ES2405779T3 - Gotas oftálmicas con difluprednato para tratamiento del edema macular - Google Patents
Gotas oftálmicas con difluprednato para tratamiento del edema macular Download PDFInfo
- Publication number
- ES2405779T3 ES2405779T3 ES10739716T ES10739716T ES2405779T3 ES 2405779 T3 ES2405779 T3 ES 2405779T3 ES 10739716 T ES10739716 T ES 10739716T ES 10739716 T ES10739716 T ES 10739716T ES 2405779 T3 ES2405779 T3 ES 2405779T3
- Authority
- ES
- Spain
- Prior art keywords
- administration
- ophthalmic drops
- difluprednate
- macular edema
- weeks
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Active
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- WYQPLTPSGFELIB-JTQPXKBDSA-N Difluprednate Chemical compound C1([C@@H](F)C2)=CC(=O)C=C[C@]1(C)[C@]1(F)[C@@H]2[C@@H]2CC[C@@](C(=O)COC(C)=O)(OC(=O)CCC)[C@@]2(C)C[C@@H]1O WYQPLTPSGFELIB-JTQPXKBDSA-N 0.000 title claims abstract description 65
- 238000011282 treatment Methods 0.000 title claims abstract description 53
- 208000001344 Macular Edema Diseases 0.000 title claims abstract description 47
- 206010025415 Macular oedema Diseases 0.000 title claims abstract description 47
- 201000010230 macular retinal edema Diseases 0.000 title claims abstract description 47
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Classifications
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- A61K31/56—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
- A61K31/57—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids substituted in position 17 beta by a chain of two carbon atoms, e.g. pregnane or progesterone
- A61K31/573—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids substituted in position 17 beta by a chain of two carbon atoms, e.g. pregnane or progesterone substituted in position 21, e.g. cortisone, dexamethasone, prednisone or aldosterone
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- Bioinformatics & Cheminformatics (AREA)
- Biophysics (AREA)
- Molecular Biology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicinal Preparation (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP2009165924 | 2009-07-14 | ||
| JP2009165924 | 2009-07-14 | ||
| PCT/JP2010/062289 WO2011007893A1 (en) | 2009-07-14 | 2010-07-14 | Eye drop with difluprednate for macular edema treatment |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ES2405779T3 true ES2405779T3 (es) | 2013-06-03 |
Family
ID=42646370
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ES10739716T Active ES2405779T3 (es) | 2009-07-14 | 2010-07-14 | Gotas oftálmicas con difluprednato para tratamiento del edema macular |
Country Status (13)
| Country | Link |
|---|---|
| US (3) | US20110190250A1 (https=) |
| EP (1) | EP2340014B1 (https=) |
| JP (1) | JP5579079B2 (https=) |
| KR (1) | KR101689847B1 (https=) |
| CN (3) | CN107569494A (https=) |
| BR (1) | BRPI1005380A2 (https=) |
| CA (1) | CA2738151C (https=) |
| ES (1) | ES2405779T3 (https=) |
| MX (1) | MX2011005043A (https=) |
| PL (1) | PL2340014T3 (https=) |
| RU (1) | RU2572707C2 (https=) |
| TW (1) | TW201105363A (https=) |
| WO (1) | WO2011007893A1 (https=) |
Families Citing this family (15)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| AU2011354895B2 (en) * | 2011-01-14 | 2016-05-05 | Sds Biotech K. K. | Agri-horticultural pest control compositions comprising 4- (3-butynyl)aminopyrimidine derivatives |
| US20140018402A1 (en) * | 2011-03-30 | 2014-01-16 | Catholic University Industry Academic Cooperation Foundation | Pharmaceutical composition for preventing or treating macular degeneration |
| CN103130857A (zh) * | 2011-11-30 | 2013-06-05 | 天津金耀集团有限公司 | 二氟泼尼酯ⅱ晶型及其制备方法 |
| CN103130859B (zh) * | 2011-11-30 | 2015-12-02 | 天津金耀集团有限公司 | 二氟泼尼酯晶型i及其制备方法 |
| EP2956144B1 (en) * | 2013-02-15 | 2017-11-22 | Senju Pharmaceutical Co., Ltd. | Difluprednate emulsion composition containing zinc |
| AU2014233363B2 (en) * | 2013-03-15 | 2017-06-29 | EyePoint, Inc. | Compositions, formulations and methods for treating ocular diseases |
| JP2017528865A (ja) | 2014-06-23 | 2017-09-28 | ショット アクチエンゲゼルシャフトＳｃｈｏｔｔ ＡＧ | 板状の別個の要素を有する蓄電システム、板状の別個の要素、並びにその製造方法、及びその使用 |
| JP2018505515A (ja) | 2014-12-01 | 2018-02-22 | ショット アクチエンゲゼルシャフトＳｃｈｏｔｔ ＡＧ | シート状の独立した部材を有する蓄電システム、独立したシート状の部材、その製造方法、およびその使用 |
| EP3302382A4 (en) * | 2015-05-29 | 2019-02-20 | Allergan, Inc. | IMPLANT FOR THE TREATMENT OF OCULAR DISEASE |
| RU2661621C2 (ru) * | 2016-12-19 | 2018-07-17 | Александр Николаевич Епихин | Способ пролонгации и усиления терапевтического эффекта действия ингибиторов ангиогенеза при лечении неоваскулярных форм макулярных дегенераций |
| CN108014172A (zh) * | 2017-12-29 | 2018-05-11 | 广州仁恒医药科技股份有限公司 | 一种含有二氟泼尼酯的药物组合物及其制备方法 |
| KR20210012346A (ko) | 2019-07-25 | 2021-02-03 | 심낙범 | 미세먼지 눈꺼풀 세정스틱 |
| US20210100856A1 (en) * | 2019-09-11 | 2021-04-08 | Adverum Biotechnologies, Inc. | Methods of treating ocular neovascular diseases using aav2 variants encoding aflibercept |
| HRP20260137T1 (hr) * | 2019-09-11 | 2026-03-13 | Adverum Biotechnologies, Inc. | Liječenje očnih neovaskularnih bolesti upotrebom aav2 varijanti koje kodiraju aflibercept |
| WO2026019885A1 (en) * | 2024-07-16 | 2026-01-22 | Adverum Biotechnologies, Inc. | Methods of treating ocular neovascular diseases using aav2 variants encoding aflibercept |
Family Cites Families (11)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP3781792B2 (ja) | 1993-12-27 | 2006-05-31 | 千寿製薬株式会社 | ジフルプレドナート含有点眼用懸濁液剤 |
| AU684115B2 (en) | 1993-12-27 | 1997-12-04 | Mitsubishi Chemical Corporation | Ophthalmic suspension containing diflupredonate |
| DE69807281T2 (de) * | 1997-05-14 | 2003-04-17 | Mitsubishi Chemical Corp., Tokio/Tokyo | Difluprednat enthaltende Zusammensetzungen |
| JP3410364B2 (ja) | 1997-05-14 | 2003-05-26 | 千寿製薬株式会社 | ジフルプレドナート含有組成物 |
| US20050048099A1 (en) * | 2003-01-09 | 2005-03-03 | Allergan, Inc. | Ocular implant made by a double extrusion process |
| WO2004073607A2 (en) * | 2003-02-20 | 2004-09-02 | Alcon, Inc. | Use of steroids to treat ocular disorders |
| US20050226814A1 (en) * | 2004-04-13 | 2005-10-13 | Bausch & Lomb Incorporated | Diagnostic method and kit for implantation of a sustained release drug-delivery implant with a steroid |
| WO2006017347A2 (en) * | 2004-07-12 | 2006-02-16 | Allergan, Inc. | Opthalmic compositions and methods for treating ophthalmic conditions |
| US20080233053A1 (en) * | 2005-02-07 | 2008-09-25 | Pharmalight Inc. | Method and Device for Ophthalmic Administration of Active Pharmaceutical Ingredients |
| WO2007025275A2 (en) | 2005-08-25 | 2007-03-01 | Psivida Inc. | Control of induced elevated intraocular pressure |
| US20090105245A1 (en) * | 2006-12-21 | 2009-04-23 | Bingaman David P | Methods for treating macular edema and ocular angiogenesis using an anti-inflammatory agent and a receptor tyrosine kinase inhibitor |
-
2010
- 2010-07-13 TW TW099122939A patent/TW201105363A/zh unknown
- 2010-07-14 WO PCT/JP2010/062289 patent/WO2011007893A1/en not_active Ceased
- 2010-07-14 RU RU2011125640/15A patent/RU2572707C2/ru active
- 2010-07-14 CN CN201710195879.3A patent/CN107569494A/zh active Pending
- 2010-07-14 ES ES10739716T patent/ES2405779T3/es active Active
- 2010-07-14 US US13/122,467 patent/US20110190250A1/en not_active Abandoned
- 2010-07-14 MX MX2011005043A patent/MX2011005043A/es active IP Right Grant
- 2010-07-14 KR KR1020117012096A patent/KR101689847B1/ko not_active Expired - Fee Related
- 2010-07-14 JP JP2010545305A patent/JP5579079B2/ja not_active Expired - Fee Related
- 2010-07-14 CN CN2010800027502A patent/CN102170865A/zh active Pending
- 2010-07-14 BR BRPI1005380A patent/BRPI1005380A2/pt not_active Application Discontinuation
- 2010-07-14 PL PL10739716T patent/PL2340014T3/pl unknown
- 2010-07-14 CA CA2738151A patent/CA2738151C/en not_active Expired - Fee Related
- 2010-07-14 EP EP10739716.8A patent/EP2340014B1/en not_active Not-in-force
- 2010-07-14 CN CN201310288639.XA patent/CN103705524A/zh not_active Withdrawn
-
2015
- 2015-03-18 US US14/661,295 patent/US9949926B2/en not_active Expired - Fee Related
-
2018
- 2018-01-10 US US15/866,744 patent/US10092514B2/en not_active Expired - Fee Related
Also Published As
| Publication number | Publication date |
|---|---|
| CA2738151C (en) | 2017-02-28 |
| TW201105363A (en) | 2011-02-16 |
| RU2011125640A (ru) | 2013-08-20 |
| CN102170865A (zh) | 2011-08-31 |
| US10092514B2 (en) | 2018-10-09 |
| MX2011005043A (es) | 2011-06-01 |
| PL2340014T3 (pl) | 2013-09-30 |
| EP2340014B1 (en) | 2013-04-24 |
| EP2340014A1 (en) | 2011-07-06 |
| KR20120040683A (ko) | 2012-04-27 |
| CA2738151A1 (en) | 2011-01-20 |
| US20180133153A1 (en) | 2018-05-17 |
| RU2572707C2 (ru) | 2016-01-20 |
| JP2012533517A (ja) | 2012-12-27 |
| US20110190250A1 (en) | 2011-08-04 |
| WO2011007893A1 (en) | 2011-01-20 |
| JP5579079B2 (ja) | 2014-08-27 |
| CN107569494A (zh) | 2018-01-12 |
| US9949926B2 (en) | 2018-04-24 |
| BRPI1005380A2 (pt) | 2016-02-10 |
| KR101689847B1 (ko) | 2016-12-26 |
| CN103705524A (zh) | 2014-04-09 |
| US20150190340A1 (en) | 2015-07-09 |
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