ES2172023T3 - Nuevos derivados tetrahidro-piridinicos sustituidos, su procedimiento de preparacion y las composiciones farmaceuticas que los contienen. - Google Patents
Nuevos derivados tetrahidro-piridinicos sustituidos, su procedimiento de preparacion y las composiciones farmaceuticas que los contienen.Info
- Publication number
- ES2172023T3 ES2172023T3 ES97948974T ES97948974T ES2172023T3 ES 2172023 T3 ES2172023 T3 ES 2172023T3 ES 97948974 T ES97948974 T ES 97948974T ES 97948974 T ES97948974 T ES 97948974T ES 2172023 T3 ES2172023 T3 ES 2172023T3
- Authority
- ES
- Spain
- Prior art keywords
- tetrahydra
- pharmaceutical compositions
- compositions containing
- preparation procedure
- new substituted
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired - Lifetime
Links
- 239000008194 pharmaceutical composition Substances 0.000 title 1
- 239000002253 acid Substances 0.000 abstract 1
- 150000001875 compounds Chemical class 0.000 abstract 1
- 229940079593 drug Drugs 0.000 abstract 1
- 239000003814 drug Substances 0.000 abstract 1
- 230000003287 optical effect Effects 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D211/00—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
- C07D211/04—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D211/68—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having one double bond between ring members or between a ring member and a non-ring member
- C07D211/70—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having one double bond between ring members or between a ring member and a non-ring member with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
- A61P25/16—Anti-Parkinson drugs
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
Abstract
LA INVENCION SE REFIERE A LOS COMPUESTOS DE FORMULA GENERAL (I) EN LA QUE R, R 1 , R 2 , X E Y SON TALES COMO SE DEFINEN EN LA DESCRIPCION, SUS ISOMEROS GEOMETRICOS Y/O OPTICOS Y SUS SALES DE ADICION A UN ACIDO O UNA BASE FARMACEUTICAMENTE ACEPTABLES. APLICACION: MEDICAMENTOS.
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
FR9614951A FR2756826B1 (fr) | 1996-12-05 | 1996-12-05 | Nouveaux derives tetrahydropyridiniques substitues, leur procede de preparation et les compositions pharmaceutiques qui les contiennent |
Publications (1)
Publication Number | Publication Date |
---|---|
ES2172023T3 true ES2172023T3 (es) | 2002-09-16 |
Family
ID=9498371
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
ES97948974T Expired - Lifetime ES2172023T3 (es) | 1996-12-05 | 1997-12-02 | Nuevos derivados tetrahidro-piridinicos sustituidos, su procedimiento de preparacion y las composiciones farmaceuticas que los contienen. |
Country Status (19)
Country | Link |
---|---|
US (1) | US6232319B1 (es) |
EP (1) | EP0937043B1 (es) |
JP (1) | JP3872821B2 (es) |
CN (1) | CN1126739C (es) |
AT (1) | ATE214051T1 (es) |
AU (1) | AU719208B2 (es) |
CA (1) | CA2274133C (es) |
DE (1) | DE69710909T2 (es) |
DK (1) | DK0937043T3 (es) |
ES (1) | ES2172023T3 (es) |
FR (1) | FR2756826B1 (es) |
HK (1) | HK1023346A1 (es) |
HU (1) | HUP0001773A3 (es) |
NO (1) | NO313589B1 (es) |
NZ (1) | NZ336111A (es) |
PL (1) | PL189372B1 (es) |
PT (1) | PT937043E (es) |
WO (1) | WO1998024765A1 (es) |
ZA (1) | ZA9710960B (es) |
Families Citing this family (10)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
FR2793245B1 (fr) * | 1999-05-05 | 2002-10-11 | Adir | Nouveaux composes pyridiniques ou piperidiniques substitues, leur procede de preparation et les compositions pharmaceutiques qui les contiennent |
DE10164139A1 (de) | 2001-12-27 | 2003-07-10 | Bayer Ag | 2-Heteroarylcarbonsäureamide |
CN1735414A (zh) * | 2002-12-06 | 2006-02-15 | 北岸长岛犹太人研究学院 | 用α7受体结合类胆碱激动剂抑制炎症 |
US7238715B2 (en) * | 2002-12-06 | 2007-07-03 | The Feinstein Institute For Medical Research | Treatment of pancreatitis using alpha 7 receptor-binding cholinergic agonists |
US8316104B2 (en) | 2005-11-15 | 2012-11-20 | California Institute Of Technology | Method and apparatus for collaborative system |
HUE037938T2 (hu) | 2008-11-19 | 2018-09-28 | Forum Pharmaceuticals Inc | Skizofrénia negatív tüneteinek kezelése (R)-7-klór-N-(kinuklidin-3-il)benzo[b]tiofén-2-karboxamiddal és ennek gyógyszerészetileg elfogadható sójával |
TW201031664A (en) | 2009-01-26 | 2010-09-01 | Targacept Inc | Preparation and therapeutic applications of (2S,3R)-N-2-((3-pyridinyl)methyl)-1-azabicyclo[2.2.2]oct-3-yl)-3,5-difluorobenzamide |
RU2011150248A (ru) * | 2009-05-11 | 2013-06-20 | Энвиво Фармасьютикалз, Инк. | Лечение когнитивных расстройств с определенными рецепторами альфа-7 никотиновой кислоты в комбинации с ингибиторами ацетилхолинэстеразы |
PT3029039T (pt) | 2010-05-17 | 2017-11-28 | Forum Pharmaceuticals Inc | Formulações farmacêuticas que compreendem formas cristalinas de cloridrato de (r)-7-cloro-n-(quinuclidin-3-il)benzo(b)tiofeno-2-carboxamida mono-hidratado |
CA2872005A1 (en) | 2012-05-08 | 2013-11-14 | Forum Pharmaceuticals, Inc. | Methods of maintaining, treating or improving cognitive function |
-
1996
- 1996-12-05 FR FR9614951A patent/FR2756826B1/fr not_active Expired - Fee Related
-
1997
- 1997-12-02 CA CA002274133A patent/CA2274133C/fr not_active Expired - Fee Related
- 1997-12-02 JP JP52527098A patent/JP3872821B2/ja not_active Expired - Fee Related
- 1997-12-02 PT PT97948974T patent/PT937043E/pt unknown
- 1997-12-02 WO PCT/FR1997/002172 patent/WO1998024765A1/fr active IP Right Grant
- 1997-12-02 ES ES97948974T patent/ES2172023T3/es not_active Expired - Lifetime
- 1997-12-02 DE DE69710909T patent/DE69710909T2/de not_active Expired - Fee Related
- 1997-12-02 US US09/319,341 patent/US6232319B1/en not_active Expired - Fee Related
- 1997-12-02 EP EP97948974A patent/EP0937043B1/fr not_active Expired - Lifetime
- 1997-12-02 AU AU76243/98A patent/AU719208B2/en not_active Ceased
- 1997-12-02 PL PL97333813A patent/PL189372B1/pl not_active IP Right Cessation
- 1997-12-02 DK DK97948974T patent/DK0937043T3/da active
- 1997-12-02 NZ NZ336111A patent/NZ336111A/xx unknown
- 1997-12-02 HU HU0001773A patent/HUP0001773A3/hu unknown
- 1997-12-02 AT AT97948974T patent/ATE214051T1/de not_active IP Right Cessation
- 1997-12-02 CN CN97180312A patent/CN1126739C/zh not_active Expired - Fee Related
- 1997-12-05 ZA ZA9710960A patent/ZA9710960B/xx unknown
-
1999
- 1999-06-04 NO NO19992731A patent/NO313589B1/no unknown
-
2000
- 2000-05-02 HK HK00102632A patent/HK1023346A1/xx not_active IP Right Cessation
Also Published As
Publication number | Publication date |
---|---|
EP0937043B1 (fr) | 2002-03-06 |
US6232319B1 (en) | 2001-05-15 |
EP0937043A1 (fr) | 1999-08-25 |
HUP0001773A3 (en) | 2002-12-28 |
CA2274133A1 (fr) | 1998-06-11 |
FR2756826B1 (fr) | 1999-01-08 |
HUP0001773A2 (hu) | 2000-11-28 |
JP3872821B2 (ja) | 2007-01-24 |
CN1239951A (zh) | 1999-12-29 |
AU7624398A (en) | 1998-06-29 |
CN1126739C (zh) | 2003-11-05 |
PL189372B1 (pl) | 2005-07-29 |
NZ336111A (en) | 2000-03-27 |
ZA9710960B (en) | 1998-06-15 |
ATE214051T1 (de) | 2002-03-15 |
FR2756826A1 (fr) | 1998-06-12 |
DK0937043T3 (da) | 2002-06-10 |
JP2001505214A (ja) | 2001-04-17 |
DE69710909D1 (de) | 2002-04-11 |
CA2274133C (fr) | 2003-09-16 |
HK1023346A1 (en) | 2000-09-08 |
AU719208B2 (en) | 2000-05-04 |
NO992731L (no) | 1999-06-04 |
WO1998024765A1 (fr) | 1998-06-11 |
NO313589B1 (no) | 2002-10-28 |
DE69710909T2 (de) | 2002-11-07 |
PT937043E (pt) | 2002-07-31 |
NO992731D0 (no) | 1999-06-04 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
FG2A | Definitive protection |
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