ES2051773T3 - Procedimiento para la obtencion de aralquil-4h,1,2,4-triazil derivados. - Google Patents

Procedimiento para la obtencion de aralquil-4h,1,2,4-triazil derivados.

Info

Publication number
ES2051773T3
ES2051773T3 ES87810579T ES87810579T ES2051773T3 ES 2051773 T3 ES2051773 T3 ES 2051773T3 ES 87810579 T ES87810579 T ES 87810579T ES 87810579 T ES87810579 T ES 87810579T ES 2051773 T3 ES2051773 T3 ES 2051773T3
Authority
ES
Spain
Prior art keywords
lower alkyl
derivatives
aralquil
triazil
procedure
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Lifetime
Application number
ES87810579T
Other languages
English (en)
Inventor
Hans Allgeier
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Novartis AG
Original Assignee
Ciba Geigy AG
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Ciba Geigy AG filed Critical Ciba Geigy AG
Application granted granted Critical
Publication of ES2051773T3 publication Critical patent/ES2051773T3/es
Anticipated expiration legal-status Critical
Expired - Lifetime legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D249/00—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms
    • C07D249/02—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms not condensed with other rings
    • C07D249/08—1,2,4-Triazoles; Hydrogenated 1,2,4-triazoles
    • C07D249/10—1,2,4-Triazoles; Hydrogenated 1,2,4-triazoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/08—Antiepileptics; Anticonvulsants

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Engineering & Computer Science (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Pain & Pain Management (AREA)
  • Animal Behavior & Ethology (AREA)
  • Biomedical Technology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Control Of High-Frequency Heating Circuits (AREA)
  • Soft Magnetic Materials (AREA)
  • General Induction Heating (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Paints Or Removers (AREA)

Abstract

LA INVENCION SE REFIERE A ARALQUIL-4H-1,2,4TRIAZOLDERIVADOS, EN ESPEFCIL 5-FENILALQUILINFERIOR-4H1,2,4-TRIAZOL-3-CARBOXAMIDAS DE FORMULA (I) DONDE PH ES FENILO SUSTITUIDO POR ALQUILO INFERIOR, HALOGENO Y/O TRIFLUORMETILO, ALK ES ALQUILO INFERIOR, R1 ES HIDROGENO O ALQUILO INFERIOR Y R2 ES CARBAMILO SUSTITUIDO POR ALQUILO INFERIOR O ALCANOILO INFERIOR, Y SUS SALES, ASI COMO, SI ES CASO, SUS TAUTOMEROS, Y SUS SALES. ESTOS COMPUESTYOS PUEDEN APLICARSE COMO PRODUCTOS FARMACEUTICOS.
ES87810579T 1986-10-09 1987-10-07 Procedimiento para la obtencion de aralquil-4h,1,2,4-triazil derivados. Expired - Lifetime ES2051773T3 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
CH403586 1986-10-09

Publications (1)

Publication Number Publication Date
ES2051773T3 true ES2051773T3 (es) 1994-07-01

Family

ID=4268591

Family Applications (1)

Application Number Title Priority Date Filing Date
ES87810579T Expired - Lifetime ES2051773T3 (es) 1986-10-09 1987-10-07 Procedimiento para la obtencion de aralquil-4h,1,2,4-triazil derivados.

Country Status (19)

Country Link
US (2) US5045556A (es)
EP (1) EP0267147B1 (es)
JP (1) JPS6396176A (es)
KR (1) KR880005103A (es)
AT (1) ATE65996T1 (es)
AU (1) AU614722B2 (es)
DD (1) DD271518A5 (es)
DE (1) DE3772006D1 (es)
DK (1) DK526887A (es)
ES (1) ES2051773T3 (es)
FI (1) FI874413A (es)
GR (1) GR3002443T3 (es)
HU (1) HU200756B (es)
IL (1) IL84093A (es)
NO (1) NO166179C (es)
NZ (1) NZ222078A (es)
PH (1) PH24571A (es)
PT (1) PT85873B (es)
ZA (1) ZA877562B (es)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IL84093A (en) * 1986-10-09 1992-09-06 Ciba Geigy Ag Aralkyl-4h-1,2,4-triazole derivatives,their preparation and pharmaceutical compositions containing them
KR101214665B1 (ko) * 2004-09-16 2012-12-21 아스텔라스세이야쿠 가부시키가이샤 트리아졸 유도체 또는 그의 염
PL2298747T3 (pl) * 2008-07-03 2017-05-31 Astellas Pharma Inc. Pochodne triazolowe lub ich sole

Family Cites Families (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR1512421A (fr) * 1966-12-22 1968-02-09 Bellon Labor Sa Roger Amides d'acides triazole-1, 2, 4 carboxyliques-5
US4209516A (en) * 1974-01-14 1980-06-24 Ciba-Geigy Corporation Triazole derivatives
CH601268A5 (en) * 1974-06-14 1978-06-30 Ciba Geigy Ag 1-(2-Benzoylphenyl)-5-aminomethyl-1,2,4-triazole-3-carboxylic acids
US4209515A (en) * 1974-06-14 1980-06-24 Ciba-Geigy Corporation Triazole derivatives
JPS5258922A (en) * 1975-11-10 1977-05-14 Fuji Photo Film Co Ltd Photographic coupler
EP0034481B1 (en) * 1980-02-14 1984-05-30 Grigg, Ronald Ernest 2-methyl-5-thiazole-methylamine and carboxamide derivatives
US4789680A (en) * 1982-12-23 1988-12-06 Ciba-Geigy Corporation Aralkyltriazole compounds
JPS59199681A (ja) * 1983-04-26 1984-11-12 Ube Ind Ltd １，２，４−トリアゾ−ル−３−カルボン酸アミド類の製造法
JPS59206368A (ja) * 1983-05-10 1984-11-22 Ube Ind Ltd １，２，４−トリアゾ−ル−３−カルボン酸アミド類の製法
EP0129509B1 (de) * 1983-06-06 1989-08-23 Ciba-Geigy Ag Triazol(2,3-c)(1,3)benzodiazepine, Verfahren zu ihrer Herstellung, pharmazeutische Präparate enthaltend diese Verbindungen, sowie ihre therapeutische Verwendung
DE3525205A1 (de) * 1984-09-11 1986-03-20 Hoechst Ag, 6230 Frankfurt Pflanzenschuetzende mittel auf basis von 1,2,4-triazolderivaten sowie neue derivate des 1,2,4-triazols
MY100938A (en) * 1986-06-06 1991-05-31 Ciba Geigy Ag Arylkylimidazole derivatives.
IL84093A (en) * 1986-10-09 1992-09-06 Ciba Geigy Ag Aralkyl-4h-1,2,4-triazole derivatives,their preparation and pharmaceutical compositions containing them

Also Published As

Publication number Publication date
HUT47256A (en) 1989-02-28
FI874413A0 (fi) 1987-10-07
ATE65996T1 (de) 1991-08-15
DK526887A (da) 1988-04-10
KR880005103A (ko) 1988-06-28
EP0267147B1 (de) 1991-08-07
JPS6396176A (ja) 1988-04-27
NO874211D0 (no) 1987-10-08
NO166179C (no) 1991-06-12
AU7946187A (en) 1988-04-14
DK526887D0 (da) 1987-10-08
IL84093A0 (en) 1988-03-31
US5045556A (en) 1991-09-03
FI874413A (fi) 1988-04-10
PT85873B (pt) 1990-07-31
IL84093A (en) 1992-09-06
GR3002443T3 (en) 1992-12-30
US5098922A (en) 1992-03-24
NZ222078A (en) 1990-07-26
EP0267147A1 (de) 1988-05-11
HU200756B (en) 1990-08-28
ZA877562B (en) 1988-04-11
DD271518A5 (de) 1989-09-06
PH24571A (en) 1990-08-03
PT85873A (de) 1987-11-01
DE3772006D1 (de) 1991-09-12
NO874211L (no) 1988-04-11
NO166179B (no) 1991-03-04
AU614722B2 (en) 1991-09-12

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