ES2395408T3 - Composiciones de fármaco lipófilas - Google Patents

Composiciones de fármaco lipófilas Download PDF

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Publication number
ES2395408T3
ES2395408T3 ES02766045T ES02766045T ES2395408T3 ES 2395408 T3 ES2395408 T3 ES 2395408T3 ES 02766045 T ES02766045 T ES 02766045T ES 02766045 T ES02766045 T ES 02766045T ES 2395408 T3 ES2395408 T3 ES 2395408T3
Authority
ES
Spain
Prior art keywords
lipid
drug
substituted
nitrotiazole
composition
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Lifetime
Application number
ES02766045T
Other languages
English (en)
Spanish (es)
Inventor
Michael T. Sung
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Individual
Original Assignee
Individual
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Individual filed Critical Individual
Application granted granted Critical
Publication of ES2395408T3 publication Critical patent/ES2395408T3/es
Anticipated expiration legal-status Critical
Expired - Lifetime legal-status Critical Current

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/50—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates
    • A61K47/51—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates the non-active ingredient being a modifying agent
    • A61K47/54—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates the non-active ingredient being a modifying agent the modifying agent being an organic compound
    • A61K47/543—Lipids, e.g. triglycerides; Polyamines, e.g. spermine or spermidine
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/50—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates
    • A61K47/51—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates the non-active ingredient being a modifying agent
    • A61K47/54—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates the non-active ingredient being a modifying agent the modifying agent being an organic compound
    • A61K47/542—Carboxylic acids, e.g. a fatty acid or an amino acid

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Chemical & Material Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Biophysics (AREA)
  • Molecular Biology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
ES02766045T 2001-08-23 2002-08-21 Composiciones de fármaco lipófilas Expired - Lifetime ES2395408T3 (es)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
US134329 1993-10-12
US31409201P 2001-08-23 2001-08-23
US314092P 2001-08-23
US10/134,329 US7125568B2 (en) 2001-08-23 2002-04-29 Lipophilic drug compositions
PCT/US2002/026571 WO2003018064A2 (en) 2001-08-23 2002-08-21 Lipophilic drug compositions

Publications (1)

Publication Number Publication Date
ES2395408T3 true ES2395408T3 (es) 2013-02-12

Family

ID=26832219

Family Applications (1)

Application Number Title Priority Date Filing Date
ES02766045T Expired - Lifetime ES2395408T3 (es) 2001-08-23 2002-08-21 Composiciones de fármaco lipófilas

Country Status (6)

Country Link
US (2) US7125568B2 (Direct)
EP (1) EP1420828B1 (Direct)
CA (1) CA2458394C (Direct)
ES (1) ES2395408T3 (Direct)
TW (1) TWI302459B (Direct)
WO (1) WO2003018064A2 (Direct)

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WO2007081974A2 (en) 2006-01-09 2007-07-19 Romark Laboratories, L.C. Viral hepatitis treatment
US20100119529A1 (en) * 2006-05-12 2010-05-13 Furgeson Darin Y Elastin-like polymer delivery vehicles
WO2008101173A2 (en) * 2007-02-16 2008-08-21 Cornell University Biodegradable compositions and materials
US8354116B2 (en) * 2007-06-18 2013-01-15 Biochemics, Inc. Bifunctional synthetic molecules
US7790401B2 (en) * 2007-08-06 2010-09-07 Siemens Healthcare Diagnostics Methods for detection of immunosuppressant drugs
TW200936180A (en) * 2007-11-27 2009-09-01 Intervet Int Bv Carrier particle for a microorganism or subunit thereof, pharmaceutical composition comprising such particles, method for preparation of this composition and its use in the treatment of animals
GB0724550D0 (en) * 2007-12-18 2008-01-30 Univ Hull Formulations
GB0812513D0 (en) * 2008-07-09 2008-08-13 Univ Hull Delivery vehicle
US20110082156A1 (en) * 2009-10-05 2011-04-07 Milne Jill C Fatty acid acipimox derivatives and their uses
CA2811931C (en) * 2010-10-20 2015-06-16 Galderma S.A. Method of treating herpes virus infection using macrocyclic lactone compound
JP2016536372A (ja) * 2013-11-05 2016-11-24 ウルトラジェニクス ファーマシューティカル インク．Ｕｌｔｒａｇｅｎｙｘ Ｐｈａｒｍａｃｅｕｔｉｃａｌ Ｉｎｃ． クレアチン類似体及びその使用
EP3475442B1 (en) * 2016-06-23 2024-10-23 The Regents of The University of Michigan 12(s)-hydroxyeicosatrienoic acid compounds and their use as therapeutic agents
AU2018375199B2 (en) 2017-12-01 2023-03-30 Ultragenyx Pharmaceutical Inc. Creatine prodrugs, compositions and methods of use thereof

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DE2655369A1 (de) * 1976-12-03 1978-06-08 Schering Ag 5-(subst. phenyl)-oxazolidinone und deren schwefelanaloga sowie verfahren zu deren herstellung
US4315018A (en) * 1978-12-07 1982-02-09 Rossignol Jean F Specific parasiticidal use of 2-benzamido-5-nitro-thiazole derivatives
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DE3884563T2 (de) 1987-10-21 1994-02-17 Du Pont Merck Pharma Aminomethyl-oxo-oxazolidinyl-ethenylbenzen-Derivate, nützlich als antibakterielles Mittel.
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Also Published As

Publication number Publication date
US7125568B2 (en) 2006-10-24
WO2003018064A3 (en) 2003-09-25
TWI302459B (Direct) 2008-11-01
WO2003018064A2 (en) 2003-03-06
CA2458394C (en) 2013-04-23
US20030108596A1 (en) 2003-06-12
EP1420828A2 (en) 2004-05-26
EP1420828B1 (en) 2012-09-26
CA2458394A1 (en) 2003-03-06
US20060147525A1 (en) 2006-07-06
US7390506B2 (en) 2008-06-24

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