12-26 | Celanese Eva Performance Polymers Llc | Dispositivo implantável para liberação sustentada de um composto de fármaco macromolecular |
| JP7817300B2 (ja) * | 2023-02-14 | 2026-02-18 | 沢井製薬株式会社 | コーティング顆粒、コーティング顆粒を含む製剤及びそれらの製造方法 |
Family Cites Families (12)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| LU85058A1 (fr) * | 1983-10-24 | 1985-06-19 | Pharlyse | Comprimes pharmaceutiques a liberation prolongee,leur preparation et leur utilisation |
| CA2068402C (en) * | 1991-06-14 | 1998-09-22 | Michael R. Hoy | Taste mask coatings for preparation of chewable pharmaceutical tablets |
| AT403988B (de) * | 1994-05-18 | 1998-07-27 | Lannacher Heilmittel | Festes orales retardpräparat |
| US6391338B1 (en) * | 1995-09-07 | 2002-05-21 | Biovail Technologies Ltd. | System for rendering substantially non-dissoluble bio-affecting agents bio-available |
| US20030064108A1 (en) * | 1996-04-23 | 2003-04-03 | Stefan Lukas | Taste masked pharmaceutical compositions |
| EP1125586A4 (en) * | 1998-10-26 | 2003-06-11 | Tanabe Seiyaku Co | EXTENDED RELEASE PARTICLE |
| FR2795326B1 (fr) * | 1999-06-28 | 2001-08-31 | Adir | Composition pharmaceutique solide thermoformable a liberation controlee |
| US6656492B2 (en) * | 2000-06-30 | 2003-12-02 | Yamanouchi Pharmaceutical Co., Ltd. | Quick disintegrating tablet in buccal cavity and manufacturing method thereof |
| FR2826274B1 (fr) * | 2001-06-21 | 2003-09-26 | Aventis Pharma Sa | Formulation pharmaceutique au gout masque et son procede de preparation |
| WO2004009059A1 (en) * | 2002-07-19 | 2004-01-29 | Aventis Pharma S.A. | Taste masked oral composition of telithromycin |
| DE10304403A1 (de) * | 2003-01-28 | 2004-08-05 | Röhm GmbH & Co. KG | Verfahren zur Herstellung einer oralen Arzneiform mit unmittelbarem Zerfall und Wirkstofffreisetzung |
| EP1734953A4 (en) * | 2004-03-02 | 2008-08-20 | Abeille Pharmaceuticals Inc | CO-PR PARATIONS OF KITS OF BIOACTIVE AGENTS |
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- 2007-01-17 BR BRPI0707465A patent/BRPI0707465B8/pt not_active IP Right Cessation
- 2007-01-17 US US12/159,538 patent/US20090011007A1/en not_active Abandoned
- 2007-01-17 CN CNA2007800030537A patent/CN101370480A/zh active Pending
- 2007-01-17 ES ES07703962T patent/ES2427724T3/es active Active
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- 2007-01-17 KR KR1020087019038A patent/KR101387249B1/ko not_active Expired - Fee Related
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- 2007-01-17 WO PCT/EP2007/050465 patent/WO2007090721A1/de not_active Ceased
- 2007-01-17 EP EP07703962.6A patent/EP1978936B1/de active Active
- 2007-02-01 TW TW096103744A patent/TWI394584B/zh not_active IP Right Cessation
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Also Published As
| Publication number | Publication date |
|---|---|
| EP1978936A1 (de) | 2008-10-15 |
| TW200808357A (en) | 2008-02-16 |
| JP2009525300A (ja) | 2009-07-09 |
| CN101370480A (zh) | 2009-02-18 |
| IL191604A (en) | 2013-05-30 |
| BRPI0707465A2 (pt) | 2011-05-03 |
| KR20080090494A (ko) | 2008-10-08 |
| CA2641351A1 (en) | 2007-08-16 |
| BRPI0707465B8 (pt) | 2022-07-05 |
| EP1978936B1 (de) | 2013-07-10 |
| PL1978936T3 (pl) | 2013-11-29 |
| BRPI0707465B1 (pt) | 2020-01-14 |
| US20090011007A1 (en) | 2009-01-08 |
| IL191604A0 (en) | 2008-12-29 |
| CA2641351C (en) | 2014-05-06 |
| WO2007090721A1 (de) | 2007-08-16 |
| TWI394584B (zh) | 2013-05-01 |
| KR101387249B1 (ko) | 2014-05-21 |
| SI1978936T1 (sl) | 2013-10-30 |
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