ES2109966T3 - Un metodo y productos intermedios para la preparacion de 6-fluorobenzisotiazoles. - Google Patents

Un metodo y productos intermedios para la preparacion de 6-fluorobenzisotiazoles.

Info

Publication number
ES2109966T3
ES2109966T3 ES92114142T ES92114142T ES2109966T3 ES 2109966 T3 ES2109966 T3 ES 2109966T3 ES 92114142 T ES92114142 T ES 92114142T ES 92114142 T ES92114142 T ES 92114142T ES 2109966 T3 ES2109966 T3 ES 2109966T3
Authority
ES
Spain
Prior art keywords
chem
preparation
formula
compound
fluorobenzisotiazoles
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Lifetime
Application number
ES92114142T
Other languages
English (en)
Inventor
David M Fink
Joseph T Strupczewski
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Aventis Pharmaceuticals Inc
Original Assignee
Hoechst Marion Roussel Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Hoechst Marion Roussel Inc filed Critical Hoechst Marion Roussel Inc
Application granted granted Critical
Publication of ES2109966T3 publication Critical patent/ES2109966T3/es
Anticipated expiration legal-status Critical
Expired - Lifetime legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D275/00—Heterocyclic compounds containing 1,2-thiazole or hydrogenated 1,2-thiazole rings
    • C07D275/04—Heterocyclic compounds containing 1,2-thiazole or hydrogenated 1,2-thiazole rings condensed with carbocyclic rings or ring systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C323/00—Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups
    • C07C323/22—Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups containing thio groups and doubly-bound oxygen atoms bound to the same carbon skeleton
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D211/00—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
    • C07D211/04—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D211/06—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
    • C07D211/08—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms
    • C07D211/18—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms with substituted hydrocarbon radicals attached to ring carbon atoms
    • C07D211/30—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms with substituted hydrocarbon radicals attached to ring carbon atoms with hydrocarbon radicals, substituted by doubly bound oxygen or sulfur atoms or by two oxygen or sulfur atoms singly bound to the same carbon atom
    • C07D211/32—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms with substituted hydrocarbon radicals attached to ring carbon atoms with hydrocarbon radicals, substituted by doubly bound oxygen or sulfur atoms or by two oxygen or sulfur atoms singly bound to the same carbon atom by oxygen atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D451/00—Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof
    • C07D451/02—Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof containing not further condensed 8-azabicyclo [3.2.1] octane or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane; Cyclic acetals thereof

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Thiazole And Isothizaole Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Lubricants (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Production Of Liquid Hydrocarbon Mixture For Refining Petroleum (AREA)
  • Detergent Compositions (AREA)
  • Plural Heterocyclic Compounds (AREA)

Abstract

SE PRESENTA UN PROCESO PARA LA PREPARACION DE 6-FLUORO-1,2-BENZISOTIAZOLAS DE LA FORMULA (I) EN DONDE R ES HIDROGENO, ALQUIL INFERIOR, CICLOALQUIL, ARALQUIL, ARIL O UN GRUPO DE LAS FORMULAS: EN DONDE R1 ES -CHO, -CO2R2, -CN O -C(=O)R2; R2 ES ALQUIL O ARIL; K, M, M*, N Y N* SON INDEPENDIENTEMENTE ENTEROS ENTRE 1 Y 4; EL PROCESO COMPRENDE: A) LA REACCION DE UN COMPUESTO DE LA FORMULA (III): EN DONDE R ES SEGUN SE HA DEFINIDO ANTERIORMENTE Y R3 ES HIDROGENO, ALQUIL INFERIOR, O ALQUIL INFERIOR DE ARIL, CON UN AGENTE HALOGENANTE PARA OBTENER UN COMPUESTO DE LA FORMULA (IV): EN LA QUE R ES SEGUN SE HA DEFINIDO Y HAL ES HALOGENO, Y B) LA REACCION DEL COMPUESTO DE LA FORMULA IV SEGUN SE HA OBTENIDO EN EL PASO A) CON AMONIO.
ES92114142T 1991-08-22 1992-08-19 Un metodo y productos intermedios para la preparacion de 6-fluorobenzisotiazoles. Expired - Lifetime ES2109966T3 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US74872991A 1991-08-22 1991-08-22

Publications (1)

Publication Number Publication Date
ES2109966T3 true ES2109966T3 (es) 1998-02-01

Family

ID=25010669

Family Applications (1)

Application Number Title Priority Date Filing Date
ES92114142T Expired - Lifetime ES2109966T3 (es) 1991-08-22 1992-08-19 Un metodo y productos intermedios para la preparacion de 6-fluorobenzisotiazoles.

Country Status (19)

Country Link
EP (1) EP0536512B1 (es)
JP (1) JP2778366B2 (es)
KR (1) KR100212584B1 (es)
AT (1) ATE159939T1 (es)
AU (1) AU652847B2 (es)
CA (1) CA2076556A1 (es)
CZ (1) CZ258392A3 (es)
DE (1) DE69223016T2 (es)
DK (1) DK0536512T3 (es)
ES (1) ES2109966T3 (es)
FI (1) FI923744A (es)
GR (1) GR3025608T3 (es)
HU (1) HU219481B (es)
IL (1) IL102884A (es)
MX (1) MX9204872A (es)
NO (1) NO300213B1 (es)
NZ (1) NZ244010A (es)
RU (1) RU2027704C1 (es)
TW (1) TW241263B (es)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5169951A (en) * 1990-04-23 1992-12-08 Ciba-Geigy Corporation Process for preparing nematicidal compositions
JP3701044B2 (ja) * 1995-04-24 2005-09-28 住友精化株式会社 シアノベンゼンスルフェニルハライドおよびそれを用いる３−置換ベンゾイソチアゾールの製造方法
GB9603127D0 (en) * 1996-02-15 1996-04-17 Rhone Poulenc Agriculture New process for preparing intermediates

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE69021645T2 (de) * 1989-05-19 1996-02-22 Hoechst Roussel Pharma N-(aryloxyalkyl)heteroarylpiperidine und -heteroarylpiperazine, Verfahren zu ihrer Herstellung und ihre Verwendung als Medikamente.
US5169951A (en) * 1990-04-23 1992-12-08 Ciba-Geigy Corporation Process for preparing nematicidal compositions

Also Published As

Publication number Publication date
ATE159939T1 (de) 1997-11-15
AU652847B2 (en) 1994-09-08
DE69223016T2 (de) 1998-06-04
TW241263B (es) 1995-02-21
EP0536512B1 (en) 1997-11-05
HU219481B (hu) 2001-04-28
HUT71552A (en) 1995-12-28
CA2076556A1 (en) 1993-02-23
NZ244010A (en) 1995-02-24
FI923744A0 (fi) 1992-08-20
RU2027704C1 (ru) 1995-01-27
HU9202666D0 (en) 1992-10-28
KR930004284A (ko) 1993-03-22
GR3025608T3 (en) 1998-03-31
MX9204872A (es) 1993-04-01
DK0536512T3 (da) 1998-07-27
JP2778366B2 (ja) 1998-07-23
NO923287L (no) 1993-02-23
CZ258392A3 (en) 1993-03-17
KR100212584B1 (ko) 1999-08-02
NO923287D0 (no) 1992-08-21
EP0536512A1 (en) 1993-04-14
IL102884A0 (en) 1993-01-31
DE69223016D1 (de) 1997-12-11
JPH05194443A (ja) 1993-08-03
IL102884A (en) 1998-02-22
FI923744A (fi) 1993-02-23
NO300213B1 (no) 1997-04-28
AU2124892A (en) 1993-02-25

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