ES2327195B1 - Composiciones de liberacion modificada que comprenden un derivado de fluorocitidina para el tratamiento del cancer. - Google Patents
Composiciones de liberacion modificada que comprenden un derivado de fluorocitidina para el tratamiento del cancer. Download PDFInfo
- Publication number
- ES2327195B1 ES2327195B1 ES200750061A ES200750061A ES2327195B1 ES 2327195 B1 ES2327195 B1 ES 2327195B1 ES 200750061 A ES200750061 A ES 200750061A ES 200750061 A ES200750061 A ES 200750061A ES 2327195 B1 ES2327195 B1 ES 2327195B1
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- composition according
- modified release
- fluorocytidine
- derivative
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Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
- A61K9/50—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals
- A61K9/5073—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals having two or more different coatings optionally including drug-containing subcoatings
- A61K9/5078—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals having two or more different coatings optionally including drug-containing subcoatings with drug-free core
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/70—Carbohydrates; Sugars; Derivatives thereof
- A61K31/7042—Compounds having saccharide radicals and heterocyclic rings
- A61K31/7052—Compounds having saccharide radicals and heterocyclic rings having nitrogen as a ring hetero atom, e.g. nucleosides, nucleotides
- A61K31/706—Compounds having saccharide radicals and heterocyclic rings having nitrogen as a ring hetero atom, e.g. nucleosides, nucleotides containing six-membered rings with nitrogen as a ring hetero atom
- A61K31/7064—Compounds having saccharide radicals and heterocyclic rings having nitrogen as a ring hetero atom, e.g. nucleosides, nucleotides containing six-membered rings with nitrogen as a ring hetero atom containing condensed or non-condensed pyrimidines
- A61K31/7068—Compounds having saccharide radicals and heterocyclic rings having nitrogen as a ring hetero atom, e.g. nucleosides, nucleotides containing six-membered rings with nitrogen as a ring hetero atom containing condensed or non-condensed pyrimidines having oxo groups directly attached to the pyrimidine ring, e.g. cytidine, cytidylic acid
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
Landscapes
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Public Health (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Chemical & Material Sciences (AREA)
- Veterinary Medicine (AREA)
- General Health & Medical Sciences (AREA)
- Epidemiology (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Molecular Biology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Organic Chemistry (AREA)
- Medicinal Preparation (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US67050705P | 2005-04-12 | 2005-04-12 | |
| US60/670,507 | 2005-04-12 |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| ES2327195A1 ES2327195A1 (es) | 2009-10-26 |
| ES2327195B1 true ES2327195B1 (es) | 2010-07-09 |
Family
ID=37087358
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ES200750061A Withdrawn - After Issue ES2327195B1 (es) | 2005-04-12 | 2006-04-12 | Composiciones de liberacion modificada que comprenden un derivado de fluorocitidina para el tratamiento del cancer. |
Country Status (7)
| Country | Link |
|---|---|
| EP (1) | EP1874271A4 (fr) |
| JP (1) | JP2008535920A (fr) |
| CA (1) | CA2604192A1 (fr) |
| DE (1) | DE112006000873T5 (fr) |
| ES (1) | ES2327195B1 (fr) |
| GB (1) | GB2442615A (fr) |
| WO (1) | WO2006110800A1 (fr) |
Families Citing this family (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US20080085310A1 (en) * | 2006-10-06 | 2008-04-10 | Maria Oksana Bachynsky | Capecitabine rapidly disintegrating tablets |
| US20110027374A1 (en) * | 2008-12-16 | 2011-02-03 | Maria Oksana Bachynsky | Capecitabine rapidly disintegrating tablets |
| US20200054659A1 (en) * | 2015-06-13 | 2020-02-20 | Intas Pharmaceuticals Ltd. | Extended release capecitabine capsules |
| BR112019016028A2 (pt) * | 2017-02-06 | 2020-03-31 | Intas Pharmaceuticals Ltd | Composição farmacêutica de capecitabina |
Family Cites Families (7)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US6586006B2 (en) * | 1994-08-04 | 2003-07-01 | Elan Drug Delivery Limited | Solid delivery systems for controlled release of molecules incorporated therein and methods of making same |
| DE69735002T2 (de) * | 1996-10-25 | 2006-10-26 | Shire Laboratories, Inc. | Osmotisches Verabreichungssystem für lösliche Dosen |
| US6005098A (en) * | 1998-02-06 | 1999-12-21 | Hoffmann-La Roche Inc. | 5'deoxycytidine derivatives |
| PL205109B1 (pl) * | 1998-11-02 | 2010-03-31 | Elan Pharma Int Ltd | Wielocząstkowa kompozycja metylofenidatu o modyfikowanym uwalnianiu i jej zastosowanie |
| US6248363B1 (en) * | 1999-11-23 | 2001-06-19 | Lipocine, Inc. | Solid carriers for improved delivery of active ingredients in pharmaceutical compositions |
| EA005619B1 (ru) * | 2000-02-28 | 2005-04-28 | Авентис Фарма С.А. | Композиция, включающая камптотецин и производное пиримидина, для лечения рака |
| CN1440278A (zh) * | 2000-06-02 | 2003-09-03 | 希龙公司 | 2′－脱氧－2′－(氟亚甲基)胞嘧啶核苷的药物组合物 |
-
2006
- 2006-04-12 GB GB0720886A patent/GB2442615A/en active Pending
- 2006-04-12 ES ES200750061A patent/ES2327195B1/es not_active Withdrawn - After Issue
- 2006-04-12 CA CA002604192A patent/CA2604192A1/fr not_active Abandoned
- 2006-04-12 WO PCT/US2006/013629 patent/WO2006110800A1/fr active IP Right Grant
- 2006-04-12 EP EP06749864A patent/EP1874271A4/fr not_active Withdrawn
- 2006-04-12 JP JP2008506628A patent/JP2008535920A/ja active Pending
- 2006-04-12 DE DE112006000873T patent/DE112006000873T5/de not_active Withdrawn
Also Published As
| Publication number | Publication date |
|---|---|
| DE112006000873T5 (de) | 2008-03-06 |
| ES2327195A1 (es) | 2009-10-26 |
| JP2008535920A (ja) | 2008-09-04 |
| GB0720886D0 (en) | 2007-12-05 |
| CA2604192A1 (fr) | 2006-10-19 |
| WO2006110800A1 (fr) | 2006-10-19 |
| GB2442615A (en) | 2008-04-09 |
| EP1874271A1 (fr) | 2008-01-09 |
| EP1874271A4 (fr) | 2012-01-25 |
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