ES2077376T3 - Derivados de 2-aminopirimidina-4-carboxamida, su preparacion y su aplicacion terapeutica. - Google Patents
Derivados de 2-aminopirimidina-4-carboxamida, su preparacion y su aplicacion terapeutica.Info
- Publication number
- ES2077376T3 ES2077376T3 ES92401771T ES92401771T ES2077376T3 ES 2077376 T3 ES2077376 T3 ES 2077376T3 ES 92401771 T ES92401771 T ES 92401771T ES 92401771 T ES92401771 T ES 92401771T ES 2077376 T3 ES2077376 T3 ES 2077376T3
- Authority
- ES
- Spain
- Prior art keywords
- aminopyrimidine
- carboxamide
- derivatives
- preparation
- therapeutic application
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired - Lifetime
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
- C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
- C07D403/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P13/00—Drugs for disorders of the urinary system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P13/00—Drugs for disorders of the urinary system
- A61P13/02—Drugs for disorders of the urinary system of urine or of the urinary tract, e.g. urine acidifiers
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P13/00—Drugs for disorders of the urinary system
- A61P13/08—Drugs for disorders of the urinary system of the prostate
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Public Health (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Engineering & Computer Science (AREA)
- General Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Urology & Nephrology (AREA)
- Endocrinology (AREA)
- Reproductive Health (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Cephalosporin Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Hydrogenated Pyridines (AREA)
- Steroid Compounds (AREA)
Abstract
COMPUESTO, EN FORMA DE ENANTIOMERO PURO O DE MEZCLA DE ENANTIOMEROS, QUE RESPONDE A LA FORMULA GENERAL (I) EN LA QUE X REPRESENTA UNO O VARIOS SUSTITUYENTES ELEGIDOS ENTRE LOS ATOMOS DE HIDROGENO, DE FLUOR Y DE CLORO Y LOS GRUPO METILO, 1-METILETILO Y METOXI, N REPRESENTA EL NUMERO 2 O 3, M REPRESENTA EL NUMERO 1, EN CUYO CASO P REPRESENTA EL NUMERO 1, O BIEN M REPRESENTA EL NUMERO 0, EN CUYO CASO P REPRESENTA EL NUMERO 2, Q REPRESENTA EL NUMERO 0 O 1, Y R1 REPRESENTA UN ATOMO DE HIDROGENO. APLICACION EN TERAPIA.
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
FR9107938A FR2678268B1 (fr) | 1991-06-27 | 1991-06-27 | Derives de 2-aminopyrimidine-4-carboxamide, leur preparation et leur application en therapeutique. |
FR9206005A FR2691148B1 (fr) | 1992-05-18 | 1992-05-18 | Derives de 2-aminopyrimidine-4-carboxamide, leur preparation et leur application en therapeutique. |
Publications (1)
Publication Number | Publication Date |
---|---|
ES2077376T3 true ES2077376T3 (es) | 1995-11-16 |
Family
ID=26228783
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
ES92401771T Expired - Lifetime ES2077376T3 (es) | 1991-06-27 | 1992-06-24 | Derivados de 2-aminopirimidina-4-carboxamida, su preparacion y su aplicacion terapeutica. |
Country Status (20)
Country | Link |
---|---|
US (1) | US5246939A (es) |
EP (1) | EP0520882B1 (es) |
JP (1) | JP3159525B2 (es) |
KR (1) | KR930000507A (es) |
CN (1) | CN1067887A (es) |
AT (1) | ATE124942T1 (es) |
AU (1) | AU645429B2 (es) |
CA (1) | CA2072434A1 (es) |
CZ (1) | CZ9202001A3 (es) |
DE (1) | DE69203401T2 (es) |
DK (1) | DK0520882T3 (es) |
ES (1) | ES2077376T3 (es) |
FI (1) | FI922981A (es) |
GR (1) | GR3017612T3 (es) |
HU (1) | HUT61745A (es) |
IE (1) | IE922092A1 (es) |
IL (1) | IL102329A0 (es) |
MX (1) | MX9203332A (es) |
NO (1) | NO922523L (es) |
PL (1) | PL295046A1 (es) |
Families Citing this family (4)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
GB9319534D0 (en) * | 1993-09-22 | 1993-11-10 | Boots Co Plc | Therapeutic agents |
AU3883099A (en) * | 1998-05-06 | 1999-11-23 | Duke University | Method of treating bladder and lower urinary tract syndromes |
RU2018145734A (ru) | 2016-06-08 | 2020-07-14 | Глэксосмитклайн Интеллекчуал Проперти Дивелопмент Лимитед | Химические соединения в качестве ингибиторов atf4 пути |
KR102177766B1 (ko) * | 2019-03-15 | 2020-11-11 | 주식회사 엠에스바이오 | 양막링 및 이의 제조방법 |
Family Cites Families (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
FR2618436B1 (fr) * | 1987-07-23 | 1989-10-27 | Synthelabo | Derives de piperidine, leur preparation et leur application en therapeutique |
HU206337B (en) * | 1988-12-29 | 1992-10-28 | Mitsui Petrochemical Ind | Process for producing pyrimidine derivatives and pharmaceutical compositions |
FR2667317B1 (fr) * | 1990-10-02 | 1992-12-04 | Synthelabo | Derives de 2-aminopyrimidine-4-carboxamide, leur preparation et leur application en therapeutique. |
-
1992
- 1992-06-24 DE DE69203401T patent/DE69203401T2/de not_active Expired - Fee Related
- 1992-06-24 EP EP92401771A patent/EP0520882B1/fr not_active Expired - Lifetime
- 1992-06-24 AT AT92401771T patent/ATE124942T1/de not_active IP Right Cessation
- 1992-06-24 DK DK92401771.8T patent/DK0520882T3/da active
- 1992-06-24 ES ES92401771T patent/ES2077376T3/es not_active Expired - Lifetime
- 1992-06-25 MX MX9203332A patent/MX9203332A/es unknown
- 1992-06-26 FI FI922981A patent/FI922981A/fi unknown
- 1992-06-26 KR KR1019920011215A patent/KR930000507A/ko not_active Application Discontinuation
- 1992-06-26 US US07/903,977 patent/US5246939A/en not_active Expired - Fee Related
- 1992-06-26 JP JP16899192A patent/JP3159525B2/ja not_active Expired - Fee Related
- 1992-06-26 NO NO92922523A patent/NO922523L/no unknown
- 1992-06-26 HU HU9202142A patent/HUT61745A/hu unknown
- 1992-06-26 AU AU18587/92A patent/AU645429B2/en not_active Ceased
- 1992-06-26 IL IL102329A patent/IL102329A0/xx unknown
- 1992-06-26 PL PL29504692A patent/PL295046A1/xx unknown
- 1992-06-26 CZ CS922001A patent/CZ9202001A3/cs unknown
- 1992-06-26 CN CN92105077A patent/CN1067887A/zh active Pending
- 1992-06-26 CA CA002072434A patent/CA2072434A1/en not_active Abandoned
- 1992-07-01 IE IE209292A patent/IE922092A1/en not_active Application Discontinuation
-
1995
- 1995-10-04 GR GR950402725T patent/GR3017612T3/el unknown
Also Published As
Publication number | Publication date |
---|---|
EP0520882B1 (fr) | 1995-07-12 |
HU9202142D0 (en) | 1992-10-28 |
MX9203332A (es) | 1992-12-01 |
US5246939A (en) | 1993-09-21 |
AU1858792A (en) | 1993-01-07 |
NO922523L (no) | 1992-12-28 |
DE69203401D1 (de) | 1995-08-17 |
AU645429B2 (en) | 1994-01-13 |
DK0520882T3 (da) | 1995-12-11 |
GR3017612T3 (en) | 1996-01-31 |
NO922523D0 (no) | 1992-06-26 |
ATE124942T1 (de) | 1995-07-15 |
HUT61745A (en) | 1993-03-01 |
DE69203401T2 (de) | 1996-03-07 |
IL102329A0 (en) | 1993-01-14 |
KR930000507A (ko) | 1993-01-15 |
CN1067887A (zh) | 1993-01-13 |
FI922981A0 (fi) | 1992-06-26 |
FI922981A (fi) | 1992-12-28 |
PL295046A1 (en) | 1993-03-22 |
JPH05194419A (ja) | 1993-08-03 |
CA2072434A1 (en) | 1993-01-28 |
IE922092A1 (en) | 1992-12-30 |
CZ9202001A3 (en) | 1993-01-13 |
EP0520882A1 (fr) | 1992-12-30 |
JP3159525B2 (ja) | 2001-04-23 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
FG2A | Definitive protection |
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