ES2190938T3 - Fenilpirazoles con actividad herbicida. - Google Patents

Fenilpirazoles con actividad herbicida.

Info

Publication number
ES2190938T3
ES2190938T3 ES00202688T ES00202688T ES2190938T3 ES 2190938 T3 ES2190938 T3 ES 2190938T3 ES 00202688 T ES00202688 T ES 00202688T ES 00202688 T ES00202688 T ES 00202688T ES 2190938 T3 ES2190938 T3 ES 2190938T3
Authority
ES
Spain
Prior art keywords
group
atom
alkyl
groups
thiadiazol
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Lifetime
Application number
ES00202688T
Other languages
English (en)
Inventor
Porta Piero La
Franco Bettarini
Giovanni Meazza
Gregorio Valea
Ernesto Signorini
Domenico Portoso
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Isagro Ricerca SRL
Original Assignee
Isagro Ricerca SRL
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Isagro Ricerca SRL filed Critical Isagro Ricerca SRL
Application granted granted Critical
Publication of ES2190938T3 publication Critical patent/ES2190938T3/es
Anticipated expiration legal-status Critical
Expired - Lifetime legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
    • C07D403/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/48—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with two nitrogen atoms as the only ring hetero atoms
    • A01N43/56—1,2-Diazoles; Hydrogenated 1,2-diazoles
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/72—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with nitrogen atoms and oxygen or sulfur atoms as ring hetero atoms
    • A01N43/74—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with nitrogen atoms and oxygen or sulfur atoms as ring hetero atoms five-membered rings with one nitrogen atom and either one oxygen atom or one sulfur atom in positions 1,3
    • A01N43/78—1,3-Thiazoles; Hydrogenated 1,3-thiazoles
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/72—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with nitrogen atoms and oxygen or sulfur atoms as ring hetero atoms
    • A01N43/80—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with nitrogen atoms and oxygen or sulfur atoms as ring hetero atoms five-membered rings with one nitrogen atom and either one oxygen atom or one sulfur atom in positions 1,2
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/72—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with nitrogen atoms and oxygen or sulfur atoms as ring hetero atoms
    • A01N43/82—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with nitrogen atoms and oxygen or sulfur atoms as ring hetero atoms five-membered rings with three ring hetero atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/14—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D231/18—One oxygen or sulfur atom
    • C07D231/20—One oxygen atom attached in position 3 or 5
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
    • C07D409/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
    • C07D409/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
    • C07D413/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Plant Pathology (AREA)
  • Engineering & Computer Science (AREA)
  • Dentistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Wood Science & Technology (AREA)
  • Zoology (AREA)
  • Environmental Sciences (AREA)
  • Pest Control & Pesticides (AREA)
  • Agronomy & Crop Science (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)

Abstract

Fenilpirazoles de fórmula general (I): **(Fórmula)** en la que: - R1 y R2, iguales o diferentes, representan un grupo alquil C1-C4 o haloalquil C1-C4; - X representa un átomo de halógeno; - X1 representa un átomo de hidrógeno, un átomo de cloro o un átomo de flúor; - X2 representa un átomo de cloro, un átomo de bromo, un grupo haloalquil C1-C4, un grupo haloalcoxil C1-C4; - Y representa un átomo de oxígeno o un átomo de azufre; - R representa un átomo de hidrógeno o un grupo alquil C1-C4; - n representa 0 ó 1; - E representa uno de los siguientes grupos heterocíclicos: 2-furanil, 3-furanil, 2-tiofenil, 3-tiofenil, 2-pirrolil, 3-pirrolil, 2-imidazolil, 4-imidazolil, 5-imidazolil, 3-pirazolil, 4-pirazolil, 5-pirazolil, 1, 2, 4triazol-3-il, 1, 2, 4-triazol-5-il, 1, 2, 4-triazol-3-on-5-il, 1, 2, 3-triazol-4-il, 1, 2, 3-triazol-5-il, 5-tetrazolil, 2-oxazolil, 4-oxazolil, 5-oxazolil, 3-isooxazolil, 4-isooxazolil, 5-isooxazolil, 2-tiazolil, 4-tiazolil, 5tiazolil, 3-isotiazolil, 4-isotiazolil, 5-isotiazolil, 1, 3 4-oxadiazol-2-il, 1, 3, 4-oxadiazol-2-on-5-il, 1, 3, 4tiadiazol-2-il, 1, 3, 4-tiadiazol-2-on-5-il, 1, 2, 4-oxadiazol-3-il, 1, 2, 4-oxadiazol-5-il, 1, 2, 4-tiadiazol-3-il, 1, 2, 4-tiadiazol-5-il; dichos grupos pueden estar sustituidos por uno o más grupos, iguales o diferentes, seleccionados de entre un átomo de halógeno, un grupo alquil C1-C6 o haloalquil C1-C6, un grupo alcoxil C1-C6 o haloalcoxil C1-C6, un grupo alcoxialquil C2-C6 o haloalcoxialquil C2-C6, un grupo alquiltio C1-C6 o haloalquiltio C1-C6, un grupo alquilsulfínico C1-C6 o haloalquilsulfínico C1-C6, un grupo alquilsulfónico C1-C6 o haloalquilsulfónico C1-C6, un grupo alcoxicarbonilo o haloalcoxicarbonilo, un grupo aminocarbonilo opcionalmente sustituido por uno o dos grupos alquil C1-C4 o por una cadena de alquileno C2-C5, un grupo ciano, un grupo formilo, un grupo alquilcarbonilo o haloalquilcarbonilo, un grupo alcoxiiminoalquil o haloalcoxiiminoalquil, un grupo fenil opcionalmente sustituido, a su vez, por átomos de halógeno, grupos alquil C1-C4 o haloalquil C1-C4, grupos alcoxil C1-C4 o haloalcoxil C1-C4.
ES00202688T 1999-08-05 2000-07-27 Fenilpirazoles con actividad herbicida. Expired - Lifetime ES2190938T3 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
IT1999MI001766A IT1313601B1 (it) 1999-08-05 1999-08-05 Fenilpirazoli ad attivita' erbicida

Publications (1)

Publication Number Publication Date
ES2190938T3 true ES2190938T3 (es) 2003-09-01

Family

ID=11383513

Family Applications (1)

Application Number Title Priority Date Filing Date
ES00202688T Expired - Lifetime ES2190938T3 (es) 1999-08-05 2000-07-27 Fenilpirazoles con actividad herbicida.

Country Status (11)

Country Link
US (1) US6265351B1 (es)
EP (1) EP1074551B1 (es)
JP (1) JP2001106688A (es)
AR (1) AR030028A1 (es)
AT (1) ATE235491T1 (es)
BR (1) BR0003352A (es)
DE (1) DE60001782T2 (es)
DK (1) DK1074551T3 (es)
ES (1) ES2190938T3 (es)
IT (1) IT1313601B1 (es)
PT (1) PT1074551E (es)

Families Citing this family (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP4937471B2 (ja) * 2001-07-13 2012-05-23 株式会社エス・ディー・エス バイオテック 置換ピラゾール誘導体を有効成分とする除草剤および植物生育調節剤
EP1407667B1 (en) * 2001-07-13 2007-09-26 SDS Biotech K.K. Herbicide containing substituted pyrazole derivative as active ingredient
CN101613321A (zh) * 2002-03-05 2009-12-30 特兰斯泰克制药公司 抑制配体与高级糖化终产物受体相互作用的单和双环吡咯衍生物
WO2005000295A1 (en) * 2003-05-20 2005-01-06 Transtech Pharma, Inc. Rage antagonists as agents to reverse amyloidosis and diseases associated therewith
ITMI20070355A1 (it) * 2007-02-23 2008-08-24 Isagro Ricerca Srl Formulazioni ad elevata efficienza e ridotto impatto ambientale
CA2772797C (en) 2009-09-30 2018-09-25 Transtech Pharma, Inc. Substituted imidazole derivatives
CN101870677A (zh) * 2010-06-28 2010-10-27 大连理工大学 一种5-芳甲氧基苯基吡唑类化合物及其制备方法
EP2602248A1 (en) 2011-12-05 2013-06-12 University Of Leicester Novel pyrrole compounds
JP6446464B2 (ja) * 2013-11-01 2018-12-26 エスアールエフ リミテッド ピラゾール誘導体の製造方法
CN103923012A (zh) * 2014-04-29 2014-07-16 南京工业大学 一种4-氯吡唑衍生物的制备方法
IL251949A0 (en) 2017-04-26 2017-07-31 Medical Res Infrastructure & Health Services Fund Tel Aviv Medical Ct Small organic molecules for use in the treatment of neuro-inflammatory diseases

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5064850A (en) * 1991-04-08 1991-11-12 Marion Merrell Dow Inc. Dihydro-3,3-diphenyl-5-(1H-pyrazol-1-ylmethyl-2(3H)-furanone and dihydro-5-((substituted-1H-pyrazol-1-yl)methyl)-3,3-diphenyl-2(3H)-furanone derivatives
DE19622189A1 (de) * 1996-06-03 1997-12-04 Bayer Ag 3-Cyanaryl-pyrazole
DE69820242T2 (de) * 1997-03-14 2004-09-09 Isk Americas Incorporated, Concord Diarylether, verfahren zu ihrer herstellung und herbizide und austrocknende zusammensetzungen, die sie enthalten
DE19803395A1 (de) * 1998-01-29 1999-08-05 Bayer Ag Substituierte Heteroarylmethylverbindungen
US6121201A (en) * 1998-09-11 2000-09-19 Ishihara Sangyo Kaisha, Ltd. Diaryl ethers and processes for their preparation and herbicidal and desiccant compositions containing them

Also Published As

Publication number Publication date
IT1313601B1 (it) 2002-09-09
EP1074551B1 (en) 2003-03-26
EP1074551A2 (en) 2001-02-07
ITMI991766A0 (it) 1999-08-05
DK1074551T3 (da) 2003-07-21
JP2001106688A (ja) 2001-04-17
EP1074551A3 (en) 2001-05-09
ITMI991766A1 (it) 2001-02-05
US6265351B1 (en) 2001-07-24
DE60001782D1 (de) 2003-04-30
BR0003352A (pt) 2001-03-13
AR030028A1 (es) 2003-08-13
PT1074551E (pt) 2003-07-31
DE60001782T2 (de) 2004-02-12
ATE235491T1 (de) 2003-04-15

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