FR2678268B1 - Derives de 2-aminopyrimidine-4-carboxamide, leur preparation et leur application en therapeutique. - Google Patents

Derives de 2-aminopyrimidine-4-carboxamide, leur preparation et leur application en therapeutique.

Info

Publication number
FR2678268B1
FR2678268B1 FR9107938A FR9107938A FR2678268B1 FR 2678268 B1 FR2678268 B1 FR 2678268B1 FR 9107938 A FR9107938 A FR 9107938A FR 9107938 A FR9107938 A FR 9107938A FR 2678268 B1 FR2678268 B1 FR 2678268B1
Authority
FR
France
Prior art keywords
aminopyrimidine
preparation
therapeutic application
carboxamide derivatives
carboxamide
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Fee Related
Application number
FR9107938A
Other languages
English (en)
Other versions
FR2678268A1 (fr
Inventor
George Pascal
Maloizel Christian
Marabout Benoit
Merly Jean-Pierre
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Synthelabo SA
Original Assignee
Synthelabo SA
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Synthelabo SA filed Critical Synthelabo SA
Priority to FR9107938A priority Critical patent/FR2678268B1/fr
Priority to AT92401771T priority patent/ATE124942T1/de
Priority to ES92401771T priority patent/ES2077376T3/es
Priority to DK92401771.8T priority patent/DK0520882T3/da
Priority to EP92401770A priority patent/EP0522914A1/fr
Priority to DE69203401T priority patent/DE69203401T2/de
Priority to EP92401771A priority patent/EP0520882B1/fr
Priority to MX9203332A priority patent/MX9203332A/es
Priority to CA002072434A priority patent/CA2072434A1/fr
Priority to MX9203453A priority patent/MX9203453A/es
Priority to AU18586/92A priority patent/AU645697B2/en
Priority to ZA924784A priority patent/ZA924784B/xx
Priority to JP4168982A priority patent/JPH07173152A/ja
Priority to HU9202142A priority patent/HUT61745A/hu
Priority to NO92922522A priority patent/NO922522L/no
Priority to KR1019920011215A priority patent/KR930000507A/ko
Priority to CN92105087A priority patent/CN1067888A/zh
Priority to AU18587/92A priority patent/AU645429B2/en
Priority to PL29504692A priority patent/PL295046A1/xx
Priority to CS922001A priority patent/CZ9202001A3/cs
Priority to HU9202141A priority patent/HUT61740A/hu
Priority to ZA924783A priority patent/ZA924783B/xx
Priority to CA002072529A priority patent/CA2072529A1/fr
Priority to CN92105077A priority patent/CN1067887A/zh
Priority to KR1019920011214A priority patent/KR930000504A/ko
Priority to NO92922523A priority patent/NO922523L/no
Priority to CS922000A priority patent/CZ9202000A3/cs
Priority to JP16899192A priority patent/JP3159525B2/ja
Priority to FI922980A priority patent/FI922980A/fi
Priority to IL102329A priority patent/IL102329A0/xx
Priority to US07/904,061 priority patent/US5254560A/en
Priority to FI922981A priority patent/FI922981A/fi
Priority to US07/903,977 priority patent/US5246939A/en
Priority to PL29504292A priority patent/PL295042A1/xx
Priority to IE209292A priority patent/IE922092A1/en
Priority to IE209192A priority patent/IE922091A1/en
Publication of FR2678268A1 publication Critical patent/FR2678268A1/fr
Application granted granted Critical
Publication of FR2678268B1 publication Critical patent/FR2678268B1/fr
Priority to GR950402725T priority patent/GR3017612T3/el
Anticipated expiration legal-status Critical
Expired - Fee Related legal-status Critical Current

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/12Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
FR9107938A 1991-06-27 1991-06-27 Derives de 2-aminopyrimidine-4-carboxamide, leur preparation et leur application en therapeutique. Expired - Fee Related FR2678268B1 (fr)

Priority Applications (37)

Application Number Priority Date Filing Date Title
FR9107938A FR2678268B1 (fr) 1991-06-27 1991-06-27 Derives de 2-aminopyrimidine-4-carboxamide, leur preparation et leur application en therapeutique.
AT92401771T ATE124942T1 (de) 1991-06-27 1992-06-24 2-aminopyrimidin-4-carboxamidderivate, deren herstellung und deren verwendung als heilmittel.
ES92401771T ES2077376T3 (es) 1991-06-27 1992-06-24 Derivados de 2-aminopirimidina-4-carboxamida, su preparacion y su aplicacion terapeutica.
DK92401771.8T DK0520882T3 (da) 1991-06-27 1992-06-24 Derivater af 2-aminopyrimidin-4-carboxamid, deres fremstilling og deres terapeutiske anvendelse
EP92401770A EP0522914A1 (fr) 1991-06-27 1992-06-24 Dérivés de 2-pipéridinylpyrimidine-4-carboxamide, leur préparation et leur application en thérapeutique
DE69203401T DE69203401T2 (de) 1991-06-27 1992-06-24 2-Aminopyrimidin-4-Carboxamidderivate, deren Herstellung und deren Verwendung als Heilmittel.
EP92401771A EP0520882B1 (fr) 1991-06-27 1992-06-24 Dérivés de 2-aminopyrimidine-4-carboxamide, leur préparation et leur application en thérapeutique
MX9203332A MX9203332A (es) 1991-06-27 1992-06-25 Derivados de 2-amino pirimidina -4- carboxamida, su preparacion y su aplicacion en terapeutica.
NO92922523A NO922523L (no) 1991-06-27 1992-06-26 Aminopyrimidinkarboksamiddrivater med terapeutisk virkning
AU18586/92A AU645697B2 (en) 1991-06-27 1992-06-26 2-piperidinylpyrimidine-4-carboxamide derivatives, their preparation and their use in therapeutics
ZA924784A ZA924784B (en) 1991-06-27 1992-06-26 2-aminopyrimidine-4-carboxamide derivatives,their preparation and their use in therapeutics
JP4168982A JPH07173152A (ja) 1991-06-27 1992-06-26 2−ピペリジニルピリミジン−4−カルボキサミド誘導体、その製造方法及びその医療上用途
HU9202142A HUT61745A (en) 1991-06-27 1992-06-26 Process for producing 2-amino-pyrimidine-4-carboxamide derivatives and pharmaceutical compositions comprising such compounds as active ingredient
NO92922522A NO922522L (no) 1991-06-27 1992-06-26 Piperidinylpyrimidin-karboksamidderivater med terapeutiskvirkning
KR1019920011215A KR930000507A (ko) 1991-06-27 1992-06-26 2-아미노피리미딘-4-카르복시아미드 유도체 그 제법 및 치료에의 이용
CN92105087A CN1067888A (zh) 1991-06-27 1992-06-26 2-哌啶基嘧啶-4-甲酰胺衍生物及其制法和医疗应用
AU18587/92A AU645429B2 (en) 1991-06-27 1992-06-26 2-Aminopyrimidine-4-carboxamide derivatives, their preparation and their use in therapeutics
PL29504692A PL295046A1 (en) 1991-06-27 1992-06-26 Method of obtaining novel derivatives of 2-aminopyrimidine 4-carboxyamide
CA002072434A CA2072434A1 (fr) 1991-06-27 1992-06-26 2-aminopyrimidine-4-carboxamides, leur obtention et leur emploi dans des produits therapeutiques
HU9202141A HUT61740A (en) 1991-06-27 1992-06-26 Process for producing 2-piperidinyl-pyrimidine-4-carboxamide derivatives and pharmaceutical compositions comprising such compounds as active ingredient
ZA924783A ZA924783B (en) 1991-06-27 1992-06-26 2-piperidinylpyrimidine-4-carboxamide derivatives,their preparation and their use in therapeutics
CA002072529A CA2072529A1 (fr) 1991-06-27 1992-06-26 Derives de 2-piperidinylpyrimidine-4-carboxamide, leur obtention et leurs applications therapeutiques
CN92105077A CN1067887A (zh) 1991-06-27 1992-06-26 2-氨基嘧啶-4-甲酰胺衍生物及其制法和医疗应用
KR1019920011214A KR930000504A (ko) 1991-06-27 1992-06-26 2-피페리디닐 피리미딘-4-카르복시아미드 유도체의 제법 및 치료에의 이용
MX9203453A MX9203453A (es) 1991-06-27 1992-06-26 Derivados de 2- piperidinil pirimidina -4- carboxamida, su preparacion y su aplicacion en terapeutica.
CS922000A CZ9202000A3 (en) 1991-06-27 1992-06-26 2-piperidinylpyrimidine-4-carboxamide derivatives, process of their preparation and pharmaceutical compositions containing said derivatives
JP16899192A JP3159525B2 (ja) 1991-06-27 1992-06-26 2−アミノピリミジン−4−カルボキサミド誘導体、その製造方法及びその医療上用途
FI922980A FI922980A (fi) 1991-06-27 1992-06-26 2-piperidinylpyrimidin-4-karboxamidderivat, framstaellning av dessa ochterapeutisk anvaendning av dessa
IL102329A IL102329A0 (en) 1991-06-27 1992-06-26 2-aminopyrimidine-4-carboxamide derivatives,their preparation and their use in therapeutics
US07/904,061 US5254560A (en) 1991-06-27 1992-06-26 2-piperidinylpyrimidine-4-carboxamide derivatives, and their use in therapeutics
FI922981A FI922981A (fi) 1991-06-27 1992-06-26 2-aminopyrimidin-4-karboxamidderivat, framstaellning av dessa och terapeutisk anvaendning av dessa
US07/903,977 US5246939A (en) 1991-06-27 1992-06-26 2-aminopyrimidine-4-carboxamide derivatives, their preparation and their use in therapeutics
PL29504292A PL295042A1 (en) 1991-06-27 1992-06-26 Method of obtaining novel derivatives of 2-piperidinylpyrimidin-4-carboxyamide
CS922001A CZ9202001A3 (en) 1991-06-27 1992-06-26 2-aminopyrimidine-4-carboxamide derivatives, process of their preparation and pharmaceutical compositions in which said derivatives are comprised
IE209292A IE922092A1 (en) 1991-06-27 1992-07-01 2-aminopyrimidine-4-carboxamide derivatives, their¹preparation and their use in therapeutics
IE209192A IE922091A1 (en) 1991-06-27 1992-07-01 2-piperidinylpyrimidine-4-carboxamide derivatives, their¹preparation and their use in therapeutics
GR950402725T GR3017612T3 (en) 1991-06-27 1995-10-04 2-Aminopyrimidin-4-carboxamide derivatives, their preparation and their application in therapy.

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FR9107938A FR2678268B1 (fr) 1991-06-27 1991-06-27 Derives de 2-aminopyrimidine-4-carboxamide, leur preparation et leur application en therapeutique.

Publications (2)

Publication Number Publication Date
FR2678268A1 FR2678268A1 (fr) 1992-12-31
FR2678268B1 true FR2678268B1 (fr) 1993-09-03

Family

ID=9414358

Family Applications (1)

Application Number Title Priority Date Filing Date
FR9107938A Expired - Fee Related FR2678268B1 (fr) 1991-06-27 1991-06-27 Derives de 2-aminopyrimidine-4-carboxamide, leur preparation et leur application en therapeutique.

Country Status (2)

Country Link
FR (1) FR2678268B1 (fr)
ZA (2) ZA924783B (fr)

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2618436B1 (fr) * 1987-07-23 1989-10-27 Synthelabo Derives de piperidine, leur preparation et leur application en therapeutique

Also Published As

Publication number Publication date
ZA924784B (en) 1993-03-31
FR2678268A1 (fr) 1992-12-31
ZA924783B (en) 1993-03-31

Similar Documents

Publication Publication Date Title
FR2601368B1 (fr) Derives de nitrofuranne, leur preparation et leur application en therapeutique.
FR2667317B1 (fr) Derives de 2-aminopyrimidine-4-carboxamide, leur preparation et leur application en therapeutique.
FR2681325B1 (fr) Derives de l'aminomethyl-4 piperidine, leur preparation et leur application en therapeutique.
FR2756563B1 (fr) Derives de benzoate de 1,4-diazabicyclo[2.2.2]oct-2-yl- methyle, leur preparation et leur application en therapeutique
MA22981A1 (fr) Derives de piperidine, leur preparation et leur application en therapeutique.
FR2675799B1 (fr) Derives de 2-aminopyrimidine-4-carboxamide, leur preparation et leur application en therapeutique.
FR2681319B1 (fr) Derives de 1-(phenoxyalkyl)piperidine, leur preparation et leur application en therapeutique.
FR2672601B1 (fr) Derives de benzo-1,5-thiazepine, leur preparation et leur application en therapeutique.
FR2634207B1 (fr) Derives de ((piperidinyl-4)methyl) benzazepines, leur preparation et leur application en therapeutique
FR2638747B1 (fr) Derives de phenyloxypropanolamines, leur preparation et leur application en therapeutique
FR2737494B1 (fr) Derives de benzenesulfonamide, leur preparation et leur application en therapeutique
FR2674853B1 (fr) Derives de piperidinylguanidine, leur preparation et leur application en therapeutique.
FR2765874B1 (fr) Derives de 6-pyrrolidin-2-ylpyrindines, leur preparation et leur application en therapeutique
FR2724382B1 (fr) Derives de 2-aminopyrimidine-4-carboxamide, leur preparation et leur application en therapeutique
FR2752839B1 (fr) Derives de benzofurane, leur preparation et leur application en therapeutique
FR2668152B1 (fr) Derives n,o spirocycliques de cyclotriphosphazenes, leur preparation et leur application en therapeutique.
FR2666582B1 (fr) Derives de benzimidazole, leur preparation et leur application en therapeutique.
FR2742152B1 (fr) Derives de 5-naphtalen-1-yl-1,3-dioxanes, leur preparation et leur application en therapeutique
FR2672891B1 (fr) Derives de 3-pyrazolones, leur preparation et leur application en therapeutique.
FR2684379B1 (fr) Derives de piperidine, leur preparation et leur application en therapeutique.
FR2663025B1 (fr) Derives de 2-aminomethylpyrrolidine, leur preparation et leur application en therapeutique.
FR2735776B1 (fr) Derives de 2,3-dihydro-1h-indole, leur preparation et leur application en therapeutique
FR2785903B1 (fr) Derives de 1-aminoethylquinoleine, leur preparation et leur application en therapeutique
FR2678268B1 (fr) Derives de 2-aminopyrimidine-4-carboxamide, leur preparation et leur application en therapeutique.
FR2759698B1 (fr) Derives de 1,4-diphenylimidazole-5-acetamide, leur preparation et leur application en therapeutique

Legal Events

Date Code Title Description
ST Notification of lapse