ES2158093T3 - Compuesto del 9-desoxotaxano. - Google Patents

Compuesto del 9-desoxotaxano.

Info

Publication number
ES2158093T3
ES2158093T3 ES95912007T ES95912007T ES2158093T3 ES 2158093 T3 ES2158093 T3 ES 2158093T3 ES 95912007 T ES95912007 T ES 95912007T ES 95912007 T ES95912007 T ES 95912007T ES 2158093 T3 ES2158093 T3 ES 2158093T3
Authority
ES
Spain
Prior art keywords
deoxotaxan
composite
compounds
taxol
oxygenated
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Lifetime
Application number
ES95912007T
Other languages
English (en)
Inventor
Larry L Klein
Clinton M Yeung
Leping Li
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Abbott Laboratories
Original Assignee
Abbott Laboratories
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Abbott Laboratories filed Critical Abbott Laboratories
Application granted granted Critical
Publication of ES2158093T3 publication Critical patent/ES2158093T3/es
Anticipated expiration legal-status Critical
Expired - Lifetime legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D493/00—Heterocyclic compounds containing oxygen atoms as the only ring hetero atoms in the condensed system
    • C07D493/02—Heterocyclic compounds containing oxygen atoms as the only ring hetero atoms in the condensed system in which the condensed system contains two hetero rings
    • C07D493/06—Peri-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/335—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D305/00—Heterocyclic compounds containing four-membered rings having one oxygen atom as the only ring hetero atoms
    • C07D305/14—Heterocyclic compounds containing four-membered rings having one oxygen atom as the only ring hetero atoms condensed with carbocyclic rings or ring systems

Abstract

COMPUESTOS QUE TIENEN LA FORMULA (I), EN DONDE -OR 1 COMPRENDE ALCANOILO O LA CADENA LATERAL C-13 DE PACLITAXEL; R{SUP,2}, R{SUP,3} Y R{SUP,6} PUEDEN SER OXIGENADOS O HIDROGENO EN VARIAS COMBINACIONES; Y R{SUP,4} Y R{SUP,5} SON GRUPOS ACILO, ASI COMO UN PROCESO PARA LA PREPARACION DE LOS MISMOS, COMPOSICIONES FARMACEUTICAS QUE CONTIENEN LOS ANTERIORES COMPUESTOS, Y UN METODO PARA SU USO EN EL INHIBICION DEL CRECIMIENTO TUMORAL.
ES95912007T 1994-03-09 1995-03-01 Compuesto del 9-desoxotaxano. Expired - Lifetime ES2158093T3 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US08/208,509 US5440056A (en) 1992-04-17 1994-03-09 9-deoxotaxane compounds

Publications (1)

Publication Number Publication Date
ES2158093T3 true ES2158093T3 (es) 2001-09-01

Family

ID=22774850

Family Applications (1)

Application Number Title Priority Date Filing Date
ES95912007T Expired - Lifetime ES2158093T3 (es) 1994-03-09 1995-03-01 Compuesto del 9-desoxotaxano.

Country Status (15)

Country Link
US (2) US5440056A (es)
EP (1) EP0749432B1 (es)
JP (1) JPH09511235A (es)
KR (1) KR970701708A (es)
AT (1) ATE201019T1 (es)
AU (1) AU688946B2 (es)
CA (1) CA2182103A1 (es)
DE (1) DE69520880T2 (es)
DK (1) DK0749432T3 (es)
ES (1) ES2158093T3 (es)
GR (1) GR3036286T3 (es)
IL (1) IL112880A0 (es)
PH (1) PH31271A (es)
PT (1) PT749432E (es)
WO (1) WO1995024402A1 (es)

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US20030054036A1 (en) * 2001-03-13 2003-03-20 Richard Liggins Micellar drug delivery vehicles and precursors thereto and uses thereof
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US20040191218A1 (en) * 2001-09-26 2004-09-30 Emlen James W Pharmaceutical compositions and methods for treating cancer
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US20050187288A1 (en) * 2004-02-20 2005-08-25 Chiang Li Beta-lapachone and methods of treating cancer
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Also Published As

Publication number Publication date
WO1995024402A1 (en) 1995-09-14
DK0749432T3 (da) 2001-07-30
PH31271A (en) 1998-06-18
CA2182103A1 (en) 1995-09-14
EP0749432B1 (en) 2001-05-09
MX9603891A (es) 1997-07-31
US5440056A (en) 1995-08-08
DE69520880T2 (de) 2001-12-20
DE69520880D1 (de) 2001-06-13
ATE201019T1 (de) 2001-05-15
JPH09511235A (ja) 1997-11-11
PT749432E (pt) 2001-09-28
AU688946B2 (en) 1998-03-19
KR970701708A (ko) 1997-04-12
AU3104795A (en) 1995-09-25
GR3036286T3 (en) 2001-10-31
US5616740A (en) 1997-04-01
IL112880A0 (en) 1995-06-29
EP0749432A1 (en) 1996-12-27

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