ES2059333T3 - Nuevos derivados de mono- y di-acilos de compuestos ll-f28249. - Google Patents

Nuevos derivados de mono- y di-acilos de compuestos ll-f28249.

Info

Publication number
ES2059333T3
ES2059333T3 ES87112277T ES87112277T ES2059333T3 ES 2059333 T3 ES2059333 T3 ES 2059333T3 ES 87112277 T ES87112277 T ES 87112277T ES 87112277 T ES87112277 T ES 87112277T ES 2059333 T3 ES2059333 T3 ES 2059333T3
Authority
ES
Spain
Prior art keywords
compounds
acyl
acilos
compuestos
mono
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Lifetime
Application number
ES87112277T
Other languages
English (en)
Inventor
Goro Asato
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Wyeth Holdings LLC
Original Assignee
American Cyanamid Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by American Cyanamid Co filed Critical American Cyanamid Co
Application granted granted Critical
Publication of ES2059333T3 publication Critical patent/ES2059333T3/es
Anticipated expiration legal-status Critical
Expired - Lifetime legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D493/00—Heterocyclic compounds containing oxygen atoms as the only ring hetero atoms in the condensed system
    • C07D493/22—Heterocyclic compounds containing oxygen atoms as the only ring hetero atoms in the condensed system in which the condensed system contains four or more hetero rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H19/00—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof
    • C07H19/01—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof sharing oxygen
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/90—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having two or more relevant hetero rings, condensed among themselves or with a common carbocyclic ring system
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N49/00—Biocides, pest repellants or attractants, or plant growth regulators, containing compounds containing the group, wherein m+n>=1, both X together may also mean —Y— or a direct carbon-to-carbon bond, and the carbon atoms marked with an asterisk are not part of any ring system other than that which may be formed by the atoms X, the carbon atoms in square brackets being part of any acyclic or cyclic structure, or the group, wherein A means a carbon atom or Y, n>=0, and not more than one of these carbon atoms being a member of the same ring system, e.g. juvenile insect hormones or mimics thereof
    • A—HUMAN NECESSITIES
    • A23—FOODS OR FOODSTUFFS; TREATMENT THEREOF, NOT COVERED BY OTHER CLASSES
    • A23K—FODDER
    • A23K20/00—Accessory food factors for animal feeding-stuffs
    • A23K20/10—Organic substances
    • A23K20/195—Antibiotics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents

Landscapes

  • Life Sciences & Earth Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • General Health & Medical Sciences (AREA)
  • Zoology (AREA)
  • Wood Science & Technology (AREA)
  • Dentistry (AREA)
  • Plant Pathology (AREA)
  • Pest Control & Pesticides (AREA)
  • Agronomy & Crop Science (AREA)
  • Environmental Sciences (AREA)
  • Polymers & Plastics (AREA)
  • Food Science & Technology (AREA)
  • Molecular Biology (AREA)
  • Veterinary Medicine (AREA)
  • Animal Husbandry (AREA)
  • Insects & Arthropods (AREA)
  • Biochemistry (AREA)
  • Biotechnology (AREA)
  • Genetics & Genomics (AREA)
  • Medicinal Chemistry (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Public Health (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Photoreceptors In Electrophotography (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)

Abstract

LA PRESENTE INVENCION SE REFIERE A NUEVOS DERIVADOS DE 5-ACILO, 23-ACILO Y 5,23-DIACILO DE LOS COMPUESTOS LL-F28249. ESTOS COMPUESTOS LL-F28249 (COLECTIVAMENTE) SON AISLADOS DEL CALDO DE FERMENTACION DE STREPTOMYCES CYNEOGRISEUS SUBESPECIE NONCYANOGENUS QUE TIENE EL NUMERO DE ACCESO DE DEPOSITO NRRL15773. LOS PRESENTES COMPUESTOS DE 5-ACILO Y 5,23-DIACILO SE PREPARAN POR ACILACION SELECTIVA USANDO CLORUROS O ANH/IDRIDOS ACIDOS EN PRESENCIA DE 4-DIMETILAMINOPIRIDINA. LOS COMPUESTOS 23-ACILO SE PREPARAN POR ACILACION SELECTIVA DE LOS COMPUESTOS 5-0-SILILADOS LL-F28249. ESTOS NUEVOS COMPUESTOS TIENEN POTENTE ACTIVIDAD ANTIHELMINTICA, INSECTICIDA, ECTOPARASITICIDA, NEMATICIDA Y ACARICIDA. TAMBIEN SE DESCRIBEN AQUI COMPOSICIONES QUE CONTIENEN ESTOS DERIVADOS DE LL-F28249.
ES87112277T 1986-09-12 1987-08-25 Nuevos derivados de mono- y di-acilos de compuestos ll-f28249. Expired - Lifetime ES2059333T3 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US06/907,281 US5149832A (en) 1986-09-12 1986-09-12 Mono and diacyl derivatives of ll-f28249 compounds

Publications (1)

Publication Number Publication Date
ES2059333T3 true ES2059333T3 (es) 1994-11-16

Family

ID=25423825

Family Applications (1)

Application Number Title Priority Date Filing Date
ES87112277T Expired - Lifetime ES2059333T3 (es) 1986-09-12 1987-08-25 Nuevos derivados de mono- y di-acilos de compuestos ll-f28249.

Country Status (17)

Country Link
US (1) US5149832A (es)
EP (1) EP0259686B1 (es)
JP (1) JPS63132890A (es)
KR (1) KR880003948A (es)
AT (1) ATE96440T1 (es)
AU (1) AU593682B2 (es)
BR (1) BR8704737A (es)
CA (1) CA1317936C (es)
DE (1) DE3787942T2 (es)
DK (1) DK475487A (es)
ES (1) ES2059333T3 (es)
HU (1) HU199145B (es)
IE (1) IE62248B1 (es)
IL (1) IL83792A (es)
NZ (1) NZ221692A (es)
PT (1) PT85673B (es)
ZA (1) ZA876834B (es)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4806527A (en) * 1987-03-16 1989-02-21 Merck & Co., Inc. Avermectin derivatives
GB8721378D0 (en) * 1987-09-11 1987-10-21 Glaxo Group Ltd Chemical process
HU9203978D0 (en) * 1988-05-10 1993-04-28 American Cyanamid Co Method for producing macrolidic compounds and preparatives containing them qs active substance by means of fermentation
US6495591B1 (en) 1997-10-02 2002-12-17 Essential Therapeutics, Inc. Fungal efflux pump inhibitors
FR2948261B1 (fr) * 2009-07-22 2015-10-30 Sarl Herbarom Laboratoire Procede insecticide et/ou repulsif
CN104860961B (zh) * 2015-04-10 2017-08-04 新宇药业股份有限公司 一种制备5‑氧（对‑硝基苯甲酰）‑尼莫克汀的方法

Family Cites Families (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4201861A (en) * 1977-10-03 1980-05-06 Merck & Co., Inc. Acyl derivatives of C-076 compounds
PH16612A (en) * 1977-12-19 1983-11-28 Merck & Co Inc 13-halo and 13-deoxy derivatives of c-076 compounds
USRE32034E (en) * 1977-12-19 1985-11-19 Merck & Co., Inc. 13-Halo and 13-deoxy derivatives of C-076 compounds
JPS57120589A (en) * 1981-01-20 1982-07-27 Sankyo Co Ltd 5-methoxy and 5-lower alkanoyloxy derivative, its preparation and acaricide and parasiticide
PT80577B (pt) * 1984-06-05 1987-09-18 American Cyanamid Co Processo para a producao de novos agentes macrolidos ll-f28249 uteis no tratamento de infeccoes helminticas por ectoparasitas artropodes e por acarideos
GB2166436B (en) * 1984-09-14 1989-05-24 Glaxo Group Ltd Antibiotic compounds and their preparation
IL78621A (en) * 1985-04-30 1991-06-30 American Cyanamid Co Mylbemycin analogs,their preparation and pesticidal compositions containing them
ES8800986A1 (es) * 1985-07-27 1987-12-01 Pfizer Un procedimiento para la produccion de un nuevo derivado de avermectina
CA1316915C (en) * 1985-09-13 1993-04-27 American Cyanamid Company Macrolide antibiotics and their preparation

Also Published As

Publication number Publication date
DK475487D0 (da) 1987-09-11
KR880003948A (ko) 1988-05-31
ATE96440T1 (de) 1993-11-15
IL83792A (en) 1993-02-21
EP0259686A1 (en) 1988-03-16
HUT45535A (en) 1988-07-28
PT85673A (en) 1987-10-01
CA1317936C (en) 1993-05-18
ZA876834B (en) 1988-03-15
DK475487A (da) 1988-03-13
DE3787942T2 (de) 1994-05-11
US5149832A (en) 1992-09-22
HU199145B (en) 1990-01-29
AU593682B2 (en) 1990-02-15
IE62248B1 (en) 1995-01-11
BR8704737A (pt) 1988-05-03
PT85673B (pt) 1990-05-31
IE872433L (en) 1988-03-12
AU7827987A (en) 1988-03-17
JPS63132890A (ja) 1988-06-04
EP0259686B1 (en) 1993-10-27
NZ221692A (en) 1990-09-26
DE3787942D1 (de) 1993-12-02

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